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(8R,9aS)-8-hydroxy-2-[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]-octahydro-1H-pyrido[1,2-a]piperazine-1,4-dione
[(5-chloro-2,4-dimethoxyphenyl)methyl][(1-ethyl-1H-imidazol-2-yl)methyl]methylamine
1-(1-benzofuran-2-ylmethyl)-4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine
[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl](methyl)[3-(oxolan-2-yl)propyl]amine
2-(1-{[2-(furan-2-yl)pyrimidin-5-yl]methyl}piperidin-3-yl)-4-methyl-1H-1,3-benzodiazole
methyl (2S,4R)-1-[(2,4-difluorophenyl)methyl]-4-[4-(trifluoromethyl)benzamido]pyrrolidine-2-carboxylate
4-{[3-(2-methoxyphenoxy)azetidin-1-yl]methyl}benzoic acid
1-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-1-yl}-2-[1-(propan-2-yl)piperidin-4-yl]ethan-1-one
2-[2-(3-methoxyphenoxy)ethyl]benzene-1-sulfonamide
1-cyclopropyl-4-[4-(1H-pyrazol-1-ylmethyl)piperidine-1-carbonyl]pyrrolidin-2-one
3-[(2-fluorophenyl)methyl]-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidine-3-carboxylic acid
2-{4-[2-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)acetyl]morpholin-3-yl}-N-(6-methylpyridin-3-yl)acetamide
1-(7-methoxy-4-methylquinazolin-2-yl)-N-methyl-N-(thiophen-3-ylmethyl)piperidine-3-carboxamide
methyl 3-{[(3-methoxyphenyl)formamido]methyl}-5-[2-(1H-pyrazol-1-yl)acetamido]benzoate
methyl (2S,4S,5R)-1,2-dimethyl-4-{methyl[(3-methyl-1,2-oxazol-5-yl)methyl]carbamoyl}-5-(2-methylphenyl)pyrrolidine-2-carboxylate
2-(2-hydroxyethyl)-9-[2-(2-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
(2E)-N-(2-{5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(4-fluorophenyl)-4H-1,2,4-triazol-3-yl}ethyl)-3-(3-fluorophenyl)prop-2-enamide
5-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-2-methyl-1,4-dihydropyridin-4-one
3-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}-1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
(2E)-N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-[3-(dimethylamino)propyl]-3-(furan-2-yl)prop-2-enamide
4-(naphthalen-1-ylmethyl)-3-[2-oxo-2-(pyrrolidin-1-yl)ethyl]piperazin-2-one
5-[(2-fluoro-5-methoxyphenyl)methyl]-5-{3-oxo-3-[4-(pyridin-3-yloxy)piperidin-1-yl]propyl}pyrrolidin-2-one
(2E)-3-(4-fluorophenyl)-1-{3-[5-(2-methylphenyl)-2-(pyridin-4-yl)pyrimidin-4-yl]piperidin-1-yl}prop-2-en-1-one
N-ethyl-4-{3-[(pyridin-2-ylmethyl)carbamoyl]piperidin-1-yl}piperidine-1-carboxamide
2-[4-(5-chloro-2-methylphenyl)piperazin-1-yl]-N-(pyrazin-2-yl)acetamide
4-(azepan-1-yl)-N-[2-(1-methylpiperidin-3-yl)ethyl]-4-oxobutanamide
2-(1-{[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl}pyrrolidin-2-yl)pyridine
N-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]-1-phenyl-1H-1,2,3-triazole-5-carboxamide
N-(2-methoxyethyl)-N-methyl-3-(2-methylphenyl)-3-phenylpropanamide
(5S,9aS,9bS)-5-(2-fluoro-5-methoxyphenyl)-2-[(4-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
4-{[(3S,4S)-3-carboxy-4-(pyridin-2-yl)pyrrolidin-1-yl]methyl}-1H-pyrazole-3-carboxylic acid
1-[cyclohexyl(methyl)amino]-3-(2-methoxy-4-{[methyl(1,2-oxazol-3-ylmethyl)amino]methyl}phenoxy)propan-2-ol
5-chloro-N-{2-[(pyridin-3-yl)amino]ethyl}thiophene-2-carboxamide
N,1-dimethyl-N-[2-(4-methylpiperidin-1-yl)ethyl]-1H-indole-2-carboxamide
2-methyl-1-(1-{3-[(2-methylprop-2-en-1-yl)oxy]benzoyl}azetidin-3-yl)piperidine
N-[2-(3-ethylphenoxy)ethyl]-N-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
6-ethyl-N-[2-(1H-imidazol-1-yl)ethyl]-2-methylquinoline-4-carboxamide
N-[2-(2-fluorophenoxy)ethyl]-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
5-(3-cyclopropyl-1-propyl-1H-1,2,4-triazol-5-yl)-4-propylpyrimidine
N-(2-hydroxyethyl)-5-(4,5,6,7-tetrahydro-1,3-benzothiazole-2-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
ethyl 5-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-1-(2-methylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
4-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridin-2-amine
1-(2-{5-[(benzyloxy)methyl]-4-phenyl-1H-imidazol-1-yl}ethyl)pyrrolidin-2-one
2-[1-cyclopropyl-3-(4-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl]-N-ethyl-N-(pyridin-4-ylmethyl)acetamide
1-[9-methoxy-7-(quinolin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(thiophen-3-yl)ethan-1-one
2-(dimethyl-1,3-thiazol-5-yl)-1-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
N-(1-{1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-phenoxypropanamide
N,N-diethyl-2-oxo-2-[3-(5-oxo-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]acetamide
2-(2,2-diphenylethyl)-4-[(2-methylpyrimidin-5-yl)methyl]morpholine
N-(1-{1-[(4-methoxy-2,5-dimethylphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)pyridine-3-carboxamide