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1-[2-(adamantan-1-yl)propan-2-yl]-3-(3-methyl-1,2,4-thiadiazol-5-yl)urea
6-cyclopentyl-2-methoxy-3-{[(thiolan-3-yl)amino]methyl}-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
1-[2-(6-fluoroquinolin-8-yl)pyrimidin-4-yl]pyrrolidin-3-ol
4-(1-butyl-1H-imidazol-2-yl)-1-(1-ethyl-5-methyl-1H-pyrazole-3-carbonyl)piperidine
N-[4-(1,3-benzoxazol-2-yl)phenyl]-1-(oxolan-3-ylmethyl)piperidine-4-carboxamide
(2R)-4-{5-[2-(ethylsulfanyl)pyrimidin-5-yl]-4-phenyl-1H-imidazol-1-yl}-2-methylbutan-1-ol
N-{1-[1-(3,4-dimethylbenzoyl)piperidin-4-yl]-2-(3-methoxyphenyl)ethyl}-N,3-dimethylbutanamide
N-[(1-cyclopentylpiperidin-4-yl)methyl]-4-(methylsulfanyl)-N-(pyridin-3-ylmethyl)benzamide
N-{1-[1-(cyclohex-1-ene-1-carbonyl)piperidin-4-yl]-2-(2-methylphenyl)ethyl}-N-methyl-2-(1H-pyrazol-1-yl)acetamide
4-methyl-5-(prop-2-en-1-yl)-6-(5,6,7,8-tetrahydro-1,6-naphthyridin-6-yl)pyrimidin-2-amine
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-7-(2-methoxyacetamido)-1-(2-phenylethyl)-1H-1,3-benzodiazole-5-carboxamide
4-{[(2-hydroxyethyl)[(2E)-3-phenylprop-2-en-1-yl]amino]methyl}-N-methylbenzene-1-sulfonamide
2-(2-fluorophenyl)-N-{[7-(6-methoxypyridazin-3-yl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
1-[(3R,4R)-3-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(pyridin-3-yl)ethan-1-one
4-(7-methyl-2,3-dihydro-1,4-benzodioxine-6-carbonyl)-2-(trifluoromethyl)morpholine
methyl[1-(pyridin-2-yl)ethyl]{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}amine
N,N-dimethyl-4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
1-[4-(pyridin-2-yl)piperazin-1-yl]-3-[1-(thian-4-yl)piperidin-3-yl]propan-1-one
4-hydroxy-N-[(1S,3S)-3-{[4-(pyridin-3-yl)pyrimidin-2-yl]amino}cyclopentyl]benzamide
N-[2-(3,4-dimethoxyphenyl)ethyl]-1-{1,3-dioxo-2-[1-(thiophen-2-yl)ethyl]-2,3-dihydro-1H-isoindol-4-yl}-N-methylpiperidine-3-carboxamide
6-{8-benzyl-2,8-diazaspiro[5.5]undecan-2-yl}pyrimidine-2,4-diamine
1-{3-[(4-methoxyphenyl)amino]piperidin-1-yl}-3-(1H-1,2,4-triazol-1-yl)propan-1-one
1-cyclopentyl-4-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-2-one
1-[cyclohexyl(methyl)amino]-3-(3-{[4-(prop-2-en-1-yl)piperazin-1-yl]methyl}phenoxy)propan-2-ol
(2S,4S,5R)-1,2-dimethyl-4-(morpholine-4-carbonyl)-5-phenylpyrrolidine-2-carboxylic acid
N-(pyridin-4-ylmethyl)-1-{[2-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
(3R,4R)-4-cyclobutyl-1-(2-methoxybenzenesulfonyl)-3-methylpiperidin-4-ol
5-(2,4-difluorophenoxymethyl)-N-methyl-N-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)-1,2-oxazole-3-carboxamide
1-[(2-chlorophenyl)methyl]-N-[5-(morpholin-4-yl)pentyl]-1H-1,2,3-triazole-4-carboxamide
2-amino-4-(3-phenyl-1H-pyrazol-4-yl)-6-propyl-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
2-[4-(3,5-dimethyl-1H-pyrazole-4-sulfonamido)-3,5-dimethyl-1H-pyrazol-1-yl]acetic acid
(3S,4R)-1-[(2-aminopyridin-3-yl)methyl]-4-(3-methoxyphenyl)pyrrolidine-3-carboxylic acid
3-({[1-(4-propyl-1,2,3-thiadiazole-5-carbonyl)piperidin-3-yl]oxy}methyl)pyridine
2-(2-{3-[benzyl(methyl)amino]piperidin-1-yl}-2-oxoethyl)-4-methyl-1,2-dihydrophthalazin-1-one
N-[(5-methyl-1,2-oxazol-3-yl)methyl]-6-oxo-1-(3-phenylpropyl)piperidine-3-carboxamide
1-[2-(1,3-thiazol-2-yl)ethyl]-3-[5-(thiophen-2-yl)-1,3,4-thiadiazol-2-yl]urea
N-[(2R,3R)-2-(pyridin-2-ylmethoxy)-1'-(thiophene-3-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
(butan-2-yl)[(4-methyl-1H-imidazol-5-yl)methyl](3-phenylprop-2-yn-1-yl)amine
N-cyclopropyl-4-{[(1-ethyl-1H-imidazol-5-yl)methyl]sulfamoyl}benzamide
2-(5-ethyl-1-benzofuran-3-yl)-1-[2-(pyrrolidine-1-carbonyl)piperazin-1-yl]ethan-1-one
1-(6-methylpyridazin-3-yl)-4-[(6-methylpyridin-3-yl)oxy]piperidine-4-carboxylic acid
N,N-diethyl-1-{1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]piperidin-4-yl}-1H-1,2,3-triazole-4-carboxamide
1-[(4-methoxy-3-methylphenyl)methyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N,N-dimethyl-3-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]aniline
N-ethyl-N-[2-(1H-pyrazol-1-yl)ethyl]-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-3-carboxamide
3-{[3-(3-chlorophenyl)-3-phenylpropanamido]methyl}-1,2,4-oxadiazole-5-carboxamide
4-{1-[4-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl}morpholine
(3S,4S)-1-(2-{[(2-chlorophenyl)methyl]carbamoyl}ethyl)-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
1-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidin-1-yl]-2-(1-methyl-1H-pyrrol-2-yl)ethane-1,2-dione
N-ethyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-[1-(3-methylbutyl)-3-oxopiperazin-2-yl]acetamide