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(3S,7S)-5-(2,6-dimethylpyrimidine-4-carbonyl)-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
2-(5-amino-1,3,4-thiadiazol-2-yl)-1-{4-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-1-yl}ethan-1-one
1-benzyl-4-{[4-(2-ethyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-1,3-oxazol-2-yl]methyl}piperazine
2-[4-methyl-3-(2-oxoimidazolidin-1-yl)benzoyl]-2,7-diazaspiro[4.5]decan-6-one
4-{[(2,3-dimethoxyphenyl)methyl]amino}-5-methyl-N-[2-(piperidin-1-yl)ethyl]thieno[2,3-d]pyrimidine-6-carboxamide
3-(3-fluorophenyl)-N,N-bis(2-methoxyethyl)-1H-pyrazole-4-carboxamide
3-({[(1-ethyl-1H-imidazol-2-yl)methyl]amino}methyl)-3-hydroxy-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
methyl 1-[(3R,5S)-1-cyclopentyl-5-[(thiophen-2-ylmethyl)carbamoyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
N-[3-(3-methylphenyl)phenyl]-1-(3,3,3-trifluoropropanoyl)piperidine-3-carboxamide
1-(piperidine-1-sulfonyl)-4-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}-1,4-diazepane
1-cyclohexyl-3-(cyclopropylmethyl)-5-(1,4-oxazepane-4-carbonyl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
(5-{[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}furan-2-yl)methanol
3-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-(1-methyl-1H-1,2,3-triazol-4-yl)benzamide
4-[(3-methoxyphenyl)methyl]-1-(2-methylpropanoyl)piperidine-4-carboxylic acid
1-(4-benzylpiperazin-1-yl)-3-{1-[(3-methoxyphenyl)methyl]piperidin-3-yl}propan-1-one
3-(benzyloxy)-1-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine
N,N-diethyl-2-{4-[4-(2-phenylethyl)piperidine-1-carbonyl]-1H-1,2,3-triazol-1-yl}acetamide
3-(3-hydroxy-1,2-oxazol-5-yl)-1-{4-[6-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-1-yl}propan-1-one
2,2-dimethyl-N-(1-{1-[3-(1-oxo-2,3-dihydro-1H-isoindol-2-yl)propanoyl]piperidin-4-yl}-1H-pyrazol-5-yl)propanamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-5-methyl-6-(4-methylpiperidine-1-carbonyl)thieno[2,3-d]pyrimidin-4-amine
1-({2-[(2-chloro-6-fluorophenyl)methoxy]phenyl}methyl)-1,4-diazepan-5-one
2-{3-[3-(3-methylpyrazin-2-yl)phenyl]-1H-pyrazol-1-yl}-N-(pyrazin-2-yl)acetamide
(3S,4R)-1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
2-(2H-1,3-benzodioxol-5-yl)-N-[2-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)ethyl]acetamide
4-{2-[3-(4-chloro-2-methylbenzoyl)piperidine-1-carbonyl]phenyl}morpholine
5-[3-(3-benzoylpiperidin-1-yl)-3-oxopropyl]-5-[(3,4-dimethoxyphenyl)methyl]pyrrolidin-2-one
methyl 3-(2,4-dimethylbenzoyl)-7-oxo-9-[2-(2-oxopyrrolidin-1-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-(3-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}phenyl)ethan-1-one
1-[5-(1H-pyrazol-1-ylmethyl)furan-2-carbonyl]-4-(thian-4-yl)piperazine
1-acetyl-N-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]piperidine-4-carboxamide
N-{[2-(dimethylamino)-8-methylquinolin-3-yl]methyl}-N-[2-(dimethylamino)ethyl]-3-(4-methylphenyl)propanamide
N-[(1R,3R)-3-aminocyclopentyl]-3,4,7-trimethyl-1H-indole-2-carboxamide
2-(adamantan-1-yl)-N-[2-(1H-1,2,4-triazol-1-yl)propyl]acetamide
1-(adamantan-1-yl)-4-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)piperazine
N-(1-{7-[(2,4,5-trimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)pyridine-3-carboxamide
N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-2-oxo-1,2-dihydroquinoline-4-carboxamide
propyl N-[(4-hydroxy-1-{imidazo[1,2-a]pyridine-3-carbonyl}azepan-4-yl)methyl]carbamate
N-[(5-{[(2-chlorophenyl)methyl]sulfanyl}-4-(2-methylpropyl)-4H-1,2,4-triazol-3-yl)methyl]-2-fluorobenzamide
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-(1-propylpiperidin-3-yl)-1,3-oxazole-4-carboxamide
1-(5-chloropyridin-2-yl)-4-[4-(methoxymethyl)-5-methyl-1,2-oxazole-3-carbonyl]piperazine
N-[2-(dimethylamino)-2-(3-methylthiophen-2-yl)ethyl]-3-(3-fluorophenyl)-1H-pyrazole-4-carboxamide
3-[4-(hydroxymethyl)phenyl]-5-(morpholine-4-sulfonyl)benzoic acid
1-{6-ethyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-3-(2-methylphenyl)pyrrolidin-3-ol
(2S,4R)-4-amino-N-ethyl-1-{[3-(morpholin-4-ylmethyl)phenyl]methyl}pyrrolidine-2-carboxamide
3-phenyl-1-(3-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-1-yl)prop-2-yn-1-one
N4-[2-(pyrrolidin-1-yl)ethyl]-5,6,7,8-tetrahydroquinazoline-2,4-diamine
4-(5-{[2-(dimethyl-1,2-oxazol-4-yl)pyrrolidin-1-yl]methyl}-1,3-thiazol-2-yl)morpholine
1-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-2-methyl-1,4-dihydroquinolin-4-one
3-methyl-5-{9-oxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carbonyl}-2,3-dihydro-1,3-benzoxazol-2-one
ethyl (2R,3S,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carboxylate