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methyl 3-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-7-oxo-9-(propan-2-yloxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
4-methyl-N-[(4-methyl-1,3-benzoxazol-2-yl)methyl]pyrimidin-2-amine
(2S)-1-{[6-(azocane-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}pyrrolidine-2-carboxamide
N-[2-(1H-indol-3-yl)ethyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-3-amine
N-{[5-fluoro-7-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(3-methoxyphenyl)propanamide
1-{4-[(4-methoxy-3-{[1-(4-phenylbenzoyl)piperidin-4-yl]oxy}phenyl)methyl]piperazin-1-yl}ethan-1-one
(1S,5R)-3-[(4-methoxyphenyl)methyl]-6-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
3-chloro-N-{[4-(4-fluorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}benzamide
5-methyl-4-[(2-phenylethyl)amino]-N-(prop-2-en-1-yl)thieno[2,3-d]pyrimidine-6-carboxamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-{1,9-dioxaspiro[5.5]undecan-4-yl}piperazine
N3-cyclohexyl-1-(2-methylpropyl)-4-oxo-N5-[2-(pyridin-4-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
3-[4-(2-cyanophenyl)-3-oxopiperazin-1-yl]-N-[(2-fluorophenyl)methyl]propanamide
5-{3-[2-(4-methoxyphenyl)ethyl]piperidine-1-carbonyl}-2-(propan-2-yl)-3,4-dihydropyrimidin-4-one
1-[2-(cyclopent-2-en-1-yl)acetyl]-4-[3-(propan-2-yl)-1H-pyrazol-1-yl]piperidine-4-carboxylic acid
{1-[6-(dimethylamino)pyrimidin-4-yl]piperidin-3-yl}methanol
2-{1-cyclopentyl-4-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]piperazin-2-yl}ethan-1-ol
N-(isoquinolin-5-ylmethyl)-N-methyl-1-{[3-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
2-[3-(2-chlorophenyl)-1-[2-(dimethylamino)ethyl]-2,5-dioxopyrrolidin-3-yl]-N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-N-methylacetamide
[(3R,4R)-1-[(2-aminopyridin-3-yl)methyl]-4-[(dimethylamino)methyl]pyrrolidin-3-yl]methanol
N-methyl-5-(1-oxo-2,3-dihydro-1H-isoindol-2-yl)-N-[(5-propyl-1H-pyrazol-3-yl)methyl]pentanamide
2-fluoro-N-{3-[3-(1H-imidazol-1-ylmethyl)piperidin-1-yl]-3-oxopropyl}benzamide
methyl 1-(2-methylpropyl)-5-{[(5-methylthiophen-2-yl)methyl]amino}-3-(pyridine-3-amido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
(1S,5R)-6-(cyclopropylmethyl)-3-[4-(4-methylphenyl)-4-oxobutyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
4-[(4-chloro-3-fluorophenyl)methyl]-1,3λ6,4-oxathiazinane-3,3-dione
5-cyclobutyl-1-(propan-2-yl)-3-(thiophen-2-ylmethyl)-1H-1,2,4-triazole
1-(2-methoxyethyl)-8-[(4-methyl-1H-imidazol-5-yl)methyl]-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(6-methylpyridin-3-yl)-1-(quinoline-2-carbonyl)piperazine-2-carboxamide
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(2-phenoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-methoxy-1-(1'-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl)ethan-1-one
3-[1-(3-chloro-4-fluoro-1-benzothiophene-2-carbonyl)azetidin-3-yl]pyridine
3-{[4-(2-ethoxyphenyl)piperazin-1-yl]methyl}-7-fluoro-1-[(3-methoxyphenyl)methyl]-1,2-dihydroquinolin-2-one
N-cyclopentyl-5-methyl-4-(4-methylpiperazin-1-yl)thieno[2,3-d]pyrimidine-6-carboxamide
{[2-(ethanesulfonyl)-1-(3-phenylpropyl)-1H-imidazol-5-yl]methyl}(methyl)(2-methylprop-2-en-1-yl)amine
N-(2-acetamidophenyl)-2-[(1S,5R)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]acetamide
2-(dimethylamino)-N-ethyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-(3-methylphenyl)acetamide
5-[(3,4-dimethoxyphenyl)methyl]-5-{3-[3-(4-methylphenoxymethyl)piperidin-1-yl]-3-oxopropyl}pyrrolidin-2-one
5-{[4-(3-methylphenoxy)piperidin-1-yl]methyl}-N-(oxolan-2-ylmethyl)pyrimidin-2-amine
3-({[2-(hydroxymethyl)quinazolin-4-yl]amino}methyl)-1,2,4-oxadiazole-5-carboxamide
1-(cyclopropylmethyl)-N-ethyl-5-[(1-methyl-1,2,3,4-tetrahydroquinolin-6-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(3aR,7aS)-N-(1,3,6-trimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)-2,3,3a,4,7,7a-hexahydro-1H-isoindole-2-carboxamide
N-({7-[2-(3-chlorophenoxy)propanoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(thiophen-3-yl)acetamide
N-[4-({[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]carbamoyl}methyl)phenyl]butanamide
6-[(dimethyl-1,2-oxazol-4-yl)methoxy]-1-(2-methylpropyl)-4-[1-(propan-2-yl)piperidin-4-yl]-1,4-diazepan-2-one
2-(3,4-dimethylphenyl)-2-{methyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}acetic acid
(1S,4S)-2-{6-[4-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carbonyl}-2-azabicyclo[2.2.1]heptane
N-(2-cyclobutyl-1-methyl-7-{4-[(3-methylpyridin-2-yl)methyl]piperazine-1-carbonyl}-1H-1,3-benzodiazol-5-yl)-2-methoxyacetamide
N-({3-methoxy-4-[2-(pyridin-2-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]cyclopropanecarboxamide
1-{[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl}piperidine-2-carboxamide
3-[4-(2-ethoxyethyl)piperazine-1-carbonyl]-N-[(4-methylphenyl)methyl]aniline
1-methyl-3-(2-methylpropyl)-N-[2-(5-phenyl-1,2,4-oxadiazol-3-yl)ethyl]-1H-pyrazole-5-carboxamide