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1-(1,4-dioxan-2-ylmethyl)-5-(1H-imidazol-4-ylmethyl)-3-(oxan-4-yl)-1H-1,2,4-triazole
4-(1-{1-[(2-methylpyrimidin-5-yl)methyl]piperidin-4-yl}piperidine-3-carbonyl)morpholine
1-[4-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]-2-(3-methyl-1,2,4-oxadiazol-5-yl)piperidine
3-methyl-1-(2-methylpropyl)-4-(pyrazine-2-carbonyl)piperazin-2-one
2-ethyl-1-{[2-(4-methoxy-2,5-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine
(2R,3R,6R)-N-tert-butyl-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carboxamide
5-(cyclohex-3-en-1-yl)-4-phenyl-1-[2-(trimethyl-1H-pyrazol-1-yl)ethyl]-1H-imidazole
4-chloro-N,N-diethyl-3-({[3-(oxolan-3-yl)propyl]carbamoyl}amino)benzamide
2-{4-[2-oxo-2-(piperidin-1-yl)acetyl]morpholin-3-yl}-N-[2-(1H-pyrazol-4-yl)ethyl]acetamide
[1-(5-{[(3-chlorophenyl)methyl]amino}-5,6,7,8-tetrahydroquinazolin-2-yl)piperidin-4-yl]methanol
4-(3,5-dimethyl-1H-pyrazol-1-yl)-1-[(3R,4R)-4-ethyl-3,4-dihydroxypiperidin-1-yl]butan-1-one
[(3R,4R)-1-(4-chloro-3-fluorobenzoyl)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)pyrrolidin-3-yl]methanol
(1S,6R)-3-methyl-9-[3-(1H-1,2,4-triazol-1-yl)propanoyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
5-{1-benzyl-3-methyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-1,3-dimethyl-1H-pyrazole
1-{[2-(2,3-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-phenylpiperidine
methyl 3-[(3S,4R)-4-(dimethylamino)-1-[(3-fluorophenyl)methyl]piperidin-3-yl]propanoate
N-[3-(1,3-benzothiazol-2-yl)propyl]-1,9-dioxaspiro[5.5]undecan-4-amine
N-({4-[(3-phenylpropyl)amino]quinazolin-2-yl}methyl)furan-3-carboxamide
2-(dimethylamino)-2-(3-fluorophenyl)-N-(2-methoxyethyl)-N-(pyridin-4-ylmethyl)acetamide
3-[1-(9H-fluoren-2-ylmethyl)piperidin-4-yl]-N-(oxolan-2-ylmethyl)propanamide
N-(1-{[methyl(2-phenoxyethyl)carbamoyl]methyl}-1H-pyrazol-4-yl)-4-oxo-4-phenylbutanamide
methyl 4-[({[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl}amino)methyl]benzoate
1-[4-(2-fluorophenyl)pyrimidin-2-yl]-5-(propan-2-yl)-N-[3-(pyridin-4-yl)propyl]-1H-pyrazole-4-carboxamide
3-{2-[(2-fluoro-5-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[(4-phenyl-1,3-thiazol-2-yl)methyl]propanamide
1-[2-(naphthalen-1-ylmethyl)morpholin-4-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
2-(2-acetyl-4,5-dimethoxyphenyl)-1-{3,5-dimethyl-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl}ethan-1-one
4-ethyl-1-methyl-3-{1-[5-(propan-2-yl)-1,3-oxazole-4-carbonyl]piperidin-3-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
2-[4-(benzyloxy)-3-chlorophenyl]-4-(pyrrolidine-1-carbonyl)pyridine
N-[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-N-methyl-2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)acetamide
N-(1-oxo-2,3-dihydro-1H-inden-5-yl)-4-(thiophen-2-ylmethyl)-1,4-diazepane-1-carboxamide
1-(cyclohexylmethyl)-N3-cyclopropyl-N5-[2-methyl-2-(morpholin-4-yl)propyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
1-(pyridin-4-ylmethyl)-5-[3-(pyrrolidin-1-yl)propanoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
1-(2,3-dihydro-1H-inden-2-yl)-N-[3-(1H-pyrazol-1-yl)phenyl]piperidine-3-carboxamide
methyl({[1-(2-methylpropyl)piperidin-4-yl]methyl})({3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}methyl)amine
N-cyclopropyl-2-(7-fluoro-2-methyl-1H-indol-3-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]acetamide
5-{1-[(2E)-4-methylpent-2-enoyl]piperidin-4-yl}-3-(oxolan-2-ylmethyl)-5-propylimidazolidine-2,4-dione
1-(4-{[bis(1,3-oxazol-4-ylmethyl)amino]methyl}thiophen-2-yl)ethan-1-one
1-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-4,4-difluoropiperidine
1-butyl-4-[1,3-dimethyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]piperazin-2-one
1-[(3R,4R)-3-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(pyridin-2-ylsulfanyl)ethan-1-one
N-[(3S,4R)-4-(5-methylfuran-2-yl)-1-[3-(thiophen-3-yl)propanoyl]pyrrolidin-3-yl]acetamide
1-[2-(3-methoxyphenyl)piperidin-1-yl]-2-(pyridin-3-yl)ethan-1-one
1-{4H,5H,6H,7H,8H-cyclohepta[b]thiophene-2-carbonyl}-N-cyclopropylpiperazine-2-carboxamide
3-chloro-N-[4-(4-{[3-(2-oxopyrrolidin-1-yl)propyl]amino}piperidin-1-yl)phenyl]benzamide
3-[3-(3-ethylphenoxy)azetidine-1-carbonyl]-5-(propan-2-yl)-1,2-oxazole
(1H-imidazol-4-ylmethyl)(methyl){2-[(4-methylphenyl)sulfanyl]ethyl}amine
1-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-4-(4-fluorophenyl)butan-1-one
N-butyl-2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-[(3-methylthiophen-2-yl)methyl]acetamide
1-{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-3-(3-methoxyphenoxymethyl)piperidine
4-(pyridin-3-yl)-2-[4-(pyrrolidine-1-sulfonyl)piperazin-1-yl]pyrimidine