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3-[(7-{trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]pyridine
7-fluoro-3-[2-(2-hydroxyethoxy)ethyl]-3,4-dihydroquinazolin-4-one
N-methyl-5-(morpholine-2-carbonyl)-4H,5H,6H,7H-thieno[3,2-c]pyridine-2-carboxamide
3-[({6-ethyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)methyl]-7-fluoro-1,2-dihydroquinolin-2-one
ethyl N-[(1R,3S)-3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)cyclopentyl]carbamate
N-[1-(3-fluoro-4-methoxyphenyl)ethyl]-5-hydroxy-4-oxo-4H-pyran-2-carboxamide
3-(3-methoxypropyl)-1-[2-(methylamino)pyrimidine-5-carbonyl]piperidine-3-carboxylic acid
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-1-{9-methyl-3,9-diazaspiro[5.6]dodecan-3-yl}ethan-1-one
N-(1H-1,3-benzodiazol-2-ylmethyl)-5-(3-methoxyphenoxymethyl)-N-methyl-1,2-oxazole-3-carboxamide
(1R,2S,6R,7S)-4-(5-propyl-1,3,4-oxadiazol-2-yl)-4-azatricyclo[5.2.2.02,6]undecane
2,6-dimethyl-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]imidazo[1,2-a]pyridine-3-carboxamide
1-{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(pyridin-2-yl)piperazine
1-{1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]piperidine-3-carbonyl}piperidin-4-ol
6-[3-(4-methylphenyl)propanoyl]-N-[3-(2-oxoimidazolidin-1-yl)phenyl]-6-azaspiro[2.5]octane-1-carboxamide
1-[3-(3-fluoro-4-phenylbenzoyl)piperidin-1-yl]pentane-1,4-dione
2-fluoro-N-[(3-methoxyphenyl)methyl]-N-(prop-2-en-1-yl)-5-sulfamoylbenzamide
N-(4-methoxy-3-pentanamidophenyl)-1H-1,2,4-triazole-5-carboxamide
1-(2-methylpropyl)-N-[2-(pyridin-3-yloxy)phenyl]pyrrolidine-2-carboxamide
(1R,5S,8S)-N-[4-(4-fluorophenoxy)phenyl]-8-methoxy-3-azabicyclo[3.2.1]octane-3-carboxamide
5-methyl-1'-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-[furan-2-yl(phenyl)methyl]-3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)propanamide
2-(3,4-difluorophenyl)-N-({3-[(4-methoxyphenyl)methyl]-4,5-dihydro-1,2-oxazol-5-yl}methyl)acetamide
3-(4-fluoro-3-methylphenyl)-6-[2-(morpholin-4-yl)propanoyl]-1-(pyridin-3-ylmethyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
7-(cyclopropylmethyl)-2-(6-methylquinoline-4-carbonyl)-2,7-diazaspiro[4.5]decane
8-(1-methyl-1H-pyrrole-2-carbonyl)-2-(2-methylpropyl)-2,8-diazaspiro[4.5]decan-3-one
N-(4-ethenylphenyl)-2-(pyrrolidin-1-ylmethyl)piperidine-1-carboxamide
3-methyl-1-phenyl-2-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carbonyl]-1,2-diazinane
1-{1-[(1-cycloheptanecarbonylpiperidin-4-yl)methyl]-1H-1,2,3-triazol-4-yl}propan-2-ol
N-[(2-fluorophenyl)methyl]-2-{[1-(3-methylpyridin-2-yl)propan-2-yl]amino}acetamide
ethyl 5-(1-benzylpyrrolidin-3-yl)-1-(2-hydroxyethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-ethyl-1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-[3-(dimethyl-1,3-thiazol-2-yl)propyl]-1-[4-(methylsulfanyl)phenyl]urea
3-(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)-1-[(3S,4R)-3-(dimethylamino)-4-(propan-2-yl)pyrrolidin-1-yl]propan-1-one
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-{[7-(pyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
methyl 1-[3-(2-chlorophenyl)-3-phenylpropanoyl]piperidine-4-carboxylate
(4aS,8aR)-1-[3-(1H-imidazol-1-yl)propyl]-6-[2-(5-methyl-3-oxo-2,3-dihydro-1H-pyrazol-4-yl)acetyl]-decahydro-1,6-naphthyridin-2-one
4-(1-cycloheptyl-6-oxopiperidine-3-carbonyl)-1-cyclopentylpiperazin-2-one
N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-N-methyl-2-(2,6,6-trimethyl-4-oxo-1-propyl-4,5,6,7-tetrahydro-1H-indol-3-yl)acetamide
1-[2-(2-chloro-6-fluorophenyl)acetyl]-4-[(3-methoxyphenyl)methyl]-1,4-diazepan-5-one
4-[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]-1-(pyridin-2-ylmethyl)pyrrolidin-2-one
(3S,4R)-4-(hydroxymethyl)-1-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}piperidin-3-ol
1-(2-methoxyethyl)-3-(2-methyl-2,3-dihydro-1-benzofuran-5-yl)-1-[(2-methylphenyl)methyl]urea
1-cyclopentyl-N-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-6-oxopiperidine-3-carboxamide
N-(4-chloro-2-methoxy-5-methylphenyl)-4-(pyrimidin-2-yl)-1,4-diazepane-1-carboxamide
2-[1-(thiophen-2-ylmethyl)-4-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-yl]ethan-1-ol
1-{2-[(3,5-dimethylphenyl)methyl]-2,7-diazaspiro[4.5]decan-7-yl}butan-1-one
7-cyclohexyl-2-[(3,5-dimethyl-4-oxo-1,4-dihydropyridin-2-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
N-({4-methyl-5-[(2-methylpropyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)thiophene-2-carboxamide
N,N-diethyl-8-methyl-2,8-diazaspiro[4.5]decane-2-sulfonamide
2-butoxy-1-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}ethan-1-one