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N-(2-methoxy-5-methylphenyl)-2-[(4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-yl)formamido]acetamide
{3-[(2-fluorophenyl)methyl]-1-[(3-methoxyphenyl)methyl]piperidin-3-yl}methanol
(1-{6-amino-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-3-(2-phenylethyl)piperidin-3-yl)methanol
5-{1-[(3-chloro-4-hydroxyphenyl)methyl]piperidin-4-yl}-5-(2-methylpropyl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
N-(2-methoxyethyl)-N-[(5-methylthiophen-2-yl)methyl]-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide
1-(2-methoxyethyl)-4-oxo-N3-(3-phenylpropyl)-N5-[1-(thiophen-2-yl)propyl]-1,4-dihydropyridine-3,5-dicarboxamide
(1S,5R)-3-[2-(2-fluorophenyl)benzoyl]-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(2-chlorophenyl)-3-methyl-N-(oxan-4-ylmethyl)-3H-imidazo[4,5-b]pyridine-6-carboxamide
N-methyl-4-(piperidin-3-yl)-N-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}benzamide
methyl 3-[(4-fluoro-3-methoxyphenyl)methyl]-7-oxo-9-[2-(thiophen-3-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
4-methyl-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-2-(propan-2-yl)-N-(pyridin-3-ylmethyl)-1,3-thiazole-5-carboxamide
N-(2-hydroxybutyl)-5-methyl-4-{[(4-phenyloxan-4-yl)methyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-2-(2,3,6-trimethylphenoxy)acetamide
2-methyl-8-(3,3,3-trifluoropropanesulfonyl)-2,8-diazaspiro[4.5]decane
4-[4-(4-ethyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-1-(2-methylpropyl)pyrrolidin-2-one
methyl({[6-(4-methyl-1,4-diazepane-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl})({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)amine
(4aR,7aS)-1-benzyl-4-(1-methylcyclopropanecarbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[4-(2-methylphenyl)-1,4-diazepan-1-yl]-3-(methylsulfanyl)propan-1-one
N-methyl-3-[(3S,4R)-4-(morpholin-4-yl)-1-(naphthalen-1-ylmethyl)piperidin-3-yl]propanamide
N-{[5-fluoro-7-(6-methoxypyridazin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(1H-indol-3-yl)propanamide
9-(cyclopropanesulfonyl)-2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
2-({2-[1-(2,3-difluorobenzoyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
3-(3-amino-4-phenyl-1H-pyrazol-1-yl)-5-[(propan-2-yl)sulfamoyl]benzoic acid
1-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-4-(7-methoxy-2H-1,3-benzodioxol-5-yl)-1H-1,2,3-triazole
N-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-N-ethyl-2,3-difluorobenzamide
ethyl 3-[(3-methoxyphenyl)methyl]-1-[3-(morpholin-4-yl)propanoyl]piperidine-3-carboxylate
N-[2-(dimethylamino)ethyl]-5-[(4-methyl-1H-imidazol-5-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
1-(furan-2-ylmethyl)-3-(4-methoxy-3,5-dimethylbenzoyl)piperidine
5-[2-(cyclopropylmethyl)pyrimidin-4-yl]-2-ethoxybenzoic acid
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[5-(morpholin-4-yl)pentyl]acetamide
7-[(2,3-dimethoxyphenyl)methyl]-2-(2,5-dimethylfuran-3-carbonyl)-2,7-diazaspiro[4.5]decane
1-{[4-(hydroxymethyl)oxan-4-yl]methyl}-1-methyl-3-(2,4,6-trimethylphenyl)urea
N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
1-[(1S,5R)-6-(6-methoxy-2,3-dihydro-1H-indene-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
N-(3-methoxyphenyl)-3-{1-[(E)-2-phenylethenesulfonyl]piperidin-4-yl}propanamide
2-(4-{[4-ethoxy-3-(hydroxymethyl)phenyl]methyl}-1-[(4-methylphenyl)methyl]piperazin-2-yl)ethan-1-ol
N-[(2R,3R)-2-methoxy-1'-[(2E)-3-(pyridin-4-yl)prop-2-enoyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
N-[1-(2,5-difluorophenyl)cyclopropyl]-3-(2-hydroxyphenyl)-1H-pyrazole-5-carboxamide
N-(1-benzylpiperidin-4-yl)-3-(2-{[4-(methylsulfanyl)phenyl]methyl}-5-oxopyrrolidin-2-yl)propanamide
3-(3-hydroxy-3-methylbutyl)-N-[1-(6-methylpyridin-2-yl)ethyl]benzamide
2-hydroxy-5-methyl-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]benzamide
(2S)-N-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}-3-hydroxy-2-(methylamino)propanamide
3-(2-{4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-oxoethyl)imidazolidine-2,4-dione
N-[(3R,4S)-4-cyclopropyl-1-(2-methoxyacetyl)pyrrolidin-3-yl]-3-(2-ethyl-1H-imidazol-1-yl)propanamide
4-(4-benzoylpiperazin-1-yl)-2-[(2,3-dimethoxyphenyl)methyl]-2,3-dihydro-1H-isoindole-1,3-dione
(3S,4R)-1-[2-(dimethyl-1,3-thiazol-5-yl)acetyl]-4-(3-fluorophenyl)pyrrolidine-3-carboxylic acid
(4aS,7aR)-1-(2-methoxyethyl)-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2,3-difluoro-4-methyl-N-[2-(2-oxoimidazolidin-1-yl)ethyl]benzamide
6-methoxy-N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-3-methyl-1-benzofuran-2-carboxamide