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N-({2,3-dimethylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)-3-{2-[(2-fluoro-5-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
N-[2-(2-fluorophenoxy)ethyl]-1-[(3-methoxyphenyl)methyl]-6-oxopiperidine-3-carboxamide
N-[(6-methylpyridin-2-yl)methyl]-6-[4-(trifluoromethyl)benzoyl]-6-azaspiro[2.5]octane-1-carboxamide
1-{[4-(2-phenylpyrrolidine-1-carbonyl)phenyl]methyl}-1H-1,2,3,4-tetrazole
N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-1-[2-(piperidin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-2-[methyl(pyridin-2-ylmethyl)amino]acetamide
1-(dimethylamino)-3-({5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}amino)propan-2-ol
3-[(4-fluorophenyl)methyl]-5-methyl-5-{1-[2-(thiophen-3-yl)acetyl]piperidin-4-yl}imidazolidine-2,4-dione
1-{3,5-dimethyl-4-[2-(4-methylpentyl)morpholine-4-carbonyl]-1H-pyrrol-2-yl}ethan-1-one
2-{1-[2-(1H-imidazol-4-yl)ethyl]-1H-imidazol-2-yl}-1H-1,3-benzodiazole
4-[4-(2-methylphenoxy)piperidine-1-carbonyl]pyridine
4-methyl-2-{1-[1-(1H-pyrazol-1-ylmethyl)cyclopropanecarbonyl]piperidin-4-yl}-1H-1,3-benzodiazole
3-[3-(6-methoxynaphthalene-2-carbonyl)piperidine-1-carbonyl]pyridine
1-cycloheptyl-6-oxo-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]piperidine-3-carboxamide
ethyl 4-benzyl-1-{[5-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}piperidine-4-carboxylate
5-[2-(2,2-diphenylethyl)morpholine-4-carbonyl]-3,4-dihydropyrimidin-4-one
methyl 2-(4-{7-methylimidazo[1,2-a]pyridine-2-carbonyl}-2-oxopiperazin-1-yl)acetate
(3aR,5S,6S,7aS)-2-[5-(pyrrolidin-2-yl)thiophene-2-carbonyl]-octahydro-1H-isoindole-5,6-diol
2-{[4-(2-fluorophenyl)piperazin-1-yl]methyl}-N-[2-(4-methyl-1H-imidazol-2-yl)ethyl]-1,3-oxazole-4-carboxamide
methyl 3-{[3-(3-methyl-1H-pyrazol-1-yl)propanamido]methyl}-5-[3-(trifluoromethyl)benzamido]benzoate
N-{3-hydroxy-1-[4-(propan-2-yl)phenyl]propyl}-[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carboxamide
methyl (2S,4R)-1-[(2,6-difluorophenyl)methyl]-4-(4-methylbenzamido)pyrrolidine-2-carboxylate
2,2-dimethylpropyl (4aS,7aR)-6,6-dioxo-4-(pyridin-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxylate
1-(1-cyclopentanecarbonylpiperidin-3-yl)-4-(2-methoxyphenyl)piperazine
[(3R,4R)-1-[1-(4-methylphenyl)cyclopropanecarbonyl]-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
(2R,3R,6R)-3-(4-methoxyphenyl)-N-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carboxamide
N-[(2R,3R)-1'-[(2,4-dimethoxyphenyl)methyl]-2-(2-methoxyethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
2-benzyl-N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1,3-thiazole-4-carboxamide
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methylbenzamide
2-methyl-4-[1-(2-methyl-1,3-thiazole-4-carbonyl)piperidin-3-yl]-5-(3-methylphenyl)pyrimidine
6-[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]pyridine-3-carboxylic acid
ethyl 4-[(2-chlorophenyl)methyl]-1-[2-(dimethyl-1,2-oxazol-4-yl)acetyl]piperidine-4-carboxylate
1-{[1-butyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}-4-(2-methoxyphenoxy)piperidine
{[3-(2H-1,3-benzodioxol-5-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}(cyclopropylmethyl)(oxolan-2-ylmethyl)amine
(3aS,6aS)-2-benzyl-5-(2-methyl-5-propylpyrimidin-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-hydroxy-N-methyl-2-(pyridin-3-yl)-N-(thian-4-yl)pyrimidine-5-carboxamide
(1S,5R)-N-(4-fluorophenyl)-7-oxo-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
N-[(2R,3R)-1'-(2,2-dimethylpropyl)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methoxybenzamide
2-tert-butyl-6-[3-(propan-2-yloxy)benzoyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
N-(2-methoxyethyl)-N-methyl-3-{5-[(4-phenylphenyl)methyl]-1,3,4-oxadiazol-2-yl}propanamide
4-{3-[(3R,4S)-3-amino-4-cyclopropylpyrrolidine-1-carbonyl]phenyl}-2-methylbutan-2-ol
(2,1,3-benzoxadiazol-5-ylmethyl)[1-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]amine
3-ethyl-6-{1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}-3H-imidazo[4,5-b]pyridin-2-amine
3-(2-{2-[(4-methylphenyl)carbamoyl]acetamido}ethoxy)benzoic acid
2-ethyl-1-{4-[(1-ethyl-1H-imidazol-2-yl)methyl]-1-methyl-1,4,9-triazaspiro[5.5]undecan-9-yl}butan-1-one
N-({3-[(1-methoxypropan-2-yl)oxy]phenyl}methyl)-3-methyl-N-(pyridin-4-ylmethyl)thiophene-2-carboxamide
N-[2-(pyridin-2-ylsulfanyl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-({5-[(2,3-dichlorophenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)acetamide
1-(3,4-dimethoxybenzenesulfonyl)-3-{[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine
N-cyclohexyl-N-methyl-3-{[(5-oxopyrrolidin-2-yl)methyl]sulfamoyl}benzamide