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2-{1-ethyl-2,5-dioxo-3-[3-(trifluoromethyl)phenyl]pyrrolidin-3-yl}-N-methyl-N-(oxan-4-yl)acetamide
3-chloro-N-({3-[(4-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazol-5-yl}methyl)thiophene-2-carboxamide
5-[1-(2-methylbenzoyl)piperidin-4-yl]-3-(oxolan-2-ylmethyl)-5-propylimidazolidine-2,4-dione
N-[2-(7-{[4-(2-hydroxyethoxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]-2,4-dimethylbenzamide
6-(3,4-difluorophenyl)-9H-purin-2-amine
methyl 4-[({1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}amino)methyl]benzoate
N-(1,1-dioxo-1λ6-thian-4-yl)-N-methyl-4-(piperidin-1-ylmethyl)benzamide
2-(4-{[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]methoxy}phenyl)acetamide
4-(5-fluoro-2-methylbenzenesulfonyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
N-[(1R,2S)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-4-(piperidin-1-ylmethyl)benzamide
N5-cyclooctyl-N3-methyl-4-oxo-N3-(propan-2-yl)-1-[2-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
(3S,4R)-4-(3-methylthiophen-2-yl)-1-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-3-carbonyl}piperidin-3-ol
N-[(1R)-1-(4-fluorophenyl)ethyl]-4-[4-(hydroxymethyl)-1H-1,2,3-triazol-1-yl]piperidine-1-carboxamide
3-(1H-pyrazol-1-yl)-N-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}benzamide
2-[3-(1-methoxyethyl)phenyl]-4,6-dimethylpyridine-3-carboxamide
6-methoxy-N-{[3-(pyrimidin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
4-[(3-methoxyphenyl)methyl]-1-[(2E)-2-methylbut-2-en-1-yl]-1,4-diazepan-5-one
3-{2-[(2-fluoro-4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[(2-fluorophenyl)methyl]propanamide
2-{[2-(cyclopropylmethyl)-7-(pyridin-3-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]amino}ethan-1-ol
6-(benzyloxy)-4-[5-(methoxymethyl)furan-2-carbonyl]-1-(pyridin-3-ylmethyl)-1,4-diazepan-2-one
3-(2-benzyl-5-oxopyrrolidin-2-yl)-N-[3-(1H-pyrazol-1-yl)propyl]propanamide
ethyl 2-[1-(5-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-1H-pyrazole-3-carbonyl)piperidin-2-yl]acetate
(1,4-dioxan-2-ylmethyl)({[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl})methylamine
N-[2-(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-2-fluorobenzamide
2-methyl-N-(2-phenylpropyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-[(2,4-dimethoxy-3-methylphenyl)methyl]-3,4-dihydro-2H-1-benzopyran-3-amine
N-[(2-chlorophenyl)methyl]-3-[1-(pyrrolidine-1-carbonyl)piperidin-3-yl]propanamide
[(3-{[1-(furan-3-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl](methyl)[(1-methyl-1H-pyrazol-4-yl)methyl]amine
1-(cyclopropylmethyl)-6-[5-(methoxymethyl)furan-2-carbonyl]-3-(2-methylquinolin-5-yl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
N-[2-methyl-2-(morpholin-4-yl)propyl]-4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}butanamide
2-{[(2-methoxyethyl)(thiophen-2-ylmethyl)amino]methyl}-6-methylphenol
2-(dimethylamino)-2-(3-fluorophenyl)-N-[2-(2-oxopyrrolidin-1-yl)ethyl]acetamide
2-(5-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl)pyridine
6-methyl-N-{[4-(morpholin-4-yl)phenyl]methyl}pyridazin-3-amine
4-(2-phenoxybenzoyl)-1,8-dioxa-4,11-diazaspiro[5.6]dodecane
7-{[4-(2-methoxyacetyl)-1,4-diazepan-1-yl]methyl}-4-methyl-2H-chromen-2-one
(2S)-2-[4-(4-chloro-1-methyl-1H-indazol-3-yl)-1H-1,2,3-triazol-1-yl]-4-methylpentan-1-ol
5-[3-(1H-1,3-benzodiazol-5-yl)-1,2,4-oxadiazol-5-yl]-1-ethylpiperidin-2-one
8-[3-(1H-imidazol-1-yl)propyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
2-{1-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl}ethan-1-ol
5-methyl-N-(2-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)pyridine-3-carboxamide
2-(2,3-dimethylphenoxy)-1-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]ethan-1-one
6-methoxy-3-[4-(pyridin-4-yl)piperidine-1-carbonyl]-1,4-dihydroquinolin-4-one
N-[(3-ethoxyphenyl)methyl]-2-(3-fluorophenoxy)-N-(2-hydroxyethyl)acetamide
2,6-dimethyl-N-[3-(1H-1,2,3,4-tetrazol-5-yl)propyl]quinoline-3-carboxamide
1-(1-{[2-(methylsulfanyl)phenyl]methyl}piperidin-4-yl)-2-phenylethan-1-ol
2,6-dimethyl-N-[2-(4H-1,2,4-triazol-4-yl)ethyl]quinoline-4-carboxamide
1-[(4-fluorophenyl)methyl]-5-(2-methoxyacetamido)-N-(oxolan-2-ylmethyl)-N-propyl-1H-1,3-benzodiazole-7-carboxamide
7-(propan-2-yl)-2-[2-(2,2,3,3-tetrafluoropropoxy)acetyl]-2,7-diazaspiro[4.5]decan-6-one
1-(2-chlorobenzenesulfonyl)-N-methyl-N-[2-(pyridin-2-yl)ethyl]piperidin-3-amine