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2-(4-{2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperazin-1-yl)-N-(propan-2-yl)acetamide
N-[(5-chlorothiophen-2-yl)methyl]-1-methyl-3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-(1H-indazol-1-yl)-1-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}ethan-1-one
2-[4-(1-benzothiophen-3-yl)-2-(morpholin-4-ylmethyl)phenoxy]-N-(furan-2-ylmethyl)acetamide
3-{[1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]carbamoyl}pyridin-1-ium-1-olate
N-[1-(butan-2-yl)-1H-pyrazol-5-yl]-2-(3-cyclopropanecarbonyl-1H-indol-1-yl)acetamide
(2R,3R,6R)-3-(4-methoxyphenyl)-5-[(6-methylpyridin-2-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
{3-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]-9-cyclopentyl-3,9-diazaspiro[5.5]undecan-1-yl}methanol
1-[2-(4-chlorophenyl)ethyl]-N-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-N-methyl-6-oxopiperidine-3-carboxamide
(3S,4S)-4-cyclopropyl-1-[(2-fluoro-4,5-dimethoxyphenyl)methyl]pyrrolidine-3-carboxylic acid
8-cyclopentyl-3-methyl-1-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(1H-indazol-5-yl)-4-{[methyl(pyrazin-2-ylmethyl)amino]methyl}benzamide
N-cyclohexyl-N-[2-(ethylsulfanyl)ethyl]-4-hydroxy-2-(pyridin-2-yl)pyrimidine-5-carboxamide
4-[4-(3-methoxyphenyl)-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]-1-[(5-methylthiophen-2-yl)methyl]piperidine
4-{2-[4-(pentan-2-yl)-1H-1,2,3-triazol-1-yl]ethyl}benzene-1-sulfonamide
6-{[(1S,2R)-2-hydroxycyclopentyl]amino}-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}pyridine-3-carboxamide
1-(4-ethyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)-3-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}urea
2-[1-(2H-1,3-benzodioxol-5-ylmethyl)-2,5-dioxo-3-phenylpyrrolidin-3-yl]-N-benzyl-N-ethylacetamide
3-{4-[6-amino-5-cyano-4-(5-methylfuran-2-yl)pyridin-2-yl]-3,5-dimethyl-1H-pyrazol-1-yl}butanoic acid
(2S)-2-amino-1-(4-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-3-hydroxypropan-1-one
3-{3-[2-(2-fluorophenyl)ethyl]piperidine-1-carbonyl}-1,5,6-trimethyl-1,2-dihydropyridin-2-one
3-cyclohexyl-1-[3-(morpholine-4-carbonyl)-1-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propan-1-one
N-[(2-chloro-4-fluorophenyl)methyl]-N-ethyloxan-4-amine
(3R,4R)-4-(hydroxymethyl)-1-(5-methyl-2-phenyl-1H-imidazole-4-carbonyl)piperidin-3-ol
6-{3-[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidin-1-yl]-3-oxopropyl}-2,3-dihydropyridazin-3-one
{3-[(2-methylphenyl)methyl]-1-[5-(propan-2-yl)pyrimidin-4-yl]piperidin-3-yl}methanol
N-[(1-methylpiperidin-3-yl)methyl]-N-(2-phenylethyl)cyclopent-1-ene-1-carboxamide
methyl 9-[2-(2-fluorophenyl)ethoxy]-7-oxo-3-[2-(thiophen-3-yl)acetyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-methyl-N-[3-(4-methylpiperazin-1-yl)propyl]-4-phenylpyridine-3-carboxamide
4-(hydroxymethyl)-1-{5-methylimidazo[1,2-a]pyridine-2-carbonyl}azepan-4-ol
(4aR,6R,8aS)-2-(2,1,3-benzoxadiazol-4-ylmethyl)-8a-(methoxymethyl)-6-(morpholin-4-yl)-decahydroisoquinoline
5,5-dimethyl-3-{2-[2-(5-methyl-1,2-oxazol-3-yl)piperidin-1-yl]-2-oxoethyl}-1,3-oxazolidine-2,4-dione
{[3-(2-chlorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amine
(4aR,7aS)-1-(2-hydroxyethyl)-4-(1-methyl-1H-1,3-benzodiazole-5-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-6-oxo-2-(propan-2-yl)-1,6-dihydropyrimidine-5-carboxamide
N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N,3-dimethyl-4,5-dihydro-1,2-oxazole-5-carboxamide
N2-benzyl-6-[3-(methylsulfanyl)phenyl]-1,3,5-triazine-2,4-diamine
{[1-(3-fluorophenyl)-3-(5-methylfuran-2-yl)-1H-pyrazol-4-yl]methyl}[2-(furan-2-yl)ethyl]amine
9-methoxy-7-(4-methoxyphenyl)-4-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl](2-methoxyethyl)[(4-methylphenyl)methyl]amine
2,3,5-trimethyl-N-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
N-{4-[5-(trifluoromethyl)pyridin-2-yl]-1H-pyrrolo[2,3-b]pyridin-6-yl}piperidin-4-amine
N-(cyclopropylmethyl)-4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}-N-propylbenzamide
2-{[4-(1-tert-butyl-1H-pyrazol-4-yl)-1,2,3,6-tetrahydropyridin-1-yl]methyl}-7-chloro-4H-pyrido[1,2-a]pyrimidin-4-one
2-(3-methoxyphenyl)-5-(thiophene-3-carbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
1-[(3S,4R)-1-(6-cyanopyridine-3-carbonyl)-4-(propan-2-yl)pyrrolidin-3-yl]-3,3-dimethylurea
(4S,6R)-4-[4-(4-benzyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-6-methyl-1,3-diazinane-2-thione
(1R,5S)-6-(5-methyl-2-{[1-(pyridin-4-ylmethyl)piperidin-4-yl]oxy}benzoyl)-6-azabicyclo[3.2.1]octane
N3-(1H-1,3-benzodiazol-2-ylmethyl)-N5-cycloheptyl-1-cyclopropyl-N3-methyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
2-({2-[1-(2-methoxyethyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)-5-methylpyrazine