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2-{1-[(3,5-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-hydroxy-2-(prop-2-en-1-yl)pent-4-en-1-yl]acetamide
1-cyclohexyl-N-(pyrimidin-4-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
6-methyl-5-[5-(2-methyl-1-benzofuran-7-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridine
2-(1-methyl-3-oxopiperazin-2-yl)-N-[5-(morpholin-4-yl)pentyl]acetamide
(1S,5R)-6-propyl-3-[3-(4H-1,2,4-triazol-4-yl)benzoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
3-(2-oxo-2-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}ethyl)-3H,4H-thieno[3,2-d]pyrimidin-4-one
2-{1-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]pyrrolidin-2-yl}-1,3-thiazole
2-{4-[1-(3,5-dimethylphenyl)piperidin-4-yl]-1-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl}ethan-1-ol
1-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
methyl 1-[(3S,5S)-5-{[2-(1H-indol-3-yl)ethyl]carbamoyl}-1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
propan-2-yl (1S,5R)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxylate
({4-ethyl-5-[1-(2-fluoro-4-methylbenzoyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
9-(1-benzofuran-5-carbonyl)-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-3-{imidazo[1,2-a]pyridin-2-yl}-N-methylpropanamide
N-methyl-4-oxo-1-(3-phenylpropyl)-5-[4-(thiophen-2-ylmethyl)piperazine-1-carbonyl]-1,4-dihydropyridine-3-carboxamide
2-(2-fluorophenyl)-1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-1-yl]ethan-1-one
1-(2-methoxy-3-methylbenzoyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-[(2,4-dimethoxyphenyl)methyl]-3-[1-(pyridin-3-ylmethyl)piperidin-3-yl]propanamide
3-ethyl-6-[4-(2-methoxyethyl)piperazine-1-carbonyl]-3H-imidazo[4,5-b]pyridin-2-amine
(3S,5S)-1-(3-phenylpropyl)-5-[(pyridin-2-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
7-(cyclopropylmethyl)-2-[2-(methylamino)-1,3-thiazole-4-carbonyl]-2,7-diazaspiro[4.5]decan-6-one
3-ethyl-8-[(2-fluoro-5-methoxyphenyl)methyl]-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-fluoro-N4-methyl-N2-{[4-(4-methylphenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}pyrimidine-2,4-diamine
(1s,4s)-4-[3-(3-chlorophenoxy)azetidine-1-carbonyl]cyclohexan-1-ol
2-{[3-(3,4-dimethoxybenzoyl)piperidin-1-yl]methyl}-3-methoxyphenol
3-(2-{4-[(3-fluorophenyl)methyl]piperazin-1-yl}-2-oxoethyl)-3-(2-methoxyphenyl)-1-methylpyrrolidine-2,5-dione
({2-[(dimethylamino)methyl]phenyl}methyl)[(2-ethylpyrimidin-4-yl)methyl]methylamine
6-[6-(piperazin-1-yl)pyridin-2-yl]quinoline
N-[2-(2-fluorophenyl)ethyl]-1-methyl-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
(1S,6R)-9-(3-chloro-4-fluoro-1-benzothiophene-2-carbonyl)-3,9-diazabicyclo[4.2.1]nonan-4-one
(3S,9aR)-8-[(3-fluoro-4-methylphenyl)methyl]-3-(1H-indol-3-ylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-(2-amino-1,3-thiazol-4-yl)-N-[2-(cyclohexylsulfanyl)ethyl]propanamide
3-{1-[2-(azepan-1-yl)acetyl]piperidin-3-yl}-N-(3,5-dimethoxyphenyl)propanamide
1-[(4aS,8aR)-decahydroisoquinolin-2-yl]-3-{5-[2-(3-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propan-1-one
5-(5-cyclohexyl-1,2,4-oxadiazol-3-yl)-6-methyl-N-(propan-2-yl)-1,2,3,4-tetrahydro-2,7-naphthyridine-2-carboxamide
1-{3-[(3,4-difluorophenyl)amino]piperidin-1-yl}-2-[methyl(piperidin-4-yl)amino]ethan-1-one
5-(2-methoxybutanoyl)-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-N-[2-(1H-pyrazol-4-yl)ethyl]piperidine-3-carboxamide
2,3,5-trimethyl-N-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
2-methyl-4-phenyl-1-{[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperazine
4-{2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]-2-oxoethyl}-3,4-dihydro-2H-1,4-benzoxazin-3-one
2-{[(2-methyl-1H-imidazol-4-yl)methyl](thiophen-2-ylmethyl)amino}butan-1-ol
4-(3-methyl-1,2,4-oxadiazol-5-yl)-2-[2-methyl-4-(pyrrolidin-1-ylmethyl)phenoxy]pyridine
methyl 3-[(3S,4R)-1-(pyridin-2-ylmethyl)-4-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-3-yl]propanoate
5-{3-[4-(4-fluorophenyl)piperazin-1-yl]piperidine-1-carbonyl}pyrazin-2-ol
3-(2-cyclohexylacetyl)-N-[1-(furan-2-yl)ethyl]-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
methyl 6-(1-benzofuran-2-carbonyl)-2-[(butan-2-yl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
(3S,4R)-1-[(2-aminopyridin-3-yl)methyl]-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
1-(5-{3-[(4-methoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}pyridin-2-yl)piperidin-4-ol
4-({3-[(2-fluorophenyl)methyl]-3-(hydroxymethyl)piperidin-1-yl}methyl)-1,5-dimethyl-2-phenyl-2,3-dihydro-1H-pyrazol-3-one