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N-{6-[2-(2,2-dimethyloxan-4-yl)-1H-imidazol-1-yl]-1,3-benzothiazol-2-yl}acetamide
2-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-6-(methoxymethyl)pyridine
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)propan-2-yl]-6-(dimethylamino)pyridine-3-carboxamide
(2S,4R)-4-amino-1-[1-(2-chlorophenyl)piperidin-4-yl]-N,N-diethylpyrrolidine-2-carboxamide
5-{4-[(3-fluorophenyl)methyl]piperazine-1-carbonyl}-4-methyl-2-oxo-1,2-dihydropyridine-3-carbonitrile
1-cyclopropanecarbonyl-N-[1-(1-propyl-1H-1,2,4-triazol-5-yl)ethyl]piperidine-4-carboxamide
1-[5-({[(3,4-difluorophenyl)methyl]amino}methyl)-2-methoxyphenoxy]-3-(piperidin-1-yl)propan-2-ol
N-[(6-methoxy-1H-1,3-benzodiazol-2-yl)methyl]-1-[(2E)-3-phenylprop-2-en-1-yl]-1H-1,2,3-triazole-4-carboxamide
5-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}-2-(pyridin-3-yl)pyrimidine
6-({[3-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-4-yl]methyl}amino)-2-methylheptan-2-ol
1-{4-[(2,2-dimethylmorpholin-4-yl)methyl]phenoxy}-3-(piperidin-1-yl)propan-2-ol
3-(2-chlorophenyl)-1-(2-methoxyethyl)-3-{2-oxo-2-[4-(pyridin-3-ylmethyl)piperazin-1-yl]ethyl}pyrrolidine-2,5-dione
2-[3-(3-methoxyphenyl)-1H-pyrazole-5-carbonyl]-2,7-diazaspiro[4.5]decane
1-[(3R,4S)-3-amino-4-phenylpyrrolidin-1-yl]-3-(dimethyl-1,2-oxazol-4-yl)propan-1-one
6-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-2-carboxylic acid
N-[(2-{4-[3-(4-methoxyphenyl)propanamido]phenyl}-5-methyl-1,3-oxazol-4-yl)methyl]-5-methyl-1,2-oxazole-3-carboxamide
N-({3-[(4-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazol-5-yl}methyl)-3,5,7-trimethyl-1H-indole-2-carboxamide
1-[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]-3-[1-(1-cyclopropylethyl)-4-methyl-1H-pyrazol-5-yl]urea
N-({4-[2-(piperidin-1-yl)ethoxy]phenyl}methyl)-N-(pyridin-2-ylmethyl)acetamide
1-{4-[(cyclobutylamino)methyl]-2-methoxyphenoxy}-3-[cyclohexyl(methyl)amino]propan-2-ol
1-(1H-pyrazol-3-ylmethyl)-4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidine
(4aS,7aR)-1-(furan-3-carbonyl)-4-(3-methylbutanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-[1-(pyrrolidin-1-yl)ethyl]-1-{[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}piperidine
2-{1-cyclopentyl-4-[5,6-dimethyl-2-(trifluoromethyl)pyrimidin-4-yl]piperazin-2-yl}ethan-1-ol
[5-(1-{4-[(E)-2-(pyridin-2-yl)ethenyl]phenyl}-1H-imidazol-2-yl)furan-2-yl]methanol
1-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)-4-(1H-pyrrole-2-carbonyl)piperazine
N-[1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-4-sulfamoylbenzamide
(1-{2-[(4-methoxyphenyl)methyl]-1,3-benzoxazole-6-carbonyl}piperidin-4-yl)methanol
9-methoxy-N-methyl-3-[3-(4-methylphenyl)propanoyl]-7-oxo-N-(thiophen-3-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
methyl 2-({[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)amino)acetate
2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]-N-(pyridin-2-ylmethyl)acetamide
1-cyclopentyl-3-(2-methoxyphenyl)-3-[2-oxo-2-(3-oxo-4-phenylpiperazin-1-yl)ethyl]pyrrolidine-2,5-dione
3-(dimethyl-1,2-oxazol-4-yl)-1-[(1R,5R)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]propan-1-one
5-methyl-N-[1-phenyl-2-(pyrrolidin-1-yl)ethyl]-1-propyl-1H-pyrazole-4-carboxamide
1-(cyclobutylmethyl)-4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine
(1S,5R)-3-(1-benzylpiperidin-4-yl)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonane
1-[3-(2-chlorophenoxymethyl)-5-(pyridin-4-yl)-1H-1,2,4-triazol-1-yl]butan-2-ol
1-{3-[3-(3-methoxybenzoyl)piperidine-1-carbonyl]phenyl}imidazolidin-2-one
N-(4-{5-pentyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}phenyl)acetamide
N-ethyl-N-(oxolan-2-ylmethyl)-1,3-benzothiazole-6-carboxamide
2-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine
1-(2,4-dimethylphenyl)-4-{[2-(4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazine
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-2-(4H-1,2,4-triazol-4-yl)pyridine-4-carboxamide
3-{[(1-{1-[(4-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperidin-3-yl)oxy]methyl}pyridine
(2E)-3-(2-chlorophenyl)-1-(4-{5-[(1E)-prop-1-en-1-yl]-2-(pyridin-3-yl)pyrimidin-4-yl}piperidin-1-yl)prop-2-en-1-one
[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl](methyl)[(2E)-2-methyl-3-phenylprop-2-en-1-yl]amine
(1S,5R)-3-(6-cyclopropylpyrimidin-4-yl)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
1'-[2-(1H-imidazol-2-yl)benzoyl]-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
1-(cyclohexylmethyl)-N,N-dimethyl-5-{[(4-phenyl-1,3-thiazol-2-yl)methyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-{1-[1-(dimethylsulfamoyl)piperidin-4-yl]-1H-pyrazol-5-yl}-4-phenylbutanamide