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3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]propanamide
4-{2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]acetyl}-1-(2-methylpropyl)-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
N-(5-chloro-2-methoxyphenyl)-3-{1-[(5-methylthiophen-2-yl)methyl]piperidin-3-yl}propanamide
ethyl 3-[(3-methoxyphenyl)methyl]-1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperidine-3-carboxylate
N-(furan-2-ylmethyl)-3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carboxamide
5-methyl-4-{[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]amino}thieno[2,3-d]pyrimidine-6-carboxylic acid
(3S)-N,N-dimethyl-1-{4-[(pyridin-2-ylsulfanyl)methyl]benzoyl}azepan-3-amine
(3R,4S)-4-({[2-(3,5-dimethyl-1H-pyrazol-1-yl)-5-fluorophenyl]methyl}(ethyl)amino)oxolan-3-ol
2-{[(3S,4S)-3,4-bis(hydroxymethyl)pyrrolidin-1-yl]methyl}-8-fluoroquinolin-4-ol
5-[2-methyl-4-(2-methylphenyl)piperazine-1-carbonyl]-4-phenylpyrimidin-2-amine
5-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-1H-pyrazole-3-carboxamide
N,2-dimethyl-N-{[2-(pyrrolidin-1-ylmethyl)phenyl]methyl}-2,8-diazaspiro[4.5]decane-3-carboxamide
2-[5-(6-oxopiperazin-2-yl)-1-[4-(trifluoromethyl)phenyl]-1H-1,2,4-triazol-3-yl]acetamide
methyl 1-benzyl-3-cyclopropaneamido-5-[(2-ethylbutyl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-3-[2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-methylpropanamide
1'-[2-(1H-1,2,4-triazol-1-yl)benzoyl]-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
3-phenyl-1-{4-[(2,4,5-trimethoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}propan-1-ol
N-[(3S,4R)-1-(5-ethyl-1,3,4-thiadiazol-2-yl)-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
2-[3-(pyridin-3-yl)phenoxy]propanamide
2-hydroxy-4-methyl-N-[3-(oxolan-3-yl)propyl]benzamide
N-[2-(furan-2-yl)ethyl]-3-[5-(phenoxymethyl)-1,3,4-oxadiazol-2-yl]propanamide
2-methoxy-5-[2-({2-methylthieno[2,3-d]pyrimidin-4-yl}amino)ethyl]phenol
N-(dimethyl-1H-1,2,4-triazol-3-yl)-3-(2-hydroxypropan-2-yl)piperidine-1-carboxamide
2-methyl-5-(4-{2-[(2-oxo-2H-chromen-7-yl)oxy]acetyl}piperazin-1-yl)-2,3-dihydropyridazin-3-one
2-methyl-6-{3-phenyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}pyridine
N-{[7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(2,4,6-trifluorophenyl)acetamide
N-(3,4-dihydro-2H-1-benzopyran-3-yl)-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
3-phenyl-N-[4-(4-{[2-(1H-pyrazol-1-yl)ethyl]amino}piperidin-1-yl)phenyl]propanamide
2-methyl-6-[1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)piperidin-4-yl]pyrimidin-4-ol
3-(2-methoxyethyl)-1-[2-(4-methoxyphenyl)ethyl]-8-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-(2,5-dihydro-1H-pyrrol-1-yl)-7-[(3-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-2-amine
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
4-[3-(diethylamino)pyrrolidin-1-yl]-6-methylpyrimidin-2-amine
2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-{[1-(propan-2-yl)pyrrolidin-3-yl]methyl}acetamide
5-(3-methylphenyl)-4-{1-[5-(2-methylpropyl)-1,2-oxazole-3-carbonyl]piperidin-4-yl}-2-(pyridin-4-yl)pyrimidine
4-[(5-fluoro-2-methoxyphenyl)methyl]-2-(6-methoxynaphthalen-2-yl)morpholine
1-{1-[5-(methoxymethyl)furan-2-carbonyl]piperidin-4-yl}-2-methyl-5-(trifluoromethyl)-1H-1,3-benzodiazole
methyl 4-(4-{[3-(2-fluorophenyl)pyrrolidin-1-yl]methyl}-5-methyl-1,3-oxazol-2-yl)benzoate
N-[(2S,4R,6S)-2-(5-methyl-1-propyl-1H-pyrazol-4-yl)-6-(2-phenylethyl)oxan-4-yl]acetamide
7-[1-(2-ethoxyethyl)-3-methyl-1H-pyrazole-5-carbonyl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
5-[(5-ethylfuran-2-yl)methyl]-2-(3,4,5-trimethoxyphenyl)-2,3,4,5-tetrahydro-1,5-benzothiazepine
1-{2-[(1S,4S)-2,5-diazabicyclo[2.2.1]heptan-2-yl]-2-oxoethyl}-3,4-diphenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[(7-{[4-(benzyloxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]oxolane-3-carboxamide
3-[(3S,4R)-1-[(4-chlorophenyl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]-N-[3-(dimethylamino)phenyl]propanamide
1-[(2-chlorophenyl)methyl]-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
3-[ethyl({[2-(naphthalen-1-yl)pyrimidin-5-yl]methyl})amino]-1λ6-thiolane-1,1-dione
N-{1-[1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-4-phenylbutanamide
N-({7-[(2E)-3-(4-hydroxy-3-methoxyphenyl)prop-2-en-1-yl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)furan-2-carboxamide
3-(3-ethyl-1,4-dimethyl-1H-pyrazol-5-yl)-1-[(2R)-1-hydroxy-3-(4-hydroxyphenyl)propan-2-yl]urea
5-{2-[(1,4-dithiepan-6-yl)amino]ethyl}-1,3,4-thiadiazol-2-amine