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1-methyl-4-{1-[1-(1-methyl-1H-imidazole-5-carbonyl)piperidin-4-yl]piperidine-3-carbonyl}piperazine
2-(1-{[1-(3,4-dimethylbenzoyl)piperidin-3-yl]methyl}-1H-1,2,3-triazol-4-yl)pyridine
(3R,4R)-1-[(5-cyclopentylthiophen-2-yl)methyl]-4-{methyl[2-(pyridin-2-yl)ethyl]amino}piperidin-3-ol
N-[4-(2-fluorophenoxy)phenyl]-1-(2-methoxyethyl)piperidine-4-carboxamide
1-[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-[(2-methoxyethyl)(methyl)amino]ethan-1-one
methyl 3-(2-methoxybenzamido)-5-{[(1-methyl-3-propyl-1H-pyrazol-5-yl)formamido]methyl}benzoate
3-[2-(methylsulfanyl)benzoyl]-1-(1,2,5-thiadiazole-3-carbonyl)piperidine
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-2-(2-oxopiperidin-1-yl)acetamide
N-{1-[1-(5-acetylthiophene-2-carbonyl)piperidin-4-yl]-2-(2-methylphenyl)ethyl}-N-methyl-2-(1H-pyrazol-1-yl)acetamide
9-[2-(4,5-dimethyl-1H-imidazol-1-yl)acetyl]-2-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-(2-benzyl-1,3-thiazole-4-carbonyl)-3-(2-methoxybenzoyl)piperidine
N-[(2,6-difluoro-3-methylphenyl)methyl]-7-acetamido-1-[2-(pyridin-2-yl)ethyl]-1H-1,3-benzodiazole-5-carboxamide
(1R,5R)-6-(1-benzothiophene-2-carbonyl)-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
6-methyl-2-[3-oxo-2-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-9-yl]pyridine-3-carbonitrile
3-[(3-fluorophenyl)methyl]-N-[(3-phenyl-1H-pyrazol-4-yl)methyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
3-[2-(2H-1,3-benzodioxol-5-ylmethyl)-5-oxopyrrolidin-2-yl]-N-[3-(pyridin-3-yl)propyl]propanamide
4-(5-methylthiophene-2-carbonyl)-9-(oxan-2-ylmethoxy)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-(but-3-enoyl)-N-[4-(2-fluorophenoxy)phenyl]piperidine-4-carboxamide
2-{1-ethyl-2,5-dioxo-3-[3-(trifluoromethyl)phenyl]pyrrolidin-3-yl}-N-methyl-N-(quinolin-5-ylmethyl)acetamide
6-(2-ethylbutyl)-N-(2-phenylethyl)-6-azaspiro[2.5]octane-1-carboxamide
1-[(4-chlorophenyl)methyl]-N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-6-oxopiperidine-3-carboxamide
N-[(4-hydroxyazepan-4-yl)methyl]-6-methoxy-1-methyl-1H-indole-2-carboxamide
2-methoxy-6-(1-propyl-1H-1,2,4-triazol-5-yl)phenol
1-[cyclohexyl(methyl)amino]-3-[2-methoxy-4-({[3-(methylsulfanyl)propyl]amino}methyl)phenoxy]propan-2-ol
5-methyl-N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-1-propyl-1H-pyrazole-4-carboxamide
(5S,9aS,9bS)-2-[(3-methoxyphenyl)methyl]-5-(pyridin-3-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-[4-(propan-2-yl)benzoyl]piperidin-3-yl]propanoic acid
N-({8-benzyl-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-1-methyl-1H-pyrazole-3-carboxamide
4-ethyl-1-methyl-3-[(1-{4H-thieno[3,2-b]pyrrole-5-carbonyl}piperidin-4-yl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
2-{5-[(2,6-difluorophenyl)methyl]-3-methyl-1H-1,2,4-triazol-1-yl}ethan-1-ol
2-({4-[6-(morpholine-4-carbonyl)pyrazin-2-yl]-1H-pyrrolo[2,3-b]pyridin-6-yl}amino)ethan-1-ol
N-(1-{1-[3-(furan-2-yl)benzoyl]piperidin-4-yl}-1H-pyrazol-5-yl)acetamide
(3S)-1,3-dimethyl-4-{[1-methyl-3-(4-phenoxyphenyl)-1H-pyrazol-4-yl]methyl}piperazin-2-one
1-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-(1H-1,2,4-triazol-1-yl)propan-1-one
methyl 2-chloro-5-{[3-(2-oxopyrrolidin-1-yl)piperidine-1-carbonyl]amino}benzoate
1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidine
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-[(4-methylphenyl)amino]cyclopentane-1-carboxamide
N-{[7-(3,6-dimethylpyrazin-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
4-{1-[(3-chlorophenyl)methyl]azetidin-3-yl}morpholine
N-[2-(1-{[2-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}piperidin-2-yl)ethyl]acetamide
4-phenyl-3-(1-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-1-ethyl-1H-pyrazole-4-sulfonamide
N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}-6-(pyridin-3-yl)pyridine-3-carboxamide
2-ethyl-6-methyl-4-oxo-1-[2-(piperidin-1-yl)ethyl]-N-(pyridin-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
4-{1-[(4aR,8aR)-6-(thiophen-3-ylmethyl)-decahydro-1,6-naphthyridin-1-yl]-1-oxopropan-2-yl}-1,2-dihydrophthalazin-1-one
2-methyl-8-(1,2,5-oxadiazole-3-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
1-(1-{5H,6H-benzo[h]quinazolin-2-yl}-5-methyl-1H-pyrazole-4-carbonyl)-4-cyclopentylpiperazine
7-(5-phenylpentanoyl)-2-(pyridin-4-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-cyclohexyl-1-(2-methoxyethyl)-5-oxo-N-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
6-fluoro-N-[2-(4-methyl-1H-1,2,3-triazol-1-yl)ethyl]-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide