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N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-3-(2-oxoazepan-1-yl)propanamide
1-[(3R,4R)-3-(hydroxymethyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]-4-(2-methyl-1H-imidazol-1-yl)butan-1-one
1-[3-hydroxy-2-(thiophen-3-ylmethyl)propyl]-3-(2-methyl-2H-1,2,3-benzotriazol-4-yl)urea
5-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]-N-(oxolan-2-ylmethyl)-N-propylpyridin-2-amine
N-[1-(7-{[4-(propan-2-yl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]cyclopropanecarboxamide
N-(2-hydroxyethyl)-3-{5-[2-(2-oxopyrrolidin-1-yl)ethyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
N-{[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-(2-hydroxyethyl)-N-{[4-(methylsulfanyl)phenyl]methyl}isoquinoline-1-carboxamide
(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]methylamine
3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-[2,2,2-trifluoro-1-(furan-2-yl)ethyl]propanamide
4-[3-(2,3-dimethoxyphenyl)pyrrolidine-1-carbonyl]-1-(2-phenylethyl)-1H-1,2,3-triazole
1-[(3R,4R)-3-{[ethyl(2-hydroxyethyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-3-methylbut-2-en-1-one
3-{[5-(1,5-dimethyl-1H-pyrazol-4-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-5-(furan-2-yl)-1,2,4-oxadiazole
2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}-1-{spiro[indene-1,4'-piperidine]-1'-yl}ethan-1-one
2-(1,1-dioxo-1λ6-thiolan-3-yl)-N-[2-(2-ethoxyphenoxy)ethyl]-N-methylacetamide
N-[(2-benzyl-1,3-thiazol-4-yl)methyl]-3,6-dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
6-(2,5-dimethylphenyl)-N-methyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
4-ethyl-5-[4-(2-methylphenoxy)piperidine-1-carbonyl]-1,3-thiazol-2-amine
N-cyclopropyl-1-[(1s,4s)-4-(2-cyclohexylacetamido)cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
10-(4-phenylpiperazine-1-carbonyl)-1-azatricyclo[6.3.1.04,12]dodeca-4(12),5,7,10-tetraen-9-one
6-(benzyloxy)-4-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetyl}-1-(pyridin-3-ylmethyl)-1,4-diazepan-2-one
6-[(diethylamino)methyl]-N-[1-(pyridin-3-yl)propyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
4-{1-[(dimethyl-1,2-oxazol-4-yl)methyl]piperidin-3-yl}benzoic acid
2-[4-(4-{[(3-fluorophenyl)methyl]amino}piperidin-1-yl)phenyl]-N-[2-(2-methoxyphenyl)ethyl]acetamide
[4-(2-methoxy-5-methylphenyl)-4H-1,2,4-triazol-3-yl](phenyl)methanol
N-[2-(2-methoxyphenyl)ethyl]-2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
2-(adamantan-1-yl)-N-[(6-hydroxypyrimidin-4-yl)methyl]acetamide
N-{5H,6H,7H,8H,9H,10H-cyclohepta[b]indol-2-ylmethyl}-3-(1,2-oxazolidin-2-yl)propanamide
3-(4-hydroxyphenyl)-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]benzamide
N5-butyl-1-(cyclohexylmethyl)-N3,N3-dimethyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
2-butyl-8-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
N-[1-(furan-2-carbonyl)piperidin-3-yl]-3-(1H-pyrazol-4-yl)benzamide
2-methyl-2-(2-{methyl[(5-methyl-1,2-oxazol-3-yl)methyl]amino}-4-(morpholin-4-yl)pyrimidin-5-yl)propanoic acid
4-{[3-(6-methoxypyrimidin-4-yl)phenyl]methyl}morpholine
5-fluoro-2-[1-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)pyrrolidin-2-yl]-1H-1,3-benzodiazole
N4-(1,2-oxazol-3-ylmethyl)-7-(1H-pyrrole-2-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
N-{2-[(4-methyl-1,2,3-thiadiazol-5-yl)sulfanyl]ethyl}-6-(piperidin-3-yl)pyrimidin-4-amine
1-cyclopentyl-4-{[1-(3-methylbutyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl}piperazine
4-(2-cyclopropylacetyl)-6-[(3-methoxyphenyl)methoxy]-1-(2-phenylethyl)-1,4-diazepan-2-one
ethyl 4-[({[2-(dimethylamino)pyridin-3-yl]methyl}amino)methyl]-1H-pyrazole-3-carboxylate
1-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)-4-(pyrrolidine-1-carbonyl)-1,4-diazepan-6-ol
3-chloro-N-[3-(4-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}phenoxy)propyl]benzene-1-sulfonamide
4-[(2-amino-5,6,7,8-tetrahydroquinazolin-4-yl)amino]-1-(2-methoxyphenyl)pyrrolidin-2-one
5-butyl-1'-[(1-propyl-1H-imidazol-2-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-[3-(1-methyl-1H-pyrazol-4-yl)propanoyl]piperidine-4-carboxamide
[(6-chloropyridin-3-yl)methyl][(4-methanesulfonylphenyl)methyl]methylamine
1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-N,5-dimethyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-1H-pyrazole-4-carboxamide
N-(4-fluoro-2-methylphenyl)-2-[(1-methyl-4,5,6,7-tetrahydro-1H-indazol-3-yl)formamido]propanamide
2-{[(4aR,8aR)-4a-hydroxy-7-(2-methoxyacetyl)-decahydro-2,7-naphthyridin-2-yl]methyl}-6-methyl-4H-pyrido[1,2-a]pyrimidin-4-one
methyl 7-oxo-9-[2-(pyridin-2-yl)ethoxy]-3-(thiophene-2-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate