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5-(1-benzylpiperidin-4-yl)-5-(3-phenylpropyl)imidazolidine-2,4-dione
1-methyl-N-({5-methylimidazo[1,2-a]pyridin-2-yl}methyl)-2,4-dioxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
[(2,6-difluorophenyl)methyl]({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)(2-methoxyethyl)amine
3-methyl-4-[6-methyl-4-(trifluoromethyl)pyridin-2-yl]-1-(2-methylpropyl)piperazin-2-one
1-[(6,7-dimethoxy-4-methylquinolin-2-yl)amino]-3-ethoxypropan-2-ol
1-{3-[(3,4-difluorophenyl)amino]piperidin-1-yl}-2-(dimethyl-1,2-oxazol-4-yl)ethan-1-one
N-ethyl-2-hydroxy-N-[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]-6-(trifluoromethyl)pyridine-3-carboxamide
6-ethyl-N-{[3-(2-methoxyethoxy)phenyl]methyl}pyrimidin-4-amine
1-(2,3-dihydro-1H-inden-2-yl)-5-[(2-methoxyethoxy)methyl]-3-(thiophen-2-ylmethyl)-1H-1,2,4-triazole
(3-{2-[1-(4-methoxy-2-methylbenzoyl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)dimethylamine
3-[3-(1H-1,3-benzodiazol-2-yl)azetidine-1-carbonyl]pyridin-2-ol
N-[2-(7-{[2-(furan-2-yl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]-2-phenoxyacetamide
6-(3-{4-[(3,5-dimethylphenyl)methyl]-3-oxopiperazin-1-yl}-3-oxopropyl)-2,3-dihydropyridazin-3-one
(3aS,6aS)-5-(naphthalen-2-ylmethyl)-1-oxo-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-methyl-N-{1-[2-(1H-pyrazol-1-yl)phenyl]ethyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N,N-dimethyl-5-{3-phenyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl}pyridin-2-amine
2-(pyridin-3-yl)-N-[2-(pyrrolidine-1-sulfonyl)ethyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
methyl 2-[2,4-dioxo-1-(2-phenylethyl)-8-(pyridin-4-ylmethyl)-1,3,8-triazaspiro[4.5]decan-3-yl]acetate
1-benzyl-N-(3-methoxypropyl)-2-methyl-5-(2-methylpropanamido)-1H-1,3-benzodiazole-7-carboxamide
N-({2-[3-(2,5-dimethylfuran-3-amido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)-5-ethyl-1,2-oxazole-3-carboxamide
1-[1-(furan-2-ylmethyl)piperidine-3-carbonyl]-4-(pyridin-3-yl)piperidin-4-ol
3-{2-[(2-fluorophenyl)carbamoyl]ethyl}-N-(furan-2-ylmethyl)piperidine-1-carboxamide
N-[3-(4-{[(1-hydroxycyclohexyl)methyl]amino}piperidin-1-yl)phenyl]-3-(trifluoromethyl)benzamide
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-(thiophen-3-yl)acetamide
N-(4-{[3-hydroxy-3-(pyrrolidin-1-ylmethyl)piperidin-1-yl]methyl}phenyl)acetamide
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]oxane-2-carboxamide
3-{[ethyl(oxan-4-yl)amino]methyl}benzoic acid
1-{6-[(dimethylamino)methyl]-1,4-oxazepan-4-yl}-2-(pyridin-3-yl)ethane-1,2-dione
N-({1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]pyrrolidin-3-yl}methyl)methanesulfonamide
N-[(3R,4S)-1-(2-methanesulfonylethyl)-4-propylpyrrolidin-3-yl]-5-methyl-2H-1,2,3-triazole-4-carboxamide
N-(2-hydroxybutyl)-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
1-(2-methoxyacetyl)-N-[2-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]piperidine-4-carboxamide
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
1-{1-[(2-chlorophenyl)methyl]piperidin-4-yl}-3-(3-methyl-1,2,4-thiadiazol-5-yl)urea
3-(2-methylphenyl)-3-[2-(2-methylpiperidin-1-yl)-2-oxoethyl]-1-(pyridin-3-ylmethyl)pyrrolidine-2,5-dione
1-(cyclopropylmethyl)-6-[(2-hydroxy-6-methoxyphenyl)methyl]-3-[(2-methylphenyl)methyl]-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
(2S,4R)-4-amino-N-methyl-1-[(1-propyl-1H-pyrazol-5-yl)sulfonyl]pyrrolidine-2-carboxamide
N-[(2,4-dimethoxyphenyl)methyl]-3-{1-[3-(pyridin-2-yl)propanoyl]piperidin-3-yl}propanamide
2-chloro-4-fluoro-N-{[7-(6-methoxypyridazin-3-yl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
2-{4-[1-(diphenylmethyl)-1H-1,2,3-triazole-4-carbonyl]piperazin-1-yl}pyrimidine
3-hexyl-8-(1-methyl-2-oxo-1,2-dihydropyridine-4-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}-N-(propan-2-yl)piperidine-1-carboxamide
4-(2,5-dimethylfuran-3-carbonyl)-6-[(3-methoxyphenyl)methoxy]-1-(pyridin-2-ylmethyl)-1,4-diazepan-2-one
N-benzyl-6-[4-(propan-2-yl)piperazin-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
1-(piperidin-1-yl)-3-{4-[({[2-(trifluoromethyl)phenyl]methyl}amino)methyl]phenoxy}propan-2-ol
ethyl 2-[1-(3-benzyl-4,5-dihydro-1,2-oxazole-5-carbonyl)piperidin-2-yl]acetate
8-[(4-hydroxyphenyl)methyl]-1-(2-phenylethyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
ethyl 4-[6-(furan-3-ylmethyl)-6-azaspiro[2.5]octane-1-amido]piperidine-1-carboxylate
2-[2-(1H-pyrazol-1-yl)ethyl]-1-[3-(1H-pyrazol-1-ylmethyl)benzoyl]piperidine
1,9-dimethyl-4-[2-(thiophen-2-yl)acetyl]-1,4,9-triazaspiro[5.6]dodecan-10-one