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3-(2-ethyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-4,6-dimethyl-1,2-dihydropyridin-2-one
3-(1-cyclohexyl-1H-pyrazol-5-yl)-1-methyl-1-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}urea
4-methoxy-N-{1-[1-(5-propyl-1,2-oxazole-3-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
1-[3-(4-fluorophenyl)-1H-pyrazole-5-carbonyl]-2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine
2-({3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl}methyl)pyridine
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-1-(difluoromethyl)-1H-pyrazole-3-carboxamide
4-[3-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]-1-(4-methylphenyl)butan-1-one
1-(4-butylphenyl)-3-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]urea
3-{[4-(2-methylpropyl)-1H-1,2,3-triazol-1-yl]methyl}-1-(3-propyl-1H-pyrazole-5-carbonyl)piperidine
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)morpholine-4-carboxamide
1-benzyl-4-(2-cyclopentylacetyl)-6-(cyclopropylmethoxy)-1,4-diazepan-2-one
3-(dimethyl-1,2-oxazol-4-yl)-1-{3-[4-(trifluoromethyl)benzoyl]piperidin-1-yl}propan-1-one
6-{[1-(4-acetylpiperazin-1-yl)hex-5-en-2-yl]oxy}pyridine-3-carbonitrile
5-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyridin-2-amine
1-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanoyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-4-(thiophen-2-yl)butanamide
1-[({2-[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]ethyl}carbamoyl)methyl]piperidine-4-carboxamide
N-(2-chlorophenyl)-3-{1-[(3-methyl-1H-indol-2-yl)methyl]piperidin-4-yl}propanamide
2-{[4-cyclohexyl-3-(2-hydroxyethyl)piperazin-1-yl]methyl}-3-methoxyphenol
2-{1-ethyl-8-[(1-methyl-1,2,3,4-tetrahydroquinolin-6-yl)methyl]-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-3-yl}acetamide
methyl 4-[(5S,9aS,9bS)-1-oxo-2-(2-phenylethyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-5-yl]benzoate
(1S,5R)-3-(trimethylpyrimidin-4-yl)-3,9-diazabicyclo[3.3.2]decan-10-one
3-(2H-1,3-benzodioxol-5-yl)-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-3-phenylpropanamide
N-[(2-{2-[(dimethylsulfamoyl)amino]phenyl}-5-methyl-1,3-oxazol-4-yl)methyl]-2,6-difluorobenzamide
6-{1-[2-amino-6-(propan-2-yloxy)pyrimidin-4-yl]piperidin-4-yl}-2-methylpyrimidin-4-ol
methyl 2-(1-{2-methylthieno[2,3-d]pyrimidin-4-yl}pyrrolidin-3-yl)acetate
[2-(4-cyclobutanecarbonylmorpholin-2-yl)ethyl]dimethylamine
ethyl 4-{6-[2-(naphthalen-2-yl)acetyl]-6-azaspiro[2.5]octane-1-amido}piperidine-1-carboxylate
5-methyl-N-(pyridin-4-ylmethyl)-4-[(1,2,3,4-tetrahydronaphthalen-1-yl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
6-methyl-5-[5-(1,3-thiazol-4-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridine
3-[2-({[2-(azocane-1-carbonyl)-6-chloroimidazo[1,2-a]pyridin-3-yl]methyl}amino)ethyl]-1,3-oxazolidin-2-one
3-chloro-N-({3-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-N-(pyridin-2-ylmethyl)benzamide
2-[(5-ethylfuran-2-yl)methyl]-7-[(2-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
3-(4-fluorophenyl)-N-{2-[(pyridin-3-yl)amino]ethyl}-1H-pyrazole-5-carboxamide
2-(2,4-dimethoxyphenyl)-1-[4-(1-hydroxy-2-phenylethyl)piperidin-1-yl]ethan-1-one
{1-[(3,5-dimethoxyphenyl)methyl]-4-(2-phenoxyethyl)piperidin-4-yl}methanol
1-[1'-(pyridin-2-ylmethyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
[(3-methyl-1H-indol-2-yl)methyl]({[2-(morpholin-4-yl)pyridin-3-yl]methyl})amine
5-cyclopropyl-3-[1-(2-ethoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-1,2-oxazole
5-{3-[5-methyl-2-(pyridin-3-yl)pyrimidin-4-yl]piperidine-1-carbonyl}-1H-indole
1-(6-methoxy-2,3-dihydro-1H-indene-5-carbonyl)-4-(1-methyl-1H-imidazol-2-yl)piperidine
2-[(2-methoxyethyl)(methyl)amino]-1-{2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}ethan-1-one
3-cyclopropyl-N-{[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methylpropanamide
2-[2-methyl-3-({[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]amino}methyl)-1H-indol-1-yl]acetamide
(3S,5R)-5-(cyclopropylcarbamoyl)-1-[2-(2-fluorophenyl)acetyl]piperidine-3-carboxylic acid
(1S,6R)-9-{3-fluoro-7-methylimidazo[1,2-a]pyridine-2-carbonyl}-3-methyl-3,9-diazabicyclo[4.2.1]nonan-4-one
N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-N-methyl-2-({6-[4-(pyridin-2-yl)piperazin-1-yl]pyridazin-3-yl}oxy)acetamide
N-({7-[4-(2,5-dimethoxybenzoyl)benzoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)acetamide
2-(furan-2-yl)-2-oxo-N-{[1-(thiophen-2-ylmethyl)pyrrolidin-3-yl]methyl}acetamide
1-[(2-chlorophenyl)methyl]-3-{[(1-hydroxy-2-methylpropan-2-yl)amino]methyl}-6-methyl-1,2-dihydroquinolin-2-one