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2-methoxy-N-{1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-4-(4H-1,2,4-triazol-4-yl)benzamide
1-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}azonan-2-one
5-[3-(3-methoxyphenyl)benzoyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
4-{[7-methyl-2-(thiophen-2-yl)quinolin-3-yl]methyl}morpholine-2-carboxamide
N-[(2R,3R)-2-ethoxy-1'-[2-(3-methyl-1H-1,2,4-triazol-5-yl)acetyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-3-carboxamide
N-[(2S,4R,6S)-2-(2,6-difluorophenyl)-6-(2-phenylethyl)oxan-4-yl]acetamide
1-[1-(methoxymethyl)cyclobutanecarbonyl]-4-phenylpiperidine-4-carbonitrile
1,3-dimethyl-5-({[4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-yl]amino}methyl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
4-{3-[4-(furan-2-carbonyl)piperazine-1-carbonyl]piperidin-1-yl}-2-[(4-methoxyphenyl)methyl]-2,3-dihydro-1H-isoindole-1,3-dione
{[2-(4-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}[1-(3-methoxyphenyl)ethyl]methylamine
8-(3-fluoro-4-methoxybenzoyl)-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}({[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl})amine
1-[4-(4-{[(2,3-dimethoxyphenyl)methyl]amino}piperidin-1-yl)benzoyl]piperidin-3-ol
N-{[3-methyl-7-(4-methylbenzoyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}thiophene-3-sulfonamide
N-{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
1-{[3-phenyl-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}azepan-2-one
2-(2-fluoro-6-methoxyphenyl)-6-methylpyridine-3-carbonitrile
(1R,2R,6S,7S)-4-(5-methoxy-1H-indazole-3-carbonyl)-4-azatricyclo[5.2.1.02,6]decane
N-cyclopropyl-5-(4-fluorobenzoyl)-1-[2-(4-methoxyphenyl)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-(2-chlorophenyl)-1-(2-methoxyethyl)-3-{2-[4-(2-methoxyethyl)piperazin-1-yl]-2-oxoethyl}pyrrolidine-2,5-dione
1-[2-(2-chlorophenyl)ethyl]-2-(methoxymethyl)-N,6-dimethyl-4-oxo-N-[1-(thiophen-2-yl)ethyl]-1,4-dihydropyridine-3-carboxamide
5-(furan-2-yl)-1-phenyl-1H,4H-pyrazolo[3,4-d]imidazole
1-methyl-4-{1-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-1H-imidazol-2-yl}piperidine
N-[2-(1,3-benzoxazol-2-ylsulfanyl)ethyl]-3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carboxamide
N-{4-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrole-5-carbonyl]phenyl}ethane-1-sulfonamide
N-[5-({7-[(4-hydroxypiperidin-1-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}methyl)thiophen-2-yl]acetamide
3-(piperidin-3-yl)-N-[2-(pyridin-2-ylsulfanyl)ethyl]benzamide
2-{[1-(adamantan-1-yl)piperidin-4-yl]oxy}-4-methoxy-N-(2-methoxyethyl)benzamide
5-(3,3-dimethylbutanoyl)-1-(2-phenylethyl)-N-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-3-azaspiro[5.5]undecan-9-amine
2-[4-(1-ethoxyethyl)phenyl]-N,N-dimethylpyrimidin-4-amine
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-2-(morpholin-4-yl)benzamide
5-(4-chloro-3,5-dimethylphenoxymethyl)-N-ethyl-N-(oxolan-2-ylmethyl)-1,2-oxazole-3-carboxamide
N-[(5-{[2-(dimethylamino)ethyl]sulfanyl}-4-(3-methoxyphenyl)-4H-1,2,4-triazol-3-yl)methyl]cyclohexanecarboxamide
N-[(5-chloro-3-methyl-2-phenyl-1H-indol-7-yl)methyl]-5-methyl-1,3-oxazole-4-carboxamide
5-propyl-N-[2-(1H-1,2,4-triazol-1-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
1-(4-{[4-(azepan-1-ylmethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)-4-methylpentan-1-one
N-[2-(4-ethyl-1,3-thiazol-2-yl)ethyl]-5-oxo-1-(propan-2-yl)pyrrolidine-3-carboxamide
(1-{4-[(2H-1,3-benzodioxol-5-ylmethyl)amino]-5-methylthieno[2,3-d]pyrimidine-6-carbonyl}piperidin-2-yl)methanol
6-{[3-(3-methoxybenzoyl)piperidin-1-yl]methyl}quinoline
6-methyl-4-(4-methyl-1H-imidazol-5-yl)-5-[3-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1,2,3,4-tetrahydropyrimidin-2-one
N-({8-[(3,4-difluorophenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-1-methyl-1H-pyrazole-5-carboxamide
3-(3,5-dimethyl-1H-pyrazol-4-yl)-N-[2-(phenylcarbamoyl)ethyl]propanamide
3-[(1-cyclopentylpiperidin-4-yl)oxy]-N-[(1R)-1-(4-methoxyphenyl)ethyl]benzamide
5-amino-3-(2-chloro-4-hydroxyphenyl)-1,6-diazatricyclo[6.2.2.02,7]dodeca-2,4,6-triene-4-carbonitrile
1-[1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-4-(propan-2-yl)-1,4-diazepane
1-(1,3-benzoxazol-2-yl)-N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}piperidin-4-amine
2-(2-hydroxypropanoyl)-N-(pyridin-3-yl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
N-{1-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-3-(5-methyl-1H-pyrazol-1-yl)propanamide