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methyl (2S,4R)-4-(4-fluorobenzamido)-1-[(5-methylthiophen-2-yl)methyl]pyrrolidine-2-carboxylate
N-[(2R,3R)-1'-[(3,5-difluorophenyl)methyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
N-cyclohexyl-6-[(diethylamino)methyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
3-[2-(naphthalen-2-ylmethyl)-5-oxopyrrolidin-2-yl]-N-(propan-2-yl)propanamide
N-{[(2S,4S)-4-fluoro-1-(2-methanesulfonylacetyl)pyrrolidin-2-yl]methyl}-2-methylpropanamide
1-{2-oxo-2-[2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]ethyl}-3-(trifluoromethyl)-1,2-dihydropyridin-2-one
2-(5-{2H,4H,5H,6H-cyclopenta[c]pyrazol-2-ylmethyl}-1,2,4-oxadiazol-3-yl)pyrazine
3-(furan-2-yl)-2-[4-(1-methyl-1H-imidazol-2-yl)-1H-1,2,3-triazol-1-yl]propanoic acid
(2S,4S)-1-cyclohexyl-N-ethyl-4-[3-(pyridin-4-yl)propanamido]pyrrolidine-2-carboxamide
2-(2,4-difluorobenzenesulfonyl)-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
N-[1-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(pyridin-2-yl)propanamide
5-(3-methoxyphenoxymethyl)-N-methyl-N-(2,2,6,6-tetramethylpiperidin-4-yl)-1,2-oxazole-3-carboxamide
8-[3-(dimethylamino)-1,2,4-thiadiazol-5-yl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
3-(2,6-dimethylhept-5-en-1-yl)-N-(furan-2-ylmethyl)-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
(3aS,6aS)-2-(cyclopropylmethyl)-1-oxo-5-{[(thiophen-2-ylmethyl)carbamoyl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-(3-methyl-1,2-oxazol-5-yl)-1-[2-(methylamino)-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-6-yl]ethan-1-one
methyl 3-(2-methylbutyl)-7-oxo-9-[2-(2-oxopyrrolidin-1-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-ethyl-1-[(3-methoxyphenyl)methyl]-5-(6-methylpyridine-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-methyl-N-[2-(2-methylphenyl)-1-{1-[5-(2-methylpropyl)-1,2-oxazole-3-carbonyl]piperidin-4-yl}ethyl]-2-(1H-pyrazol-1-yl)acetamide
N-ethyl-2-[2-({methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)-4-(thiophen-2-yl)phenoxy]acetamide
N,N-diethyl-2-({4-[(3-hydroxyphenyl)methyl]-2-oxo-1-(2-phenylethyl)-1,4-diazepan-6-yl}oxy)acetamide
N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-(2-methoxyphenyl)-1H-pyrazole-4-carboxamide
1-{3-[benzyl(methyl)amino]piperidin-1-yl}-3-(4-fluorophenyl)propan-1-one
9-hydroxy-N-(2-methoxyethyl)-4-oxo-N-(pyridin-2-ylmethyl)-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
(2R,6R)-11-methoxy-4-[(4-methyl-1H-imidazol-5-yl)methyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
3-[5-(3-hydroxypyridine-2-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]-1-(morpholin-4-yl)propan-1-one
1-(morpholin-4-yl)-3-{1-[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzoyl]piperidin-4-yl}propan-1-one
{1-[5-(naphthalen-2-yl)-1,2,4-triazin-3-yl]piperidin-3-yl}methanol
5-ethyl-3-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-5-(1-{[3-(trifluoromethyl)phenyl]methyl}piperidin-4-yl)imidazolidine-2,4-dione
1-methyl-5-(3-methylbenzoyl)-N-[2-(morpholin-4-yl)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-(2,3-dihydro-1H-inden-2-yl)-5-[1-(3-methoxybenzoyl)piperidin-4-yl]-5-methylimidazolidine-2,4-dione
(3aS,6aS)-2-cyclopentyl-5-(4-methylbenzoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-[4-(2H-1,3-benzodioxol-5-yl)-2-[(diethylamino)methyl]phenoxy]-N-(quinolin-3-ylmethyl)acetamide
N-ethyl-5-(methoxymethyl)-1-[5-methyl-4-(thiophen-2-yl)pyrimidin-2-yl]-N-(pyridin-4-ylmethyl)-1H-pyrazole-4-carboxamide
methyl 3-(4-tert-butylbenzoyl)-7-oxo-9-(pyridin-3-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-(4-cyclohexanecarbonylpiperazine-1-carbonyl)-8-fluoroquinoline
N-(pyridin-3-yl)-3-{[2-(pyridin-3-yl)piperidin-1-yl]methyl}benzamide
5-amino-N-({1-[(2-fluorophenyl)methyl]pyrrolidin-3-yl}methyl)-1H-pyrazole-3-carboxamide
N-(3-{5-methyl-4-[(3-methyl-2-oxopentanamido)methyl]-1,3-oxazol-2-yl}phenyl)oxane-4-carboxamide
(3aS,6aS)-2-cyclohexyl-5-[(3-methyl-1,2-oxazol-5-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-{[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}-N,N-dimethyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-3-carboxamide
(1S,4S)-2-(3-chloro-4-fluoro-1-benzothiophene-2-carbonyl)-2,5-diazabicyclo[2.2.1]heptane
2-{[4-methyl-5-(4-methyl-1H-imidazol-5-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
3-hydroxy-1-[(1S,5R)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
3-methoxy-N-[(2-{4-[3-(4-methoxyphenyl)propanamido]phenyl}-5-methyl-1,3-oxazol-4-yl)methyl]propanamide
(2E)-3-(3-chlorophenyl)-1-[3-(3-fluoro-4-methoxybenzoyl)piperidin-1-yl]prop-2-en-1-one
2-(2,3-dihydro-1-benzofuran-7-yl)-2-[4-(pyrrolidin-1-yl)piperidin-1-yl]acetic acid
N-[4-(4-{2-[(2-methylphenyl)methyl]-3H-imidazo[4,5-b]pyridin-3-yl}piperidine-1-carbonyl)phenyl]acetamide
1-{[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-methylpiperidine
2-(dimethylamino)-2-(2-methylphenyl)-N-{[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]methyl}acetamide