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(3aS,6aR)-3-[2-(3-chlorophenyl)ethyl]-5-(5-methylpyrazine-2-carbonyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
9-[2-(hydroxymethyl)-1H-1,3-benzodiazole-5-carbonyl]-2-methyl-2,9-diazaspiro[5.5]undecan-3-one
1-(cyclohex-3-ene-1-carbonyl)-4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]piperidine
N-{[7-(3,6-dimethylpyrazin-2-yl)-4-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(pyridin-2-ylsulfanyl)acetamide
3-amino-1-[(6-acetamidoquinolin-2-yl)methyl]pyrrolidine-3-carboxylic acid
(2S)-2-(3-ethyl-1,2,4-oxadiazol-5-yl)-N-(2-methyl-5-sulfamoylphenyl)pyrrolidine-1-carboxamide
1-(benzyloxy)-8-[(3-chlorophenyl)methyl]-1,8-diazaspiro[4.5]decan-2-one
6-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine-8-carbonyl}imidazo[2,1-b][1,3]thiazole
9-methoxy-4-(2-phenylpropyl)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-({7-[4-(thiophen-2-yl)butanoyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)pyridine-4-carboxamide
(5S,9aS,9bS)-2-(pyridin-3-ylmethyl)-5-[2-(trifluoromethyl)phenyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
2,5-difluoro-N-{[8-(2-phenylacetyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}benzamide
N-benzyl-5-{[benzyl(methyl)amino]methyl}-N-methyl-1,2-oxazole-3-carboxamide
N-(dimethyl-1,2-oxazol-4-yl)-3-{[2-(3-methyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methyl}benzamide
4-(4-methylpyridine-3-carbonyl)-1-(2-phenylphenyl)piperazin-2-one
4-({[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]amino}methyl)benzene-1-sulfonamide
2-[1-ethyl-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-[(5-phenyl-1,2-oxazol-3-yl)methyl]acetamide
2-(dimethylamino)-N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-2-(3-methylphenyl)acetamide
N-cyclobutyl-4-[(4-methyl-1,4-diazepan-1-yl)sulfonyl]benzamide
3-(3-hydroxy-3-methylbutyl)-N-methyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}benzamide
3-{[1-(dimethylsulfamoyl)piperidin-4-yl]oxy}-N-(1-phenylethyl)benzamide
1-{4-[(3-fluorophenyl)methyl]-4-(hydroxymethyl)piperidin-1-yl}-3-(pyridin-3-yl)propan-1-one
N-[2-(pyridin-3-yl)-5,6,7,8-tetrahydroquinazolin-5-yl]propanamide
2-({5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)-1-(pyridin-3-yl)ethan-1-ol
2-[(6-{[(4-fluorophenyl)methyl](methyl)amino}pyridazin-3-yl)oxy]-1-[2-(pyridin-2-yl)piperidin-1-yl]ethan-1-one
3-[(4-methoxyphenyl)methyl]-N-[1-(trimethyl-1H-pyrazol-4-yl)ethyl]-1,2-oxazole-5-carboxamide
2-(2,3-dihydro-1H-inden-1-yl)-N-[2-oxo-2-(piperazin-1-yl)ethyl]acetamide
2-(dimethyl-1,3-thiazol-5-yl)-N-[(2S)-1-methoxypropan-2-yl]acetamide
N-{2-[4-(4-fluorophenyl)-5-{[(2-methylphenyl)methyl]sulfanyl}-4H-1,2,4-triazol-3-yl]ethyl}-3,5-dimethoxybenzamide
3-[(3S,4R)-1-[(3-chlorophenyl)methyl]-4-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-3-yl]-N-[(3-fluorophenyl)methyl]propanamide
2-amino-1-[(3R,4S)-3-{[2-(dimethylamino)-5,6-dimethylpyrimidin-4-yl]amino}-4-(propan-2-yl)pyrrolidin-1-yl]ethan-1-one
methyl 4-[3-(2H-1,3-benzodioxole-5-carbonyl)piperidin-1-yl]-4-oxobutanoate
8-(cyclopropylmethyl)-N-(2-methoxyphenyl)-9-oxo-2,8-diazaspiro[5.5]undecane-2-carboxamide
(1S,5R)-N-[2-(2-fluorophenyl)ethyl]-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
N-(4-chlorophenyl)-6-hydroxy-1,4-oxazepane-4-carboxamide
N-{2-[3-(2-methylphenyl)pyrrolidin-1-yl]ethyl}-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N-(5-hydroxyadamantan-2-yl)-3-(2-{[4-(methylsulfanyl)phenyl]methyl}-5-oxopyrrolidin-2-yl)propanamide
1-cyclohexyl-3-[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]urea
3-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecane-9-carbonyl}-1-methyl-1,4-dihydroquinolin-4-one
[1-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)-3-(2-methoxyethyl)piperidin-3-yl]methanol
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N-methyl-3,4-dihydro-2H-1-benzopyran-3-carboxamide
(1S,5R)-3-[6-(methoxymethyl)pyrimidin-4-yl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(5-chloropyridin-2-yl)-4-[4-(4H-1,2,4-triazol-4-yl)benzoyl]piperazine
N-[(1-ethylpyrrolidin-2-yl)methyl]-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-3,5-dimethylfuran-2-carboxamide
[2-(4-methoxyphenyl)ethyl]({[7-(methylsulfanyl)-2-(thiophen-2-yl)quinolin-3-yl]methyl})amine
4-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-6-(propan-2-yl)pyrimidine
N-[(4,6-dimethylpyridin-3-yl)methyl]-3-(pyrrolidine-1-carbonyl)benzene-1-sulfonamide
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-(oxolan-2-ylmethyl)-N-(pyridin-4-ylmethyl)acetamide
1-{4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3,3-dimethylbutan-1-one
3-(2,3-dihydro-1H-inden-2-yl)-5-methyl-5-[1-(quinolin-7-ylmethyl)piperidin-4-yl]imidazolidine-2,4-dione