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N-[2-(N-methylmethanesulfonamido)ethyl]-1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
1-(4,4-difluoropiperidin-1-yl)-2-(naphthalen-2-yloxy)propan-1-one
(2-methoxyethyl)(1-{1-[(2-methoxyphenyl)methyl]piperidin-4-yl}-2-phenylethyl)(pyridin-3-ylmethyl)amine
N-{[7-(6-methoxypyridazin-3-yl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-methylpentanamide
(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)({[8-methyl-2-(thiophen-2-yl)quinolin-3-yl]methyl})amine
N-benzyl-2-[2,5-dioxo-3-phenyl-1-(thiophen-2-ylmethyl)pyrrolidin-3-yl]-N-(2-hydroxyethyl)acetamide
9-[2-(4-fluoro-2-methylphenyl)acetyl]-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
(2S)-2-{[5-(2-methoxyacetamido)-1-(2-phenylethyl)-1H-1,3-benzodiazol-7-yl]formamido}propanamide
(3R,4R)-4-{methyl[2-(pyridin-2-yl)ethyl]amino}-1-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidin-3-ol
(1S,5R)-3-{2,6-dimethylimidazo[1,2-a]pyridine-3-carbonyl}-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
5-{6-oxa-9-azaspiro[4.5]decane-9-carbonyl}-2-(pyridin-3-yl)pyrimidin-4-ol
2,4-dimethoxy-6-(1H-pyrazol-3-yl)pyrimidine
3-(2H-1,3-benzodioxole-5-carbonyl)-1-{[3-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperidine
2-({[6-(pyrrolidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}(thiophen-2-ylmethyl)amino)ethan-1-ol
3-methyl-6-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]pyridazine
5-(3,4-difluorophenoxymethyl)-N-[(1R)-1-(3-methoxyphenyl)ethyl]-1,2-oxazole-3-carboxamide
8-butanoyl-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(3S,4S)-4-cyclopropyl-1-[2-(3,4-dimethoxyphenyl)acetyl]pyrrolidine-3-carboxylic acid
2-[4-(3-chlorophenyl)piperazin-1-yl]-N-ethylpyridine-3-carboxamide
6-oxo-1-(pyridin-2-ylmethyl)-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]piperidine-3-carboxamide
1-(oxolan-2-ylmethyl)-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
N-benzyl-N-ethyl-3-[(4-methoxyphenyl)methyl]-1,2-oxazole-5-carboxamide
2-(1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}piperidin-3-yl)-1,3-benzoxazole
7-(3,5-dimethyl-4,5-dihydro-1,2-oxazole-5-carbonyl)-2,3-dimethyl-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
ethyl 4-[1-(3-phenylpropyl)-1H-1,2,3-triazole-4-amido]piperidine-1-carboxylate
N-ethyl-6-({1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}amino)pyridine-3-carboxamide
2-(2,5-dimethoxyphenyl)-N-{[5-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
3-(1-methyl-1H-pyrazol-4-yl)-1-[4-(3-phenylpropyl)-1,4-diazepan-1-yl]propan-1-one
2-[(4S,6R)-6-methyl-2-sulfanylidene-1,3-diazinan-4-yl]-N-[2-(4-methylphenyl)propan-2-yl]acetamide
4-methoxy-N-[(2R,3R)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-3-methylbenzamide
2,4,5-trimethyl-6-[3-(piperidin-1-yl)azetidin-1-yl]pyrimidine
(3R,5S)-N-[2-(1-methylpyrrolidin-2-yl)ethyl]-1-(pyridin-4-ylmethyl)-5-[3-(trifluoromethyl)phenoxymethyl]piperidine-3-carboxamide
1-[2-(2-butyl-4-methyl-3-oxopiperazin-1-yl)-2-oxoethyl]-2-methyl-1,4-dihydroquinolin-4-one
3-[4-(1H-imidazol-2-yl)piperidine-1-carbonyl]piperidine-1-carboxamide
(1R,5S)-6-({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl)-6-azabicyclo[3.2.1]octane
3-[2-(4-chlorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-1-methylpiperidine
1-[(3,5-dimethoxyphenyl)methyl]-4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidine
(3aR,7aS)-2-[4-(4H-1,2,4-triazol-4-yl)benzoyl]-2,3,3a,4,7,7a-hexahydro-1H-isoindole
2-(pyridin-3-yl)-N-[3-(1H-1,2,4-triazol-1-yl)propyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
4-benzyl-3-ethyl-1-(4,4,4-trifluorobutyl)-1,4-diazepan-5-one
N-(2-{7-[4-(2-fluorophenyl)benzoyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-4-methylbenzamide
N,7-dimethyl-N-[2-(1H-pyrazol-1-yl)ethyl]imidazo[1,2-a]pyridine-2-carboxamide
2-methoxy-1-{1-[3-(trifluoromethyl)phenyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}ethan-1-one
1-(cyclopropylmethyl)-4-({1-[(2-fluorophenyl)methyl]-2-methanesulfonyl-1H-imidazol-5-yl}methyl)piperazine
1-{3-cyclobutyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-3-(1,2-oxazinan-2-yl)propan-1-one
1-(5-chloro-2-methylphenyl)-4-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]piperazine
1-(4-ethenylbenzoyl)-N-phenylpiperidin-3-amine
1-(3-chlorophenyl)-4-[1-(1,4-dithiepan-6-yl)piperidin-3-yl]piperazine
4-(3-{[1-(thiophene-2-carbonyl)piperidin-4-yl]oxy}benzoyl)morpholine
(5S,9aS,9bS)-5-(1-ethyl-1H-imidazol-2-yl)-2-methyl-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one