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1-[(1-methyl-1H-pyrazol-4-yl)methyl]-6-(pyridin-4-ylmethoxy)-4-[2-(thiophen-2-yl)acetyl]-1,4-diazepan-2-one
(3S,4R)-1-(2,6-difluoro-4-methoxybenzoyl)-4-phenylpyrrolidine-3-carboxylic acid
N-[(3S,4S)-4-hydroxy-1,1-dioxo-1λ6-thiolan-3-yl]-N-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-(2H-1,3-benzodioxol-5-yl)-1-(1-cyclobutanecarbonylpiperidin-4-yl)-5-fluoro-1H-1,3-benzodiazole
dimethyl({[(1R,5S,6S)-3-[(3R)-1,2,3,4-tetrahydroisoquinoline-3-carbonyl]-3-azabicyclo[3.1.0]hexan-6-yl]methyl})amine
2-(benzylsulfanyl)-5-{[3-(piperidin-1-yl)pyrrolidin-1-yl]methyl}pyrimidine
1-cyclopentyl-N-methyl-6-oxo-N-(1H-pyrazol-5-ylmethyl)piperidine-3-carboxamide
N-(2,4-difluorophenyl)-4-({ethyl[(3S,4R)-4-hydroxyoxolan-3-yl]amino}methyl)benzamide
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-2-(3-hydroxyadamantan-1-yl)acetamide
N-[1-(4-ethoxy-3-fluorophenyl)ethyl]-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide
1-[3-(azepane-1-carbonyl)phenyl]-3-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]urea
[(3-tert-butyl-1H-pyrazol-5-yl)methyl](methyl)[(2E)-2-methylbut-2-en-1-yl]amine
2-(4-benzyl-1-oxo-1,2-dihydrophthalazin-2-yl)-N-({4-benzyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)acetamide
2-({2-[2-(1H-imidazol-1-yl)ethyl]piperidin-1-yl}methyl)-1-methyl-1H-indole
N-[2-(7-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]pyridine-3-carboxamide
N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]-2-{4-[2-(phenylsulfanyl)acetamido]-1H-pyrazol-1-yl}acetamide
3-[1-(3-chloro-2-fluorobenzoyl)piperidin-3-yl]-1-(pyrrolidin-1-yl)propan-1-one
4-(2-ethylbenzoyl)-1-(2-methoxyphenyl)piperazin-2-one
1-[(3R,4R)-3-hydroxy-4-methyl-3-(propan-2-yl)pyrrolidin-1-yl]-3-(5-methyl-1H-1,2,4-triazol-3-yl)propan-1-one
1-[4-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
N-[2-(1,3-benzoxazol-2-ylsulfanyl)ethyl]-2-(trifluoromethyl)pyrimidin-4-amine
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-(5-tert-butyl-1,3,4-oxadiazol-2-yl)piperazine
N-({5-[(3,4-dimethylphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cyclobutanecarboxamide
(1S,5R)-6-(cyclobutylmethyl)-3-(4-methoxypyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
4-({[3-(2-methoxyethyl)-1-methyl-1H-1,2,4-triazol-5-yl]methyl}sulfanyl)pyridine
1-(2,5-dimethylphenyl)-3-[2-(ethylsulfanyl)ethyl]urea
N-(2,3-dihydro-1H-inden-2-yl)-N-propyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carboxamide
methyl 5-[(2,2-dimethylpropyl)amino]-3-(oxolane-2-amido)-1-(3-phenylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
3-(hydroxymethyl)-1-[(8-methylquinolin-5-yl)methyl]pyrrolidin-3-ol
N-[4-(3-fluorophenyl)phenyl]-1-(3-methyl-1H-pyrazole-4-carbonyl)piperidine-3-carboxamide
2-(dimethylamino)-N-{[4-(dimethylamino)oxan-4-yl]methyl}-2-(2-methylphenyl)acetamide
5-chloro-2-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidine-1-carbonyl]phenol
2-[4-({[(1-ethyl-1H-imidazol-2-yl)methyl](methyl)amino}methyl)phenyl]-3H,4H,5H,7H-thieno[3,4-d]pyrimidin-4-one
3-{1-[2-(2,5-difluorophenyl)acetyl]piperidin-4-yl}-1-(morpholin-4-yl)propan-1-one
2-(2-oxo-4-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}piperazin-1-yl)benzonitrile
8-(4-aminopyrimidin-2-yl)-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
4-{4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}azepane
4-hydroxy-1-(6-methyl-2-propylpyrimidin-4-yl)piperidine-4-carboxylic acid
2-cyclopentyl-9-(4-fluoro-2-methylbenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-N-methyl-2-[1-methyl-2,5-dioxo-3-(4-phenylphenyl)pyrrolidin-3-yl]acetamide
7-(3-methoxypyrazin-2-yl)-N-(1,2-oxazol-3-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
3-(but-2-yn-1-yl)-5-(1-cyclohexanecarbonylpiperidin-4-yl)-5-(2-phenylethyl)imidazolidine-2,4-dione
methyl 9-(cyclopentyloxy)-3-methyl-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-{methyl[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]amino}-1-phenylethan-1-ol
7-acetamido-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-1-[2-(pyridin-2-yl)ethyl]-1H-1,3-benzodiazole-5-carboxamide
(1S,5R)-3-(benzenesulfonyl)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
5-(2,6-dimethylphenoxymethyl)-N-[2-(pyridin-4-yl)ethyl]-1,2-oxazole-3-carboxamide
N-(1-carbamoylcyclopentyl)-1-methyl-3-(trimethyl-1H-pyrazol-4-yl)-1H-pyrazole-5-carboxamide
9-(2,6-diaminopyrimidin-4-yl)-2-(2-phenylethyl)-2,9-diazaspiro[5.5]undecan-3-one
{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}({1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl})amine