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methyl 6-{[ethyl(2-methylprop-2-en-1-yl)amino]methyl}-3-(2-phenylacetamido)thieno[2,3-b]pyridine-2-carboxylate
methyl({4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl})(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)amine
(2E)-3-(2,6-difluorophenyl)-N-({8-[(2-methylphenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)prop-2-enamide
1-{4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pentane-1,2-dione
[(3R,4S)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-{[4-(methylsulfanyl)phenyl]methyl}pyrrolidin-3-yl]methanol
{2-ethoxy-5-[4-phenyl-1-(pyridin-4-ylmethyl)-1H-imidazol-5-yl]phenyl}methanol
5-ethyl-2,3-dimethyl-N-[(1-propyl-1H-pyrazol-4-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
methyl 3-{[(3-ethyl-1-methyl-1H-pyrazol-5-yl)formamido]methyl}-5-(2-phenylacetamido)benzoate
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-cyclopropyl-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-3-methoxy-1,2-dihydropyridin-2-one
5-ethyl-N-({3-methyl-7-[2-(thiophen-3-yl)acetyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-1,2-oxazole-3-carboxamide
2-[(3-fluorophenyl)methyl]-4-{4-[3-(3-methyl-1H-pyrazol-1-yl)propanoyl]piperazin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
N-(2-{[7-acetyl-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]amino}ethyl)propanamide
methyl 4-[({3-[(4-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazol-5-yl}formamido)methyl]benzoate
2-[1-cyclohexyl-3-(2-fluorophenyl)-2,5-dioxopyrrolidin-3-yl]-N-(cyclopropylmethyl)-N-(oxolan-2-ylmethyl)acetamide
N-[(1S,3R)-3-aminocyclopentyl]-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
1-[2-(3-chloro-4-fluorophenyl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]piperidine-3-carboxamide
2-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{[7-(4,6-dimethylpyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}propanamide
N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-5-(naphthalen-1-yl)-1,2,4-triazin-3-amine
5-(3-chlorophenyl)-N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-1,2,4-triazin-3-amine
(4aS,8aR)-1-[3-(1H-imidazol-1-yl)propyl]-6-methanesulfonyl-decahydro-1,6-naphthyridin-2-one
N-({8-[(2-fluorophenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-4-(trifluoromethyl)benzamide
1-benzyl-3-(2-methylphenyl)-3-{2-oxo-2-[4-(pyrimidin-2-yl)-1,4-diazepan-1-yl]ethyl}pyrrolidine-2,5-dione
1-(2-hydroxyethyl)-5-(1-methylpiperidine-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
3-chloro-2-fluoro-N-{[7-(5-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
N-benzyl-N-methyl-3-{[methyl(quinoxalin-6-ylmethyl)amino]methyl}imidazo[1,2-a]pyridine-2-carboxamide
1-[1'-(dimethyl-1,3-thiazole-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]-2-methoxyethan-1-one
3-{[(2,6-difluoro-3-methylphenyl)methyl](propan-2-yl)amino}propanamide
1-(4-ethylpiperazin-1-yl)-3-[3-({[(4-fluorophenyl)methyl](methyl)amino}methyl)phenoxy]propan-2-ol
(3S,4S)-4-(propan-2-yl)-1-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
methyl 3-{[2-(2,5-dimethoxyphenyl)acetamido]methyl}-5-(2-phenylacetamido)benzoate
1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
N-[5-({[2-(5-ethyl-1,2,4-oxadiazol-3-yl)ethyl]carbamoyl}amino)-2-methoxyphenyl]acetamide
4-methoxy-3-[(1R,5S,8R)-8-methoxy-3-azabicyclo[3.2.1]octane-3-carbonyl]benzene-1-sulfonamide
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]acetamide
{[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)(pyrimidin-4-ylmethyl)amine
(2S,4S)-4-[(1-benzylpiperidin-4-yl)amino]-1-[(2-chlorophenyl)methyl]-N-ethylpyrrolidine-2-carboxamide
N-[(2R,3R)-1'-(4-hydroxybenzoyl)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-phenylacetamide
1-{1-[(8-methoxy-2H-chromen-3-yl)methyl]piperidin-3-yl}-4-(4-methoxyphenyl)piperazine
{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)(quinoxalin-6-ylmethyl)amine
(3S,4S)-3-[({3-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)(methyl)amino]-4-hydroxy-1λ6-thiolane-1,1-dione
(1S,5R)-6-(cyclobutylmethyl)-3-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonane
1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
4-(4-chlorophenyl)-N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)propyl]butanamide
N-(3-cyclopropyl-1-methyl-1H-pyrazol-5-yl)-2-[3-(3,4-dimethoxyphenyl)-1H-pyrazol-1-yl]acetamide
(3aS,6aR)-3-[3-(4-fluorophenyl)propyl]-5-(pyridin-2-yl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
3-[(3R,7S,8aS)-1,4-dioxo-3-(propan-2-yl)-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3,5-dimethylphenyl)urea
1-{[(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)carbamoyl]methyl}piperidine-4-carboxamide
N-[5-(3-chloro-4-methoxyphenyl)pyridin-2-yl]methanesulfonamide
1-[1-(2-cyclohexylethyl)-1H-1,2,3-triazole-4-carbonyl]-3-(1-methyl-1H-imidazole-2-carbonyl)piperidine