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1-[(1-cyclopropyl-1H-imidazol-5-yl)methyl]-4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine
(3S,4R)-4-methyl-1-(5,6,7,8-tetrahydronaphthalene-2-carbonyl)piperidine-3,4-diol
N-[2-ethyl-4-(2-methoxypyridin-3-yl)phenyl]acetamide
4-[5-methyl-4-(1-methyl-1H-pyrazol-4-yl)-1H-imidazol-2-yl]-1-(pyridin-2-ylmethyl)pyrrolidin-2-one
methyl 4-{6-[(3-fluorophenyl)methoxy]-4-(2-methylpropyl)-3-oxo-1,4-diazepan-1-yl}-4-oxobutanoate
4-[2-(dimethylamino)-4-methylpyrimidine-5-carbonyl]-1-[(4-methylphenyl)methyl]piperazin-2-one
N-{[2-chloro-5-(trifluoromethyl)phenyl]methyl}-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
2-{[7-(1-ethylpiperidine-3-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]amino}ethan-1-ol
N-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-amine
N-[(2-ethoxypyridin-3-yl)methyl]-3-(1,2-oxazinan-2-yl)propanamide
N-{[7-methoxy-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}-3-(2-methoxyphenyl)-N-(oxolan-2-ylmethyl)propanamide
1-ethyl-5-[ethyl(2-methylprop-2-en-1-yl)amino]-N-(furan-3-ylmethyl)-N-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-cyclohexyl-4-{1-[(2E)-3-phenylprop-2-en-1-yl]-1H-1,2,3-triazole-4-carbonyl}-1,4-diazepane
9-[2-(3-methoxyphenoxy)acetyl]-2-methyl-2,9-diazaspiro[5.5]undecan-3-one
4-({[2-(2,3-difluoro-4-methylphenoxy)pyridin-3-yl]methyl}carbamoyl)pyridin-1-ium-1-olate
1-{1-[(4-fluorophenyl)methyl]piperidin-3-yl}-3-(1-oxo-1,3-dihydro-2-benzofuran-5-yl)urea
7-methoxy-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
1-(1-{[5-(oxan-2-yl)thiophen-2-yl]methyl}piperidin-4-yl)-N-(propan-2-yl)piperidine-4-carboxamide
{3-[(2-fluorophenyl)methyl]-1-[(4-phenyl-1,3-thiazol-2-yl)methyl]piperidin-3-yl}methanol
3-phenyl-7-(2-phenylpropyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
5-cyclopropyl-N-{[4-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-1,3-oxazole-4-carboxamide
N-{[5-chloro-7-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzamide
1-(furan-2-ylmethyl)-N-[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]piperidine-4-carboxamide
N-({5-[(3-ethoxyphenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)acetamide
8-(2-methoxyacetyl)-3-(2-phenylethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-{3-[(2S)-2-(methoxymethyl)pyrrolidine-1-carbonyl]benzenesulfonyl}-4-methyl-1,2,3,6-tetrahydropyridine
1-[4-(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)ethan-1-one
N'-(4-methylphenyl)-N-[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]propanediamide
2-{[4-(1H-pyrazol-1-yl)phenyl]methyl}benzene-1-sulfonamide
1-{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}-4-(furan-2-carbonyl)-1,4-diazepane
1-{[4-(4-fluorophenyl)-1,3-thiazol-2-yl]methyl}-4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazine
(1R,2S,9R)-11-[6-(4-hydroxypiperidin-1-yl)pyrimidin-4-yl]-7,11-diazatricyclo[7.3.1.02,7]tridecan-6-one
3-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1-[3-(5-ethyl-4H-1,2,4-triazol-3-yl)phenyl]urea
2-{3-[3-(2,6-dimethylphenoxy)azetidine-1-carbonyl]phenyl}-1H-imidazole
N-[3-(dimethylamino)propyl]-N-methyl-1-[3-(1,3-thiazol-4-yl)phenyl]piperidin-4-amine
2-methyl-N-{1-[7-(2-methylpropyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}benzamide
2-butyl-N-(oxan-4-yl)-1,3-benzoxazole-5-carboxamide
1-{1-[(3-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-4-[(2E)-3-phenylprop-2-en-1-yl]piperazine
N-butyl-N-(furan-2-ylmethyl)-5-(methoxymethyl)furan-2-carboxamide
N-cyclohexyl-2-(methoxymethyl)-6-methyl-4-oxo-1-(3-phenylpropyl)-1,4-dihydropyridine-3-carboxamide
[(2-fluoro-3-methoxyphenyl)methyl](methyl){[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
2-hydroxy-N-{2-[5-(hydroxymethyl)-1,2,4-oxadiazol-3-yl]ethyl}-4-(methylsulfanyl)butanamide
8-cyclopropanecarbonyl-2-(1H-indole-2-carbonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
8-[(2-methoxynaphthalen-1-yl)methyl]-1-(2-methylpropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-methyl-N-[2-(oxan-2-yl)ethyl]-2H-1,3-benzodioxole-5-carboxamide
(4aS,8aR)-1-(3-hydroxypropyl)-6-(quinolin-2-yl)-decahydro-1,6-naphthyridin-2-one
(4aR,7aS)-1-methanesulfonyl-4-(2-phenylacetyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}benzonitrile
5-({[(1-ethyl-1H-imidazol-2-yl)methyl](methyl)amino}methyl)-N,N-dimethylpyridin-2-amine
N-(2-hydroxypropyl)-5-(2-methoxyphenoxymethyl)-N-methyl-1H-pyrazole-3-carboxamide