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(1R,3S)-7-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-3-methoxy-7-azaspiro[3.5]nonan-1-ol
2-butyl-4-{[1-(2,3-dimethoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1H-imidazole
N-methyl-5-{[(6-methylpyridin-3-yl)oxy]methyl}-N-[1-(1,2-oxazol-3-yl)ethyl]-1,2-oxazole-3-carboxamide
2-ethoxy-4-{[3-(2-hydroxyethyl)-4-[(3-methoxyphenyl)methyl]piperazin-1-yl]methyl}phenol
N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
1-[(2-fluorophenyl)methoxy]-8-[3-(5-methylfuran-2-yl)benzoyl]-1,8-diazaspiro[4.5]decan-2-one
N-[(2R,3R)-1'-(furan-3-carbonyl)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-phenoxyacetamide
N1,N1-dimethyl-N4-(pyridin-3-yl)piperidine-1,4-dicarboxamide
1-(7-{[3-(methoxymethyl)piperidin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-2-(piperidin-1-yl)ethan-1-one
4-(4-fluorophenyl)-N-{[5-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
2-(3-methyl-1H-pyrazol-1-yl)-1-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
3-(2-methylpropyl)-1-{5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}pyrrolidine
1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-[4-(1H-pyrazol-1-yl)phenyl]piperidine-2-carboxamide
N-cyclopropyl-N-{[2-(2,3-dimethoxyphenyl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}-2-(thiophen-3-yl)acetamide
N-{[5-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-1-methylpiperidine-3-carboxamide
N-(3-phenylpropyl)-2-(pyridin-3-yl)-5,6,7,8-tetrahydroquinazolin-5-amine
3-(7-chloro-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-1-{4-[1-(morpholin-4-yl)ethyl]piperidin-1-yl}propan-1-one
[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)(2-methylpropyl)amine
[4-(2-phenylquinoline-4-carbonyl)-1,4-oxazepan-6-yl]methanol
N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}piperidin-3-amine
1-[2-(1H-imidazol-5-yl)ethyl]-3-methyl-5-[3-(1H-pyrazol-4-yl)propyl]-1H-1,2,4-triazole
5-{[3-ethyl-4-(propan-2-yl)piperazin-1-yl]methyl}-2-(piperidin-1-yl)pyrimidine
1-{1-[(2-chloro-4-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-2-(1,3-thiazol-2-yl)piperidine
N-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}thiolan-3-amine
4-{5-[(3-methoxyphenyl)methyl]-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}piperazin-2-one
3-({ethyl[(1-methyl-1H-imidazol-2-yl)methyl]amino}methyl)-7-methoxy-1,2-dihydroquinolin-2-one
(2S,4S)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-1-[(2-methoxynaphthalen-1-yl)methyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-hydroxy-N-methyl-4-(1H-1,2,3,4-tetrazol-1-yl)benzamide
N-[(4-fluorophenyl)methyl]-N-(oxolan-2-ylmethyl)-2-(2-oxopyrrolidin-1-yl)acetamide
2-[1-(cyclohexylmethyl)-4-{[5-(methoxymethyl)furan-2-yl]methyl}piperazin-2-yl]ethan-1-ol
(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-6-(3-propyl-1H-pyrazole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-(3-{[(2-methylphenyl)methyl]sulfanyl}propyl)-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
2-fluoro-6-{6-[(pyridin-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}benzamide
1-cyclopentyl-4-{3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]propanoyl}piperazin-2-one
1-[3-({[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]amino}methyl)pyridin-2-yl]piperidin-3-ol
4-(dimethyl-1,2-oxazol-4-yl)-3-(1-methyl-1H-pyrazol-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
4-[2-(2-methylphenyl)pyrimidin-5-yl]-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-2-amine
3-[(4-methyl-1,2,3,6-tetrahydropyridin-1-yl)methyl]-2-(morpholin-4-yl)quinoline
N-{[3-(furan-2-ylmethoxy)-4-methoxyphenyl]methyl}-1-methyl-4-oxo-N-(oxolan-2-ylmethyl)-1,4-dihydroquinoline-3-carboxamide
2-[4-(2H-1,3-benzodioxol-5-yl)-2-({methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)phenoxy]-N-cyclohexyl-N-methylacetamide
N-(2-hydroxyethyl)-3-(1H-imidazol-2-yl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]benzamide
N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-3-(pyridin-3-yl)propanamide
4-({8-methylimidazo[1,2-a]pyridin-2-yl}methyl)-1-[2-(naphthalen-2-yl)acetyl]-1,4-diazepan-5-one
2-[5-(1-methyl-1H-imidazol-2-yl)-4-phenyl-1H-imidazol-1-yl]propane-1,3-diol
4-(1-{3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}-2-methylpropan-2-yl)morpholine
4-{1-[1-(hydroxymethyl)cyclopropanecarbonyl]piperidin-3-yl}benzoic acid
N-[(2,5-dimethoxyphenyl)methyl]-4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
N-(3-acetylphenyl)-3-(4-chlorobenzoyl)piperidine-1-carboxamide
2-(4-{[1-(2-chlorophenyl)-1H-pyrazol-4-yl]methyl}-1-(thiophen-3-ylmethyl)piperazin-2-yl)ethan-1-ol
N-cyclopropyl-3-{1-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}propanamide