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N-[3-(1H-imidazol-1-yl)propyl]-2-(1H-pyrazole-3-carbonyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
1-methyl-4-[2-(propan-2-yl)pyrimidin-4-yl]-3-(pyridin-3-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-[1-(2,3-dihydro-1H-inden-2-yl)-5-oxopyrrolidin-3-yl]-3-phenoxypropanamide
(3-{2-[1-(3-fluoropyridine-4-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}propyl)dimethylamine
5-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-N-(2-hydroxyethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
2-(1-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}piperidin-4-yl)-N-methylacetamide
2-amino-4-(1-ethyl-5-methyl-1H-pyrazol-4-yl)-6-(4-hydroxyphenyl)-5-methylpyridine-3-carbonitrile
3-[2-(1-cyclopentylpiperidin-4-yl)ethyl]-8-(trifluoromethyl)-3,4-dihydroquinazolin-4-one
2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-1-[(3R,4S)-3-amino-4-(4-methoxyphenyl)pyrrolidin-1-yl]ethan-1-one
(1S,5R)-6-benzyl-3-(2-hydroxy-4-methoxybenzoyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(cyclopentylmethyl)-4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
[(3R,4R)-1-[(4-phenylphenyl)methyl]-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
N-[(3,4-difluorophenyl)methyl]-3-{1-[2-(6-methylpyridin-2-yl)ethyl]piperidin-3-yl}propanamide
2-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]phenoxymethyl}pyridine
N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}-2,3-dihydro-1,4-benzodioxine-6-carboxamide
{1-[(2,4-diethoxy-3-methylphenyl)methyl]pyrrolidin-3-yl}methanamine
3-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[1-(5-methyl-1,3,4-oxadiazol-2-yl)ethyl]benzamide
1-{5-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]thiophen-2-yl}ethan-1-one
(2S,4S)-1-[(2-chlorophenyl)methyl]-N-ethyl-4-({[4-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
1-(4-{[4-(quinoline-6-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}piperazin-1-yl)ethan-1-one
4-[2-(dimethylamino)ethyl]-N-[4-methyl-3-(2-oxopyrrolidin-1-yl)phenyl]piperazine-1-carboxamide
N-[1-(3,4-dimethyl-5-sulfamoylbenzoyl)piperidin-3-yl]acetamide
2-[5-benzyl-1-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]-1,2,3,4-tetrahydroisoquinoline
[2-(3-methoxyphenyl)-1-[1-(1-methylcyclohexanecarbonyl)piperidin-4-yl]ethyl](methyl)(pyridin-2-ylmethyl)amine
2-(3,5-difluorophenyl)-N-[2-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]acetamide
(2R,3R)-3-(morpholin-4-yl)-1'-(pyridin-3-ylmethyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
(2S,4R)-4-amino-N,N-diethyl-1-[6-ethyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]pyrrolidine-2-carboxamide
methyl 3-(3-methylbutyl)-7-oxo-9-(3-phenylpropoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-(1,4-dioxan-2-ylmethyl)-5,6-dimethoxy-1,2-dihydroisoquinolin-1-one
methyl 4-(5-{[methyl(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)amino]methyl}-1,2,4-oxadiazol-3-yl)benzoate
N-{[4-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
5-[1-(1-methylpiperidin-4-yl)-3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]-1,2-dihydropyridin-2-one
3-(1H-1,3-benzodiazol-2-yl)-1-[2-(2-phenylethyl)morpholin-4-yl]propan-1-one
3-(3-ethynylbenzoyl)-9-methoxy-7-oxo-N-(thiophen-3-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-4-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}piperazine
4-(1H-indol-3-ylmethyl)-6-[(5-methyl-1,2,4-oxadiazol-3-yl)methoxy]-1-(propan-2-yl)-1,4-diazepan-2-one
ethyl 3-benzyl-1-[(1,5-dimethyl-3-oxo-2-phenyl-2,3-dihydro-1H-pyrazol-4-yl)methyl]piperidine-3-carboxylate
3-methyl-N-{5-[(2-methylphenyl)methyl]-1,3,4-thiadiazol-2-yl}-1-propyl-1H-pyrazole-4-carboxamide
2-methyl-4-phenyl-N-[2-(pyrrolidin-1-yl)ethyl]pyrimidine-5-carboxamide
1-(3-chloro-4-propoxyphenyl)-3-cyclopropyl-3-[(1-methyl-1H-imidazol-2-yl)methyl]urea
N-(2-methoxyethyl)-2-(pyrrolidin-3-yl)-N-(1,3-thiazol-2-ylmethyl)benzamide
(1S,5R)-N,N-dimethyl-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane-6-sulfonamide
5-(naphthalen-1-ylmethyl)-5-{3-oxo-3-[2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]propyl}pyrrolidin-2-one
2-acetamido-3-hydroxy-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}propanamide
1-{2-[4-(4-methanesulfonylphenyl)phenoxy]ethyl}pyrrolidine
N-[2-(5-chloro-2-methyl-1H-indol-3-yl)ethyl]-2-(ethylamino)pyrimidine-5-carboxamide
1-{4-[3-(4-fluorophenoxy)propyl]piperazin-1-yl}-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]({[2-(2-methylphenoxy)pyridin-3-yl]methyl})amine
(3R,5S)-N3-[3-(furan-2-yl)propyl]-N5-(6-methylpyridin-3-yl)piperidine-3,5-dicarboxamide
N-(2-{7-[(2,4-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)furan-2-carboxamide