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(3aS,6aS)-2-[2-(phenylsulfanyl)acetyl]-5-propyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-{3-[1-tert-butyl-3-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]phenyl}imidazolidin-2-one
N-[1-(4-fluorophenyl)-4-(propan-2-yloxy)-1H-indazol-3-yl]-2-(furan-2-yl)-2-oxoacetamide
3-({6-oxo-3-phenyl-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl}methyl)-2,3-dihydro-1,3-benzoxazol-2-one
1-[5-({[(3,4-difluorophenyl)methyl]amino}methyl)-2-methoxyphenoxy]-3-(4-methylpiperazin-1-yl)propan-2-ol
5-(1-{[2-(furan-2-yl)phenyl]methyl}pyrrolidin-2-yl)-3-(propan-2-yl)-1,2,4-oxadiazole
2-(2-methylpropyl)-8-[5-(pyrrolidin-1-yl)pyridazin-3-yl]-2,8-diazaspiro[4.5]decan-3-one
N-[4-(3-methylphenyl)phenyl]-1-(thian-4-yl)piperidine-4-carboxamide
4-[7-(3-methyl-1H-pyrazole-5-carbonyl)-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl]benzamide
N-[(4-ethoxyphenyl)methyl]-N-(2-methoxyethyl)-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(2-methyl-1,3-oxazol-4-yl)methyl]piperidine
{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]amine
N-[(1R,2R)-2-hydroxycyclohexyl]-2-(4-oxo-1,4-dihydroquinolin-1-yl)-N-propylacetamide
1-tert-butyl-4-{7,7-dimethyl-4-oxo-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-2-yl}pyrrolidin-2-one
2-(5-{2-[(2-methylprop-2-en-1-yl)oxy]benzoyl}-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl)pyridine
N-(3-cyclopentylpropyl)-3-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]benzamide
2-{2-[1-(2-{8-methylimidazo[1,2-a]pyridin-3-yl}acetyl)piperidin-4-yl]-1H-imidazol-1-yl}acetamide
N-methyl-N-phenyl-4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carboxamide
2-{4-[(3,5-dimethoxyphenyl)methyl]-1-methylpiperazin-2-yl}ethan-1-ol
4-{imidazo[1,2-a]pyrimidine-2-carbonyl}-2-(trifluoromethyl)morpholine
N-ethyl-5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-N-[2-(1H-pyrazol-1-yl)ethyl]-1,2-oxazole-3-carboxamide
3-(1-methyl-1H-pyrrol-2-yl)-N-{[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}-1H-pyrazole-5-carboxamide
1,4-dimethyl-4-[3-(thiophen-3-ylmethyl)-1,2,4-oxadiazol-5-yl]piperidine
N-[3-(2-ethyl-1H-imidazol-1-yl)propyl]-1-(propan-2-yl)piperidine-4-carboxamide
(7-methyl-2-{4-[1-(morpholin-4-yl)ethyl]piperidin-1-yl}quinolin-3-yl)methanol
1-(3-methylbut-2-en-1-yl)-4-(3-methylphenoxy)piperidine-4-carboxylic acid
1-(5-methoxyfuran-2-carbonyl)-N-methyl-N-(2-phenylethyl)piperidin-3-amine
(3R,9aR)-3-(hydroxymethyl)-8-(quinolin-6-ylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-{1-[1-(5-methylhex-5-en-2-yl)piperidin-4-yl]-1H-pyrazol-5-yl}-4-phenylbutanamide
3-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(2-chloro-3,5-difluorophenyl)urea
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-1H-pyrrole-3-carboxamide
2-{[2-(1H-imidazol-1-yl)ethyl](methyl)amino}pyridine-3-carboxamide
6-chloro-4-(3,3-dimethylpyrrolidine-1-carbonyl)-2-(1-methyl-1H-pyrazol-4-yl)quinoline
{4-[2-(morpholin-4-yl)benzoyl]-1,4-oxazepan-6-yl}methanol
1-[3-(4-{[(1R,2R,4R)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]amino}piperidin-1-yl)phenyl]pyrrolidin-2-one
ethyl 5-[(2-chloro-6-fluorophenyl)methyl]-1-(2-hydroxyethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
2-cyclopentyl-N-{[4-fluoro-7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
[1-(5-ethyl-1,3,4-oxadiazol-2-yl)piperidin-4-yl](pyridin-2-yl)methanol
(1R,2R)-1-({2-methylpyrido[2,3-d]pyrimidin-4-yl}amino)-2,3-dihydro-1H-inden-2-ol
1-{6-[(3-methoxyphenyl)methoxy]-3-oxo-4-(2-phenylethyl)-1,4-diazepan-1-yl}-3-methylpentane-1,4-dione
N-{1-[2-(3-chlorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-2-(pyridin-2-ylsulfanyl)acetamide
3-(cyclobutylmethyl)-1-{4-[(5-methyl-4H-1,2,4-triazol-3-yl)methyl]phenyl}-3-(oxolan-2-ylmethyl)urea
ethyl 3-benzyl-1-(benzylcarbamoyl)piperidine-3-carboxylate
4-fluoro-3-[(3R,4S)-4-hydroxy-3,4-dimethylpiperidine-1-carbonyl]benzene-1-sulfonamide
(2E)-N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-3-(3,4-dimethoxyphenyl)-N-methylprop-2-enamide
1-[6-(4-methoxyphenyl)pyridine-3-carbonyl]-4-(pyrimidin-2-yl)-1,4-diazepane
ethyl 4-(6-{[3-(trifluoromethyl)phenyl]methyl}-6-azaspiro[2.5]octane-1-carbonyl)piperazine-1-carboxylate
3-(4-methyl-1,3-thiazol-5-yl)-N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}propanamide
1-(2-cyclohexylethyl)-3-hydroxy-3-{[methyl(2-phenylethyl)amino]methyl}piperidin-2-one
1-(furan-2-ylmethyl)-3-[5-(2-methylbutan-2-yl)-1,3,4-thiadiazol-2-yl]urea