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2-methyl-9-[(2-oxo-2,3-dihydro-1,3-benzoxazol-5-yl)sulfonyl]-2,9-diazaspiro[5.5]undecan-3-one
N-{[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N,4-dimethylpyridine-3-carboxamide
2-[3-(3-methoxybenzoyl)piperidin-1-yl]pyridine-4-carbonitrile
1-(4-chlorobenzoyl)-N-(4-methoxyphenyl)piperidin-3-amine
3-[(4-methoxyphenyl)methyl]-1-(2-methylpropyl)-8-(quinolin-5-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-(4-{[2-(cyclohex-1-en-1-yl)ethyl]amino}piperidin-1-yl)-N-cyclopentylbenzamide
4-(1-{1-[(2,3-difluoro-4-methoxyphenyl)methyl]piperidin-4-yl}ethyl)morpholine
4-{[4-({1-[4-(4-fluorophenyl)benzoyl]piperidin-3-yl}methoxy)phenyl]methyl}morpholine
2,5-dimethyl-3-{4-[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]piperazin-1-yl}pyrazine
5-(2H-1,3-benzodioxol-4-ylmethyl)-3-(3-methoxyphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
3-(3-methoxyphenyl)-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]benzamide
N-benzyl-N-[(4-methyl-1,3-thiazol-5-yl)methyl]-2-(1H-pyrazol-1-yl)butanamide
4-({3-[3-(4-fluorophenoxy)azetidine-1-carbonyl]-1,2-oxazol-5-yl}methyl)morpholine
4-[2-({3-[(2-oxopyrrolidin-1-yl)methyl]piperidin-1-yl}methyl)-1H-pyrrol-1-yl]benzonitrile
N-methyl-1-[(4-methylphenyl)amino]-N-(1H-pyrazol-5-ylmethyl)cyclopentane-1-carboxamide
7-(2-cyclohexylethyl)-6-oxo-N-(prop-2-en-1-yl)-2,7-diazaspiro[4.5]decane-2-carboxamide
2-(2-{4-[(dimethylamino)methyl]-4-hydroxypiperidin-1-yl}pyrimidin-4-yl)pyridine-4-carboxylic acid
2-(1-{[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]methyl}pyrrolidin-2-yl)-1,3-thiazole
1-ethyl-N-[(4-fluorophenyl)methyl]-5-(2-methoxyacetamido)-2-(pyridin-3-yl)-1H-1,3-benzodiazole-7-carboxamide
5-[6-amino-5-cyano-4-(2-methoxyphenyl)pyridin-2-yl]thiophene-3-carboxylic acid
(3R,4R)-4-(2-ethyl-4-methyl-1H-imidazol-5-yl)-N-[(2-methoxyphenyl)methyl]-1-methylpyrrolidine-3-carboxamide
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(2-methoxyethyl)-N-(propan-2-yl)acetamide
1-ethyl-3-[2-oxo-2-(3-oxopiperazin-1-yl)ethyl]-3-[3-(trifluoromethyl)phenyl]pyrrolidine-2,5-dione
(4aS,8aR)-6-[2-(pyrrolidin-1-yl)acetyl]-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
3-acetamido-N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]benzamide
(3S,7S)-5-(6-methoxyhexanoyl)-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
methyl 1-({4-[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzoyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperidine-2-carboxylate
N-{2-[(2E)-3-(1H-imidazol-4-yl)prop-2-enoyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}-1-phenylcyclopropane-1-carboxamide
3-methoxy-N-({5-methyl-2-[2-(3-phenoxypropanamido)phenyl]-1,3-oxazol-4-yl}methyl)propanamide
4-{[4-(aminomethyl)-1H-1,2,3-triazol-1-yl]methyl}-N-(2-phenylphenyl)piperidine-1-carboxamide
N-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-N-methyl-2-[(4S)-2-oxo-4-(propan-2-yl)-1,3-oxazolidin-3-yl]acetamide
N,N-dimethyl-2-[(1S,5R)-3-[2-(2-methylphenoxy)acetyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
4-[4-(thiophene-2-carbonyl)piperazin-1-yl]-5,6,7,8-tetrahydroquinazolin-2-amine
(3aR,6aR)-2-(cyclobutylmethyl)-5-(2,3-dimethyl-1H-indole-5-carbonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[(2S)-2-aminopropyl]-2-(1H-1,2,4-triazol-3-yl)benzamide
N-[(5-methyl-1,2-oxazol-3-yl)methyl]-4-(1-phenyl-1H-pyrazol-4-yl)pyrimidin-2-amine
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-[4-(1H-pyrazol-1-yl)benzoyl]piperidin-3-amine
2-({4-[(4-fluorophenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)phenol
1-(4-chlorophenyl)-N-{[2-(dimethylamino)-7-methoxyquinolin-3-yl]methyl}-N-(2-methoxyethyl)cyclobutane-1-carboxamide
4-[(1-methyl-1H-pyrazol-4-yl)methyl]-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(3S,4R)-4-(4-methoxyphenyl)-1-(6-methoxypyrimidin-4-yl)-N,N-dimethylpyrrolidin-3-amine
3-[2-(2-fluorophenyl)ethyl]-1-(1-propyl-1H-pyrazole-5-carbonyl)piperidine
N,N-dimethyl-6-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}pyrazine-2-carboxamide
N-[(3S,4R)-1-[2-(4-fluoro-3-methylphenyl)acetyl]-4-(4-methoxyphenyl)pyrrolidin-3-yl]acetamide
1,3-dimethyl-4-[(1S,5R)-7-oxo-6-propyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-1H-pyrazolo[3,4-b]pyridine-5-carboxylic acid
N-[2-(2-fluorophenyl)-1-[1-(1,2,3-thiadiazole-4-carbonyl)piperidin-4-yl]ethyl]-N,2-dimethylfuran-3-carboxamide
(1S,5R)-6-(2-methoxyethyl)-3-{[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
(1-{1-[3-(diphenylmethyl)-1,2-oxazole-5-carbonyl]piperidin-4-yl}piperidin-3-yl)methanol
6-{4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}pyridin-3-ol
6-(aminomethyl)-N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-2-methylpyrimidin-4-amine