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1-cyclohexyl-3-(cyclopropylmethyl)-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}-2-(methylamino)acetamide
3,3-dimethyl-1-[(3S,4R)-4-(propan-2-yl)-1-[4-(4H-1,2,4-triazol-4-yl)benzoyl]pyrrolidin-3-yl]urea
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)-N,7-dimethylimidazo[1,2-a]pyridine-2-carboxamide
2-{4-[(4-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)methyl]piperazin-1-yl}ethan-1-ol
1-{3-[(4-methoxyphenyl)amino]piperidin-1-yl}-2-(phenylsulfanyl)ethan-1-one
6-(3,5-dimethoxyphenyl)pyridin-2-amine
N-[(5-methylfuran-2-yl)methyl]-4-[(oxolan-3-yl)sulfamoyl]benzamide
N-({1-[(2E)-3-(4-hydroxy-3-methoxyphenyl)prop-2-en-1-yl]piperidin-3-yl}methyl)furan-2-carboxamide
3-{2-[2-(hydroxymethyl)piperidin-1-yl]-2-oxoethyl}-3-phenyl-1-[2-(pyridin-2-yl)ethyl]pyrrolidine-2,5-dione
1-{3-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]propyl}azepane
methyl 3-(furan-3-amido)-1-(2-methylpropyl)-5-[(thian-4-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-(dimethylamino)-2-(4-fluorophenyl)-1-[4-(pyridin-4-ylmethyl)-1,4-diazepan-1-yl]ethan-1-one
methyl 3-{4-[(2S,4R,6R)-6-cyclohexyl-4-acetamidooxan-2-yl]-1H-pyrazol-1-yl}propanoate
N-({[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl](methyl)carbamoyl}methyl)-2-methylpropanamide
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-3-(trimethyl-1H-pyrazol-1-yl)propanamide
(2S)-1-{2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-5-methoxybenzoyl}-4-methyl-2-(propan-2-yl)piperazine
5-[1-(4-methoxybenzoyl)piperidin-4-yl]-5-(pyridin-3-yl)-3-(thiophen-3-ylmethyl)imidazolidine-2,4-dione
dimethyl({[4-methyl-5-(1-{pyrazolo[1,5-a]pyridine-7-carbonyl}piperidin-3-yl)-4H-1,2,4-triazol-3-yl]methyl})amine
3-(dimethyl-1,2-oxazol-4-yl)-N-[(1R,3S)-3-(thiomorpholine-4-carbonyl)cyclopentyl]propanamide
1-{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-methyl-1,4-diazepan-5-one
N-(3-methoxypropyl)-1-methyl-5-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
methyl 3-[(4-ethoxyphenyl)methyl]-7-oxo-9-(pyridin-3-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-{4-[5-(2-chloro-4-methoxyphenoxymethyl)-1,2-oxazole-3-carbonyl]-1,4-diazepan-1-yl}ethan-1-one
2-[2-(1H-imidazol-4-yl)ethyl]-9-[2-(propylsulfanyl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
2-fluoro-6-methoxy-4-{[methyl(quinolin-5-ylmethyl)amino]methyl}phenol
dimethyl[(5-{[4-(pyridin-3-yloxy)piperidin-1-yl]methyl}thiophen-3-yl)methyl]amine
3-[2-(azepan-1-yl)-2-oxoethyl]-1-cyclohexyl-3-(2-fluorophenyl)pyrrolidine-2,5-dione
methyl 2-chloro-4-({[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]carbamoyl}amino)benzoate
2-[(1-methyl-1H-indol-3-yl)sulfanyl]-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}acetamide
N-{imidazo[1,2-a]pyridin-2-ylmethyl}-1-[2-(morpholin-4-yl)ethyl]-6-oxopiperidine-3-carboxamide
3-chloro-N-[2-(dimethylamino)ethyl]-4-{[1-(pyridin-4-ylmethyl)piperidin-4-yl]oxy}benzamide
3-hydroxy-3-{[(2-methanesulfonylethyl)amino]methyl}-1-[(3-methoxyphenyl)methyl]piperidin-2-one
N-{2-azatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-5-yl}-2-(2-{[(furan-3-ylmethyl)(methyl)amino]methyl}-4-(pyrazin-2-yl)phenoxy)acetamide
4-[8-(2-methoxyethyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]pyridine-2-carboxylic acid
1-[(3R,4R)-3-(hydroxymethyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]-2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethan-1-one
(2S,4R)-4-amino-1-(2-amino-4-phenylpyrimidine-5-carbonyl)-N-methylpyrrolidine-2-carboxamide
1-{6-[2-(3,4-dichlorophenyl)morpholin-4-yl]pyridin-3-yl}ethan-1-one
5-[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-3,4-dihydropyrimidin-4-one
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-2-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
(1S,6R)-9-[2-(pyridin-2-yl)acetyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
methyl 4-{4-[(2R)-2-cyclohexyl-2-hydroxyacetyl]piperazin-1-yl}benzoate
3-{[1-(dimethylcarbamoyl)propyl]sulfamoyl}-N-(prop-2-en-1-yl)benzamide
2-(1-benzothiophen-2-ylmethyl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decane
5-{5-[3-(piperidin-1-yl)propyl]-1,2,4-oxadiazol-3-yl}-1H-1,3-benzodiazole
N-[2-(ethanesulfonyl)ethyl]-2-methyl-1-benzofuran-7-carboxamide
(3aS,6aR)-3-[2-(3-chlorophenyl)ethyl]-5-(1H-pyrazole-3-carbonyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
3-[({5-methylpyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]-1,2,4-oxadiazole-5-carboxamide
{[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}(methyl)(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)amine
2-[(3-fluorophenyl)methyl]-6-methyl-1-[3-(morpholin-4-yl)propyl]-3-(pyrrolidine-1-carbonyl)-1,4-dihydropyridin-4-one