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5-benzyl-N-[1-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
1-{2-oxo-2-[4-(piperidine-1-carbonyl)piperidin-1-yl]ethyl}-1,2-dihydropyrimidin-2-one
(4aS,7aR)-1-[2-hydroxy-4-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(2R,3R)-2-hydroxy-1'-[(1-phenyl-1H-pyrazol-4-yl)methyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-phenylacetamide
5-methyl-5-{1-[2-(4-phenylphenyl)acetyl]piperidin-4-yl}-3-(pyridin-4-ylmethyl)imidazolidine-2,4-dione
1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-1-yl]-2-[(2-methylphenyl)sulfanyl]ethan-1-one
1,5-dimethyl-4-{octahydro-1H-pyrido[1,2-a]piperazin-2-ylmethyl}-1H-pyrazole
1-benzyl-4-({2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)pyrrolidin-2-one
N-[(2R,3R)-2-(pyridin-3-ylmethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-1H-pyrazole-3-carboxamide
2-methoxy-N,N-bis(propan-2-yl)-6-(5-propanoylthiophen-2-yl)benzamide
2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-1-{4-[1-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}ethan-1-one
2-{2-[2-(2-aminoethyl)morpholin-4-yl]-2-oxoethyl}-2,3-dihydro-1,2-benzothiazol-3-one
N-[2-(4-methoxyphenyl)propan-2-yl]-2-[1-(3-methylbut-2-en-1-yl)-3-oxopiperazin-2-yl]acetamide
1-{3-fluoro-5-methylimidazo[1,2-a]pyridine-2-carbonyl}-2-(3-methoxyphenyl)azetidine
(3S,4S)-1-{6-chloroimidazo[1,2-a]pyridine-2-carbonyl}-4-(4-fluorophenyl)piperidin-3-ol
{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}(pyridin-2-ylmethyl)amine
N-(oxolan-2-ylmethyl)-1-{1-[(2E)-3-phenylprop-2-en-1-yl]piperidin-4-yl}piperidine-4-carboxamide
3-chloro-2-[3-(1H-imidazol-1-ylmethyl)piperidin-1-yl]pyridine
1-[(2-fluorophenyl)methyl]-4-{1-[(4-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-1,4-diazepane
3-{2-[(2-fluoro-4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[3-(1H-pyrazol-1-yl)propyl]propanamide
2-amino-4-[2-(furan-2-yl)pyrimidin-5-yl]-6,8-dimethyl-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxy-N-(oxolan-3-ylmethyl)benzamide
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(2-methoxyacetyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3-[(1-{5-[2-(methylsulfanyl)ethyl]-4-phenyl-1H-imidazol-1-yl}propan-2-yl)oxy]pyridine
1-[(3-fluorophenyl)methyl]-N-methyl-6-oxo-N-(1H-pyrazol-5-ylmethyl)piperidine-3-carboxamide
5-methyl-4-(2-{2-methyl-2,8-diazaspiro[4.5]decan-8-yl}-2-oxoethyl)-2,3-dihydro-1H-pyrazol-3-one
4-[(2-chlorophenyl)methyl]-1-(quinolin-8-ylmethyl)-1,4-diazepan-5-one
3-(4-methoxyphenyl)-N-[(3-methylpyridin-2-yl)methyl]prop-2-ynamide
1,2,2-trimethyl-4-{[3-(methylsulfanyl)phenyl]methyl}piperazine
3-(1-{1-[(4-fluorophenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-1-(2-methylphenyl)urea
N-(4-methoxy-2-methylphenyl)-3-[1-(pyridin-2-yl)piperidin-3-yl]propanamide
(3aR,6aR)-2-(3-methoxy-5-methylthiophene-2-carbonyl)-5-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-(oxolan-2-ylmethyl)-1-(pyrimidin-2-yl)-N-(thiophen-3-ylmethyl)piperidine-4-carboxamide
2-(6-{4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazin-1-yl}pyrimidin-4-yl)ethan-1-amine
ethyl 4-{1-[(3-fluorophenyl)methyl]-6-oxopiperidine-3-carbonyl}piperazine-1-carboxylate
5-{[(3S,4R)-3-(dimethylamino)-4-propylpyrrolidin-1-yl]methyl}-2-methoxyphenol
1-{3-[benzyl(methyl)amino]piperidin-1-yl}-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
N-cyclopentyl-2-[3-oxo-1-(3-phenylpropyl)piperazin-2-yl]acetamide
1-[(1S,5R)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-phenoxypropan-1-one
N-{2-[5-(1H-imidazol-2-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}-4-methylpyridin-2-amine
1-[2-({[2-(pyrazin-2-yl)ethyl]amino}methyl)phenoxy]-3-(thiomorpholin-4-yl)propan-2-ol
ethyl 3-[(2,4-difluorophenyl)methyl]-1-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}piperidine-3-carboxylate
3-(1H-1,2,3-benzotriazol-1-yl)-N-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}propanamide
N-[(2R,3R)-1'-[(2-chlorophenyl)methyl]-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-phenylacetamide
N-{1-[(3-methoxyphenyl)methyl]piperidin-3-yl}-1-propyl-1H-pyrazole-5-carboxamide
6-[(5-ethylfuran-2-yl)methyl]-N-(2-methyl-1,3-benzothiazol-5-yl)-6-azaspiro[2.5]octane-1-carboxamide
N-(butan-2-yl)-6-(3-fluorophenyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
2-(6-methoxynaphthalen-2-yl)-4-{6-methylthieno[2,3-d]pyrimidin-4-yl}morpholine
[(3R,4R)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-1-(5-methylpyridine-2-carbonyl)pyrrolidin-3-yl]methanol
{[2-(benzylsulfanyl)pyrimidin-5-yl]methyl}[(1,3-dimethylpyrrolidin-3-yl)methyl]methylamine