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3-{1-[2-(5-oxopyrrolidin-2-yl)acetyl]piperidin-4-yl}-N-phenylpropanamide
1-(2-{[(cyclobutylmethyl)(methyl)amino]methyl}-6-methoxyphenoxy)-3-(morpholin-4-yl)propan-2-ol
(2S,4R)-N-[(1-benzylpiperidin-4-yl)methyl]-4-hydroxy-N-methylpyrrolidine-2-carboxamide
1-[2-(1H-imidazol-2-yl)benzoyl]-4-(2-phenoxyethyl)piperazine
2-(ethoxymethyl)-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
(1-{5-[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}piperidin-3-yl)methanol
2-cyclohexyl-N-[(4,6-dimethylpyrimidin-2-yl)methyl]-1,3-benzoxazole-6-carboxamide
N-(isoquinolin-5-ylmethyl)-N-methyl-2-(2-phenyl-1H-imidazol-1-yl)acetamide
3-[(3-methoxyphenyl)methyl]-1-(3-methylbutyl)-8-(thiophen-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N4-[(2,4-dimethoxyphenyl)methyl]-6-ethyl-5-methylpyrimidine-2,4-diamine
4-[1-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-4-yl]-1-[(dimethyl-1,2-oxazol-4-yl)methyl]-1,2,3,6-tetrahydropyridine
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-ethylbenzamide
2-methyl-8-(1H-pyrrole-2-carbonyl)-2,8-diazaspiro[4.5]decane
N-(6-methoxy-2H-1,3-benzodioxol-5-yl)-2-(3-methoxyphenyl)piperidine-1-carboxamide
5-{methyl[(3-methylthiophen-2-yl)methyl]amino}-1-propyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
2-({4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}methyl)benzoic acid
1-{5H,6H-benzo[h]quinazolin-2-yl}-5-cyclopropyl-N-(2-methoxyethyl)-N-methyl-1H-pyrazole-4-carboxamide
4-acetamido-N-[1-(3-fluoro-4-methoxyphenyl)ethyl]-3-methylbenzamide
4-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-4H-1,2,4-triazole
4-({[3-(2-chlorophenyl)-1,2-oxazol-5-yl]methyl}amino)-N-cyclopropylpyridine-2-carboxamide
3-phenoxy-N-[1-({[(2-phenyl-1,3-thiazol-4-yl)methyl]carbamoyl}methyl)-1H-pyrazol-4-yl]propanamide
9-[6-(1-hydroxyethyl)pyridin-2-yl]-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}-N-(2-methoxyphenyl)piperidine-1-carboxamide
4-ethyl-3-{[1-(2-phenylethyl)piperidin-4-yl]methyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
4-({2-[1-(3-ethyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
N-benzyl-N-methyl-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-sulfonamide
2-methyl-N-[3-(1-methyl-1H-1,3-benzodiazol-2-yl)propyl]imidazo[1,2-a]pyrimidine-3-carboxamide
3-chloro-N-({4-[2-(piperidin-1-yl)ethoxy]phenyl}methyl)-N-(pyridin-2-ylmethyl)benzamide
2-(3-fluorophenoxymethyl)-N-[(3R,4R)-4-(pyrrolidin-1-yl)oxolan-3-yl]-1,3-oxazole-4-carboxamide
(1S,5R)-3-benzyl-6-(1-ethyl-1H-pyrazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-amino-4-[5-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-6-(thiophen-3-yl)pyridine-3-carbonitrile
N-(1-{1-[(4-acetamidophenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)cyclopropanecarboxamide
N-[2-(1H-imidazol-1-yl)ethyl]-2-(N-phenylmethanesulfonamido)propanamide
N-{[7-(4-methanesulfonylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-1-phenyl-1H-pyrazole-4-carboxamide
1-[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
3-[(2-methoxyethyl)sulfamoyl]-5-[3-(pyrazin-2-yl)-1H-pyrazol-1-yl]benzoic acid
5-{1-[(6-methyl-4-oxo-4H-chromen-3-yl)methyl]piperidin-4-yl}-5-(3-methylbutyl)imidazolidine-2,4-dione
{[3-(6-methoxynaphthalen-2-yl)-1H-pyrazol-4-yl]methyl}[1-(thiophen-2-yl)propan-2-yl]amine
N-methyl-N-(2-phenylethyl)-1-(propane-1-sulfonyl)piperidin-3-amine
2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-N-[(2S)-pyrrolidin-2-ylmethyl]-2,3-dihydro-1H-indene-2-carboxamide
N-(2-{[1-(ethylsulfanyl)propan-2-yl]amino}ethyl)-N-methylmethanesulfonamide
2-(1,4-dimethylpiperazin-2-yl)-1-[4-(4-fluorophenyl)-4-hydroxypiperidin-1-yl]ethan-1-one
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-[2-(2-ethylphenoxy)ethyl]-N-methylacetamide
4-(3-hydroxy-3-methylbutyl)-N-[1-(methoxymethyl)cyclopropyl]-N-methylbenzamide
N-{[7-(4-ethenylbenzoyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2H-1,3-benzodioxole-5-carboxamide
2-{4-[2-(2,6-dimethylphenyl)-1H-imidazol-1-yl]phenyl}acetic acid
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-5-[(5,6,7,8-tetrahydronaphthalen-2-yloxy)methyl]-1,2-oxazole-3-carboxamide
1-{4-[3-(4-fluorophenoxy)propyl]piperazine-1-carbonyl}-6-azaspiro[2.5]octane
2-(2,3-dihydro-1H-inden-1-yl)-1-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]ethan-1-one
4-[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]-6-methylpyrimidin-2-amine