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N-[(3,4-dimethoxyphenyl)methyl]-3-[2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propanamide
methyl 3-(2-methoxybenzoyl)-7-oxo-9-[2-(piperidin-1-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-[3-(morpholine-4-carbonyl)-1-(2-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-(pyridin-4-ylsulfanyl)ethan-1-one
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-1-{2-[(3-fluorophenyl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}piperidine-3-carboxamide
4-{[4-(3-phenylpiperazine-1-carbonyl)furan-2-yl]methyl}morpholine
N-({8-benzyl-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-3-cyclopentylpropanamide
1-[2-(3-methoxyphenyl)piperidin-1-yl]-3-(methylsulfanyl)propan-1-one
4-(cyclopropylmethyl)-1-[(1-methyl-1H-indol-3-yl)methyl]-1,4-diazepan-5-one
9-[(2-methoxy-4-methylphenyl)methyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[2-(dimethylamino)ethyl]-3-{1-[1-(2,3-dimethylphenyl)piperidin-4-yl]piperidin-4-yl}propanamide
N-[2-(2-fluorophenyl)-1-[1-(4-methylbenzoyl)piperidin-4-yl]ethyl]-N,2-dimethylfuran-3-carboxamide
N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
6-[(2-propoxyethyl)amino]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
2-(3,6-dimethylpyrazin-2-yl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
3-[benzyl({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl})amino]-1λ6-thiolane-1,1-dione
(1S,5R)-6-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
(3R,4S)-1-(butane-1-sulfonyl)-4-(5-methylfuran-2-yl)pyrrolidin-3-amine
1-methyl-8-[(2E)-3-phenylprop-2-en-1-yl]-3-[3-(pyridin-4-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-{methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
1-[1-(5-methyl-1,2-oxazole-3-carbonyl)piperidin-4-yl]-3-(pyrrolidine-1-carbonyl)piperidine
4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-(1-phenyl-1H-1,2,3-triazole-4-carbonyl)piperidine
6-chloro-2-{2-[3-(4-ethyl-1-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]-2-oxoethyl}-2,3-dihydropyridazin-3-one
N-{[2-(1H-imidazol-1-yl)phenyl]methyl}-1-methyl-1H-indole-6-carboxamide
N,5-dimethyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1-benzofuran-2-carboxamide
1-(3-benzyl-4,5-dihydro-1,2-oxazole-5-carbonyl)-3-(2-fluorophenoxymethyl)piperidine
1-[2-oxo-2-(2-{[3-(trifluoromethyl)phenyl]methyl}morpholin-4-yl)ethyl]pyrrolidin-2-one
4-(5-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}-1H-pyrazol-3-yl)pyridine
4-{[1-(dimethylsulfamoyl)piperidin-4-yl]oxy}-N-(2-hydroxypropyl)benzamide
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}cyclobutanecarboxamide
2-(5-{3-cyclopropyl-1-methyl-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl}furan-2-yl)benzonitrile
6-{imidazo[1,2-a]pyridin-3-ylmethyl}-3-propyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
N-cyclopropyl-1-{1-[6-methyl-2-(propan-2-yl)pyrimidin-4-yl]piperidin-4-yl}piperidine-3-carboxamide
2-amino-6-tert-butyl-4-[1-(2-hydroxyethyl)-3,5-dimethyl-1H-pyrazol-4-yl]pyridine-3-carbonitrile
N-methyl-2-{3-[2-methyl-6-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-1-yl}acetamide
4-[2-(dimethyl-1H-1,2,4-triazol-1-yl)acetyl]-6-[(3-methoxyphenyl)methoxy]-1-(2-phenylethyl)-1,4-diazepan-2-one
N-ethyl-1-(3-phenylpropyl)-N-[2-(pyrrolidin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
2-methyl-6-{1-[(4-phenyl-1,3-thiazol-5-yl)methyl]-1H-imidazol-2-yl}pyridine
N-{[2-(2-ethanesulfonamidophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-(2-methylphenyl)benzamide
[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl](methyl)[(3-phenyl-1H-pyrazol-5-yl)methyl]amine
N-ethyl-1-(7-methoxy-4-methylquinazolin-2-yl)-N-(oxolan-2-ylmethyl)piperidine-3-carboxamide
3,5-dichloro-N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-N,4-dimethylbenzamide
(3aS,6aS)-2-(6-cyclopropylpyrimidin-4-yl)-5-[2-(dimethylamino)acetyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-(4-fluorophenyl)-4-[4-(4H-1,2,4-triazol-4-yl)benzoyl]piperazin-2-one
3-ethoxy-N-[(3S,4R)-4-ethoxyoxolan-3-yl]-4-(prop-2-en-1-yloxy)benzamide
1-benzyl-8-cyclobutyl-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(3,5-dimethylphenyl)-6-[3-(2-methyl-1H-1,3-benzodiazol-1-yl)propanoyl]-6-azaspiro[2.5]octane-1-carboxamide
1-{1,9-dimethyl-1,4,9-triazaspiro[5.5]undecan-4-yl}-2-[(5-ethyl-1,3,4-oxadiazol-2-yl)sulfanyl]ethan-1-one
(furan-3-ylmethyl)[3-(1H-imidazol-1-yl)propyl](pyridin-4-ylmethyl)amine
1-methyl-2-{2-[(4-methyl-1H-imidazol-2-yl)methyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl}-1H-1,3-benzodiazole
3-[(2-methoxyethyl)sulfamoyl]-5-(1H-pyrazol-3-yl)benzoic acid