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N-ethyl-5-{1-[(1-methyl-1,2,3,4-tetrahydroquinolin-6-yl)methyl]pyrrolidin-2-yl}thiophene-2-carboxamide
2-methyl-4-(2-methylpropyl)-6-[1-(6-methylpyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]pyrimidine
1-methyl-N-({5-methyl-2-[3-(3-methylbutanamido)phenyl]-1,3-oxazol-4-yl}methyl)-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
N-methyl-3-{3-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}propanamide
5-methoxy-N-[1-(4-methoxyphenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]furan-2-carboxamide
1-(7-methanesulfonyl-4-methylquinazolin-2-yl)-N-(naphthalen-1-ylmethyl)azepan-4-amine
3-{1-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]piperidin-4-yl}-N-(2,3-dihydro-1,4-benzodioxin-6-yl)propanamide
3,3-dimethyl-1-[(5-{[2-(methylsulfanyl)phenyl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)methyl]urea
2-methoxy-5-[(2-methylphenyl)methyl]benzamide
(5S,9aS,9bS)-5-[2-(dimethylamino)-1,3-thiazol-5-yl]-2-(2-phenylethyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
2-(4-fluorophenyl)-1-{2-[2-(3-{[methyl(quinolin-8-ylmethyl)amino]methyl}phenoxy)ethyl]piperidin-1-yl}ethan-1-one
2-[5-(methoxymethyl)thiophene-2-carbonyl]-7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decane
[2-(3-fluorophenyl)ethyl](oxolan-2-ylmethyl)(pyridin-2-ylmethyl)amine
3-[(cyclopropylmethyl)amino]-N-(pyridin-2-ylmethyl)-5-(pyrrolidine-1-sulfonyl)benzamide
6-(5-fluoro-2-methoxyphenyl)-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}pyridine-3-carboxamide
N-{2-[(4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}phenyl)formamido]ethyl}acetamide
4-[3-(3-methoxyphenoxy)propyl]-1,3λ6,4-oxathiazinane-3,3-dione
3-(but-2-yn-1-yl)-5-{1-[(3,5-difluorophenyl)methyl]piperidin-4-yl}-5-(2-phenylethyl)imidazolidine-2,4-dione
N-{[4-(2-methylphenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}propanamide
1-{[5-fluoro-2-(trifluoromethyl)phenyl]methyl}-3-methylimidazolidin-2-one
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(2-methyl-1,3-thiazole-4-carbonyl)pyrrolidin-3-yl]-1H-pyrrole-2-carboxamide
(1R,3S)-3-(2-hydroxyethoxy)-7-[(2Z)-5-methyl-2-phenylhex-2-en-1-yl]-7-azaspiro[3.5]nonan-1-ol
7-(2-methoxyacetamido)-N-methyl-N-(oxan-4-yl)-1-(2-phenylethyl)-1H-1,3-benzodiazole-5-carboxamide
1-(2-methylpropyl)-4-oxo-5-(piperidine-1-carbonyl)-N-[2,2,2-trifluoro-1-(furan-2-yl)ethyl]-1,4-dihydropyridine-3-carboxamide
4-ethyl-3-[(1-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}piperidin-4-yl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-(2-methylpropyl)-4-oxo-N-(thiophen-3-ylmethyl)-3,4-dihydroquinazoline-2-carboxamide
N-(6-fluoro-2-oxo-1,2,3,4-tetrahydroquinolin-8-yl)-4-methyl-1,2,3,6-tetrahydropyridine-1-carboxamide
2-{[(1-{[2-(4-methoxy-2,5-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-yl)oxy]methyl}pyridine
3-[(4-methoxy-4-phenylpiperidin-1-yl)methyl]piperidin-3-ol
1-(3-{3-[(2-methyl-1H-imidazol-1-yl)methyl]piperidin-1-yl}-3-oxopropyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
{[2-(ethanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(methyl)[1-(1,3-thiazol-2-yl)ethyl]amine
(2S,4R)-4-amino-1-[(2-tert-butylpyrimidin-5-yl)methyl]-N-methylpyrrolidine-2-carboxamide
1-{[3-(pyrrolidine-1-carbonyl)-1,2-oxazol-5-yl]methyl}piperidin-4-ol
ethyl 4-[1-(2,3-dimethyl-1H-indole-5-carbonyl)piperidin-3-yl]piperazine-1-carboxylate
(1S,5R)-3-(1,7-dimethyl-1H-indole-2-carbonyl)-3,9-diazabicyclo[3.3.2]decan-10-one
5-ethyl-3-[2-(4-methoxyphenyl)ethyl]-5-(1-propylpiperidin-4-yl)imidazolidine-2,4-dione
1-ethyl-3-[(3-methoxyphenyl)methyl]-8-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(5-fluoro-2-methoxybenzoyl)-N-(2-phenylethyl)piperidine-1-carboxamide
2-{2-[5-(methoxymethyl)furan-2-carbonyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl}-6-methylpyridine
2-[4-({methyl[(1,2,2-trimethylpyrrolidin-3-yl)methyl]amino}methyl)phenyl]ethan-1-amine
N-{[4-(oxolan-3-yloxy)phenyl]methyl}-N-(pyridin-2-ylmethyl)-4,5,6,7-tetrahydro-2H-indazole-3-carboxamide
N-({7-chloro-5-[2-(methylsulfanyl)pyrimidin-4-yl]-2,3-dihydro-1-benzofuran-2-yl}methyl)-2-(3-fluorophenyl)acetamide
3-acetyl-N-[3-hydroxy-1-(4-methylphenyl)propyl]-1H-pyrazole-5-carboxamide
(1R,5R)-N,N-dimethyl-6-[1-(propan-2-yl)-1H-pyrrole-2-carbonyl]-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
1-[(2-chlorophenyl)methyl]-N,N-bis(prop-2-en-1-yl)-1H-1,2,3-triazole-4-carboxamide
6-{[2-(2-fluorophenyl)-1H-imidazol-1-yl]methyl}-1H-indole
8-(3-hydroxy-2-methylbenzoyl)-2-(3-methylbut-2-en-1-yl)-2,8-diazaspiro[4.5]decan-3-one
2-amino-3-ethyl-N-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
4-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}benzonitrile
4,4-difluoro-1-{[2-(4-methoxynaphthalen-1-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine