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1-(3-methylthiophene-2-carbonyl)-4-[2-(1H-pyrazol-1-yl)ethyl]piperidine
8-fluoro-N-methyl-N-[(1-phenylpyrrolidin-3-yl)methyl]quinoline-2-carboxamide
(4aS,7aR)-1-(ethanesulfonyl)-4-(2-methoxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}-2-(pyrrolidin-1-yl)propanamide
2-{2-cyclopropyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}-N-methylacetamide
6-hydroxy-4-[(2-phenyl-1,3-thiazol-5-yl)methyl]-1-(pyridin-3-ylmethyl)-1,4-diazepan-2-one
1-(benzenesulfonyl)-N-(2,3-dihydro-1H-inden-2-yl)piperidin-4-amine
9-ethyl-1-methyl-4-[4-(thiophen-2-yl)butanoyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
4-{2-[(4aS,7aS)-octahydro-1H-pyrrolo[3,4-b]pyridin-6-yl]-2-oxoethyl}-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one
1-methyl-4-{[4-(5-methylfuran-2-yl)phenyl]methyl}piperazine
N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-1-(3-phenylbutyl)piperidine-4-carboxamide
2-[(1S,5R)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]pyridin-3-ol
{1-[(1-cycloheptanecarbonylpiperidin-3-yl)methyl]-1H-1,2,3-triazol-4-yl}methanol
[(5-ethylpyridin-2-yl)methyl](methyl){[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}amine
{[5-(4-methoxy-3,5-dimethylphenyl)-1,2,4-oxadiazol-3-yl]methyl}dimethylamine
4-[1-(2-methyl-1,3-benzothiazole-5-carbonyl)piperidin-3-yl]benzoic acid
6-cyclobutyl-2-(4-{[methyl(oxan-4-yl)amino]methyl}phenyl)-3,4-dihydropyrimidin-4-one
(1S,5R)-6-(3,5-difluoropyridine-2-carbonyl)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
N-{[7-methoxy-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)cyclopropanecarboxamide
{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)(1,3-thiazol-2-ylmethyl)amine
N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-2-ethyl-4-methyl-1,3-oxazole-5-carboxamide
2-ethyl-1-(2-methyl-1-benzofuran-7-carbonyl)-2,5-dihydro-1H-pyrrole
N-{1-[(2-chlorophenyl)methyl]-3-methyl-1H-pyrazol-5-yl}-2-(2-propyl-1H-imidazol-1-yl)acetamide
benzyl(ethyl)({1-[(2-fluorophenyl)methyl]-2-(propane-2-sulfonyl)-1H-imidazol-5-yl}methyl)amine
5-(2-chlorophenyl)-3-[2-(1H-pyrazol-1-yl)ethyl]-3H,4H-thieno[2,3-d]pyrimidin-4-one
4-(3-tert-butyl-1H-pyrazol-1-yl)-1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidine-4-carboxylic acid
1-methyl-8-(pyridin-3-ylmethyl)-3-[3-(pyridin-4-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-{1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]piperidin-4-yl}-N-[2-(dimethylamino)ethyl]propanamide
1-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidin-1-yl]-4-(4-fluorophenyl)butane-1,4-dione
methyl 3-[2-(1-ethylpiperidin-3-yl)-1H-imidazol-1-yl]propanoate
N-methyl-5-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]-N-(oxan-2-ylmethyl)pyridin-2-amine
2-[4-(dimethylamino)phenyl]-1-{2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidin-1-yl}ethan-1-one
5-(3,4-difluorophenoxymethyl)-N-methyl-N-(pyridin-3-ylmethyl)-1,2-oxazole-3-carboxamide
1-(4-{[4-(5-chloro-2-fluorobenzoyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}piperazin-1-yl)ethan-1-one
4-(3-hydroxypyridine-2-carbonyl)-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-(2-chlorophenyl)-3-{2-[4-(2-methoxyethyl)piperazin-1-yl]-2-oxoethyl}-1-(3-methoxypropyl)pyrrolidine-2,5-dione
N-methyl-2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-(quinolin-4-ylmethyl)acetamide
1-(4-ethyl-5-methylthiophene-3-carbonyl)-4-(1H-imidazol-1-yl)piperidine-4-carboxylic acid
2-cyclopropyl-9-methanesulfonyl-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
2-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-[2-(3-methylpyridin-2-yl)ethyl]benzamide
8-[(4-methylphenyl)methyl]-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
3-(1,2-oxazinan-2-yl)-N-[1-(pyrazin-2-yl)propan-2-yl]propanamide
3-{[3-(piperidin-1-yl)pyrrolidin-1-yl]methyl}pyridin-2-amine
N-(2,2-dimethyloxan-4-yl)-N-ethyl-3-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]propanamide
1-methyl-4-(5-{[(6-methylpyridin-3-yl)oxy]methyl}-1,2-oxazole-3-carbonyl)-2-phenylpiperazine
N-ethyl-2-(1H-pyrazol-4-yl)-N-(pyridin-3-ylmethyl)quinoline-4-carboxamide
4-{[5-(5-methyl-1,3-oxazole-4-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}thiomorpholine
2-ethyl-8-{2-[4-(trifluoromethyl)phenyl]acetyl}-2,8-diazaspiro[4.5]decan-3-one
[1-(2-chlorophenyl)ethyl]({[3-(3-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl})amine
3-methoxy-N-{[4-(4-methylphenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}propanamide