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(2S,4S)-4-amino-N-ethyl-1-(5-methyl-3-phenyl-1,2-oxazole-4-carbonyl)pyrrolidine-2-carboxamide
2-cyclohexyl-5-({4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}methyl)pyrimidine
1-[7-(pyrrolidine-1-sulfonyl)-1,2,3,4-tetrahydroisoquinoline-2-carbonyl]cyclopropane-1-carboxamide
3-methyl-N-{2-[(pyridin-2-ylmethyl)carbamoyl]phenyl}furan-2-carboxamide
N,2,8-trimethyl-N-[(trimethyl-1H-pyrazol-4-yl)methyl]quinoline-4-carboxamide
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
5-[1-(2,6-difluorobenzoyl)piperidin-4-yl]-3-[2-(dimethylamino)ethyl]-5-(3-methylbutyl)imidazolidine-2,4-dione
5-cyclopropyl-N-[2-(dimethylamino)-1-phenylethyl]-N-methyl-1,3-oxazole-4-carboxamide
1-cyclopropanecarbonyl-N-[2-methyl-1-(1-methyl-1H-imidazol-2-yl)propyl]piperidine-4-carboxamide
2-methyl-7-{3-[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]propanoyl}-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-{[4-(3,4-dimethoxyphenyl)-1H-1,2,3-triazol-1-yl]methyl}-4-methyl-5,6,7,8-tetrahydroquinazoline
(3S,4S)-3-(dimethylamino)-N-(2-fluorophenyl)-4-hydroxypyrrolidine-1-carboxamide
2-[1-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperidin-2-yl]pyridine
1-[(5-chlorofuran-2-yl)methyl]-4-{[1,2,4]triazolo[4,3-a]pyrimidin-5-yl}piperazine
(1S,4S)-2-[2-(3-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]-2-azabicyclo[2.2.1]heptane
methyl 3-(2-methoxyacetamido)-1-[2-(4-methoxyphenyl)ethyl]-5-{[1-(methylsulfanyl)propan-2-yl]amino}-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-[(4-methoxypyridin-2-yl)methyl]-5-(pyrrolidin-1-yl)-2,3-dihydropyridazin-3-one
N,N-dimethyl-4-(2,3,4,5-tetrahydro-1-benzoxepine-4-carbonyl)piperazine-1-carboxamide
N-(4-{4-phenyl-1-[2-(1H-pyrazol-4-yl)ethyl]-1H-imidazol-5-yl}phenyl)acetamide
N-cyclopentyl-N-[(2,4-dimethoxyphenyl)methyl]imidazo[1,2-a]pyridine-6-carboxamide
1-(2-{2-carbamoyl-1-methyl-1H,4H,5H,6H,7H-pyrrolo[2,3-c]pyridin-6-yl}-2-oxoethyl)piperidine-4-carboxamide
2-[5-(cyclopropylmethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl]-1-(prop-2-en-1-yl)-1H-1,3-benzodiazole
N,N-dimethyl-2-{[2-(pyridin-3-yl)acetamido]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
1-(morpholin-4-yl)-3-[3-(pyrrolidin-1-ylmethyl)phenoxy]propan-2-ol
5-(3-phenylpropyl)-5-[1-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl)piperidin-4-yl]imidazolidine-2,4-dione
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-4-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]butanamide
2-[4-(dimethylamino)phenyl]-1-[6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]ethan-1-one
2-cyclopentyl-8-[4-methyl-6-(methylamino)pyrimidin-2-yl]-2,8-diazaspiro[5.5]undecan-3-one
3-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1,2-dimethyl-1H-indol-5-ol
5-[1-(2,2-dimethyl-4-oxo-3,4-dihydro-2H-pyran-6-carbonyl)piperidin-4-yl]-5-propyl-3-[2-(pyridin-2-yl)ethyl]imidazolidine-2,4-dione
4-(4-ethoxy-3-methylphenyl)-N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}butanamide
(3aR,5R,6S,7aS)-2-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-octahydro-1H-isoindole-5,6-diol
N-(3-hydroxypropyl)-2-{1-[(2-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-(propan-2-yl)acetamide
(2S,4S)-4-[(cyclohexylmethyl)amino]-N-ethyl-1-(propan-2-yl)pyrrolidine-2-carboxamide
4-{[3-(dimethylamino)propyl]amino}-N-ethyl-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
N5-[(1-methyl-1H-imidazol-2-yl)methyl]-N5-(propan-2-yl)-N6-(thiophen-2-ylmethyl)-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
2-[(3,5-difluorophenyl)methyl]-8-(2-hydroxybutyl)-2,8-diazaspiro[4.5]decan-3-one
5-(2-{2-[(6-aminopyrimidin-4-yl)amino]ethyl}morpholin-4-yl)-2-methyl-2,3-dihydropyridazin-3-one
5-acetyl-N-{[7-(2-chloro-6-fluorobenzoyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}thiophene-3-carboxamide
4-[1-(3-methyl-1H-pyrazole-4-carbonyl)piperidin-3-yl]morpholine
N-({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-(5-methyl-1,3-diphenyl-1H-pyrazole-4-carbonyl)piperazine
2-[4-(5-methoxy-1,2-dimethyl-1H-indole-3-carbonyl)morpholin-3-yl]-N,N-dimethylacetamide
N-[2-(cyclohex-1-en-1-yl)ethyl]-5-[4-(1H-1,2,4-triazol-1-yl)phenoxymethyl]-1,2-oxazole-3-carboxamide
1-methyl-4-{2-methyl-2-[5-(2-methylprop-1-en-1-yl)-4-phenyl-1H-imidazol-1-yl]propyl}piperazine
3-[3-fluoro-4-(trifluoromethyl)phenyl]-1-(2-methoxyethyl)-1-(1-methylpiperidin-4-yl)urea
4-{1,9-dimethyl-1,4,9-triazaspiro[5.5]undecane-4-carbonyl}benzene-1-sulfonamide
(3S,5R)-1-(1H-1,2,3-benzotriazole-5-carbonyl)-5-(cyclopropylcarbamoyl)piperidine-3-carboxylic acid
6-(cyclohex-1-ene-1-carbonyl)-N-(3-fluorophenyl)-6-azaspiro[2.5]octane-1-carboxamide
N-[2-(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]-2-(methylsulfanyl)acetamide