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4-(6-methoxypyridin-2-yl)-2-({[2-(piperidin-1-yl)ethyl]amino}methyl)phenol
N-{1-[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]ethyl}-7-methylimidazo[1,2-a]pyridine-2-carboxamide
(3aS,6aS)-5-[5-(4-methoxyphenyl)furan-2-carbonyl]-1-methyl-octahydropyrrolo[3,4-b]pyrrole
1-[4-({[(1-ethyl-1H-imidazol-2-yl)methyl](methyl)amino}methyl)-2-methoxyphenoxy]-3-(thiomorpholin-4-yl)propan-2-ol
1-[(4-fluorophenyl)methyl]-4-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}-2-(propan-2-yl)-1,4-diazepane
N-(2,3-dihydro-1H-inden-2-yl)-4-(methoxymethyl)-N,5-dimethyl-1,2-oxazole-3-carboxamide
N-(1-{2-butyl-4-oxo-1,3,8-triazaspiro[4.5]dec-1-en-8-yl}-3-methyl-1-oxobutan-2-yl)acetamide
1-[2-(5-{2H,4H,5H,6H-cyclopenta[c]pyrazol-3-yl}-1,2,4-oxadiazol-3-yl)ethyl]pyrrolidin-2-one
(4aS,7aR)-1-(2-ethoxyethyl)-4-ethyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1'-(3,4-dihydro-2H-1-benzopyran-2-carbonyl)-5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-1-[(3-methoxyphenyl)methyl]-N-methyl-6-oxopiperidine-3-carboxamide
N-methyl-3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-(2-phenoxyethyl)propanamide
6-[(2,4-dimethoxy-3-methylphenyl)methyl]-N-(3-fluorophenyl)-6-azaspiro[2.5]octane-1-carboxamide
7-(5-chloropyridin-2-yl)-4-(2-methylfuran-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-[(1-{4-[(butylsulfanyl)methyl]-5-methylfuran-2-carbonyl}piperidin-4-yl)methyl]pyrrolidin-2-one
3-[(4-methoxyphenyl)methyl]-1-methyl-8-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
[(1-ethyl-1H-pyrazol-4-yl)methyl](1H-indol-3-ylmethyl)(2-methylpropyl)amine
N-(cyclohexylmethyl)-5-[4-(2,3-dimethylphenyl)piperazine-1-carbonyl]-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
3-{4-[4-(4-fluorophenyl)-1-phenylbut-3-yn-2-yl]piperazin-1-yl}propanamide
methyl 9-[3-(dimethylamino)propoxy]-3-[3-(4-methoxyphenyl)propanoyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-[(1S,5R)-7-oxo-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]pyridine-4-carbonitrile
N-(cyclobutylmethyl)-N-(oxolan-2-ylmethyl)-4-(1H-pyrazol-3-yl)benzamide
3-(3-methoxyphenyl)-N-[(5-phenyl-1,2-oxazol-3-yl)methyl]-1H-pyrazole-4-carboxamide
N-{[5-fluoro-7-(pyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-1-methylpiperidine-3-carboxamide
methyl (2S,4S)-1-[(2-chlorophenyl)methyl]-4-[2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)acetamido]pyrrolidine-2-carboxylate
methyl (2S,4R)-1-[2-(3-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]-4-hydroxypyrrolidine-2-carboxylate
N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-(methoxymethyl)-N-[2-(1-methylpiperidin-3-yl)ethyl]cyclobutane-1-carboxamide
4-(2-{[6-methyl-2-(pyridin-3-yl)pyrimidin-4-yl]amino}ethyl)benzene-1-sulfonamide
[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl](methyl)[3-(1-methyl-1H-imidazol-2-yl)propyl]amine
N-({7-[2-(2,3-difluorophenyl)acetyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2H-1,3-benzodioxole-5-carboxamide
2-(2H-1,3-benzodioxol-5-yl)-1-[4-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]ethan-1-one
2-{[(2-chlorophenyl)methyl]sulfanyl}-N-[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]acetamide
(1S,5R)-6-methyl-3-[4-(3-methylphenoxy)benzoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
4-ethyl-3-[(1-{[2-(furan-2-yl)pyrimidin-5-yl]methyl}piperidin-4-yl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
3-(3-hydroxy-3-methylbutyl)-N-[1-(4-methylphenyl)-5-oxopyrrolidin-3-yl]benzamide
N-(2,1,3-benzothiadiazol-5-ylmethyl)-5-(2,6-dimethoxyphenyl)-N-methyl-1,2,4-triazin-3-amine
N-cyclopropyl-1-[(3-methoxyphenyl)methyl]-5-[4-(1H-pyrazol-1-yl)benzoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(1S,5R)-6-benzyl-3-(2-cyclopentylacetyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3-[(1-acetylpiperidin-4-yl)oxy]-4-methoxy-N-[1-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]benzamide
1-cyclohexyl-6-hydroxy-4-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-1,4-diazepan-2-one
5-ethyl-N-{[1-(1H-imidazol-1-ylmethyl)cyclopropyl]methyl}-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
5-{1-[2-(3,4-difluorophenyl)acetyl]piperidin-4-yl}-3-(oxolan-2-ylmethyl)-5-propylimidazolidine-2,4-dione
3-({1-[3-(4-fluorophenyl)phenyl]piperidin-4-yl}amino)propanamide
2-[1-(cyclohexylmethyl)-3-oxopiperazin-2-yl]-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)acetamide
(3S,7S)-5-(dimethyl-1,3-thiazole-5-carbonyl)-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
6-[(3-cyanopiperidin-1-yl)methyl]-N-({2-methylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)-2-oxo-1,2-dihydropyridine-3-carboxamide
1-(1-cyclohexanecarbonylpiperidin-4-yl)-3-(pyrrolidine-1-carbonyl)piperidine
N-({8-benzyl-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-2-(1,3-dioxo-2,3-dihydro-1H-isoindol-2-yl)acetamide
N-ethyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide