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N-[2-(4-chlorophenyl)ethyl]-3-[(3S,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-1-(pyridin-2-ylmethyl)piperidin-3-yl]propanamide
methyl 7-oxo-9-[2-(piperidin-1-yl)ethoxy]-3-(1H-pyrazole-4-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
5-{4-[1-methyl-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]piperazin-1-yl}-2,3-dihydropyridazin-3-one
3-[5-(2H-1,3-benzodioxol-5-ylmethyl)-1,3,4-oxadiazol-2-yl]-N-[2-(diethylamino)ethyl]propanamide
methyl 2-(4-{6-tert-butyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-3-methyl-2-oxopiperazin-1-yl)acetate
N-ethyl-N-(2-hydroxyethyl)-4-{[(2-methoxyphenyl)methyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-6-({5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}amino)pyridine-3-carboxamide
1-(2-methoxyphenyl)-N-methyl-N-(quinolin-3-ylmethyl)-1H-pyrazole-4-carboxamide
N-cyclohexyl-2-[3-(2-methoxyphenyl)-1-(3-methoxypropyl)-2,5-dioxopyrrolidin-3-yl]-N-methylacetamide
3-(2-fluorophenyl)-N-methyl-N-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-1H-pyrazole-4-carboxamide
2-{4-[6-(methoxymethyl)-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl]piperazin-1-yl}benzonitrile
1-{2-[2-(3-fluorophenyl)ethyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}-N-methyl-N-(thiophen-2-ylmethyl)piperidine-4-carboxamide
dimethyl({4-methyl-5-[1-(2-methyl-5-propylpyrimidin-4-yl)piperidin-3-yl]-4H-1,2,4-triazol-3-yl}methyl)amine
N-cyclopentyl-1-(2-methoxyacetyl)-N-(thiophen-3-ylmethyl)piperidine-4-carboxamide
N-[2-hydroxy-2-(pyridin-4-yl)ethyl]-5-phenyl-1,2-oxazole-3-carboxamide
N-[(2-chlorophenyl)methyl]-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide
N-ethyl-N-[1-({[5-(methoxymethyl)-1,3,4-thiadiazol-2-yl]carbamoyl}methyl)pyrrolidin-3-yl]acetamide
3-(3-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}phenyl)-1H-1,2,4-triazole
(9aR)-N-cyclohexyl-8-methyl-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxamide
1-[(2R,3S,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-(methylsulfanyl)propan-1-one
N-methyl-4-[3-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]pyridin-2-amine
{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl)(thiophen-2-ylmethyl)amine
2-{3-[({[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)methyl]phenoxy}acetamide
N-[(1R,3R)-3-aminocyclopentyl]-2-(phenylamino)pyrimidine-5-carboxamide
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
1-(5-chlorothiophene-2-carbonyl)-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
1-{3-[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]propyl}-1H-1,2,3,4-tetrazole
(1-ethyl-5-{imidazo[1,2-a]pyridine-6-carbonyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl)methanol
2-(4-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl)ethan-1-ol
methyl (2S,4R)-1-[(3-ethoxy-4-methoxyphenyl)methyl]-4-(2-phenylbenzamido)pyrrolidine-2-carboxylate
2-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}-6-methylpyridine-3-carbonitrile
8-chloro-N-[2-(dimethylamino)-2-(furan-2-yl)ethyl]-2-methylquinoline-4-carboxamide
2,5-difluoro-N-(1-{7-[(2-phenyl-1,3-thiazol-5-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)benzamide
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-4-oxo-3,4-dihydrophthalazine-1-carboxamide
4-methoxy-6-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidine
3-methoxy-N-({3-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-N-(pyridin-2-ylmethyl)benzamide
ethyl 5-cyclopentyl-1-[2-(dimethylamino)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)-N-[2-(2-methylphenyl)-1,3-benzoxazol-6-yl]acetamide
2-(3-fluorophenyl)-1-(3-phenyl-1H-pyrazole-4-carbonyl)piperidine
2-[1-(2,2-dimethylpropyl)-4-[(1-phenyl-1H-pyrazol-4-yl)methyl]piperazin-2-yl]ethan-1-ol
N-[1-(adamantan-1-yl)-2-methylpropan-2-yl]-3-{2-[(3,4-dimethoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
(1S,7R)-2-methyl-4-{[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]methyl}-4-azatricyclo[5.2.1.02,6]dec-8-ene-3,5-dione
2-{1-methyl-4-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperazin-2-yl}ethan-1-ol
N-[(3S)-1-{5-[(2H-1,3-benzodioxol-5-yloxy)methyl]-1H-pyrazole-3-carbonyl}pyrrolidin-3-yl]acetamide
{[3-(2H-1,3-benzodioxol-5-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}(methyl)[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amine
3-[(3S,4R)-1-benzyl-4-(morpholin-4-yl)piperidin-3-yl]-N-(4-methoxyphenyl)propanamide
5-{[benzyl(methyl)amino]methyl}-N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-1,2-oxazole-3-carboxamide
1-cyclopentyl-3-(2-methylphenyl)-3-{2-oxo-2-[4-(piperidine-1-carbonyl)piperidin-1-yl]ethyl}pyrrolidine-2,5-dione
(3S)-1-(4-{[(3R)-3-methylpiperazin-1-yl]sulfonyl}benzoyl)pyrrolidin-3-amine
N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)-2-(pyrrolidin-1-yl)propanamide