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1-[(4-acetylphenyl)methyl]-4-(3-fluorophenoxy)piperidine-4-carboxylic acid
N-{[7-(5-acetyl-2-fluorophenyl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-[(4S,6R)-6-methyl-2-sulfanylidene-1,3-diazinan-4-yl]acetamide
2-{5-methyl-4-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]-1H-pyrazol-1-yl}pyridine
N-methyl-3-(1-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}piperidin-3-yl)-N-[2-(pyridin-2-yl)ethyl]propanamide
5-[2-(3-methoxypropyl)piperidine-1-carbonyl]pyridin-2-amine
4-methyl-5-{1-[1-(thiophen-2-yl)ethyl]-1H-imidazol-2-yl}-1H-imidazole
[1-(5-cyclopropyl-1,3-oxazole-4-carbonyl)piperidin-4-yl]diphenylmethanol
2,8-dimethyl-4-[2-(1-methyl-1H-pyrazol-3-yl)piperidine-1-carbonyl]quinoline
1-methyl-6-(pyridin-4-ylmethyl)-3-[4-(trifluoromethoxy)phenyl]-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
methyl (2S,4S)-4-{2-[(dimethylamino)methyl]-1,3-thiazole-4-amido}-1-methylpyrrolidine-2-carboxylate
1-{1-[5-(1H-imidazol-1-ylmethyl)pyridin-2-yl]piperidin-4-yl}-2-phenylethan-1-ol
4-methyl-3-{2-[4-(4-methylphenoxy)piperidin-1-yl]-2-oxoethyl}piperazin-2-one
(5S,9aS,9bS)-5-(1-benzothiophen-2-yl)-2-[(2-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-[(2R,3R)-1'-[(3-hydroxy-4-methoxyphenyl)methyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
3-{3-[(2,3-dihydro-1,4-benzodioxin-6-yl)amino]piperidine-1-carbonyl}-5,6-dimethyl-1,2-dihydropyridin-2-one
(3R,5S)-N-[2-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-5-(morpholine-4-carbonyl)piperidine-3-carboxamide
N-[(1-ethylpyrrolidin-2-yl)methyl]-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-2-{[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}acetamide
(3S,4S)-1-[(2,6-dichloro-3-hydroxyphenyl)methyl]-4-(pyrrolidin-1-yl)pyrrolidin-3-ol
1-tert-butyl-N-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-N-methyl-5-oxopyrrolidine-3-carboxamide
2-{[(1-{[1,2,4]triazolo[1,5-a]pyrimidine-2-carbonyl}piperidin-4-yl)oxy]methyl}pyridine
2-{[1-(2,5-difluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}pyridine
5-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)-3-[4-(trifluoromethyl)phenyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
1-[(3R,4R)-3-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
(4aR,7aS)-1-(2-methoxyethyl)-4-{2-[methyl(phenyl)amino]acetyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3,6-dimethyl-N-[2-(4-methyl-1H-imidazol-2-yl)ethyl]-1-benzofuran-2-carboxamide
N-(3-cyano-4-methylphenyl)-3-(dimethylamino)pyrrolidine-1-carboxamide
1-ethyl-3-[2-(4-fluorophenyl)piperidine-1-carbonyl]-6-methyl-1,2-dihydropyridin-2-one
3-[(4-methylpiperazin-1-yl)sulfonyl]-5-(pyridin-3-yl)benzoic acid
N-[(3R,4S)-4-cyclopropyl-1-(4-fluorobenzoyl)pyrrolidin-3-yl]-3-(pyridin-3-yl)propanamide
3-{1-[2-(2-chlorophenyl)acetyl]piperidin-3-yl}-N-methyl-N-[2-(pyridin-2-yl)ethyl]propanamide
N-{[1-(2,3-dimethylquinoxaline-6-carbonyl)piperidin-3-yl]methyl}-4-fluorobenzamide
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-1-ethyl-1H-pyrazole-4-carboxamide
N-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
4-(1-cyclohexyl-1H-1,2,3-triazole-4-carbonyl)-1-[(3-methylphenyl)methyl]piperazin-2-one
2-(morpholin-4-yl)-N-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]-2-(pyridin-3-yl)acetamide
3-fluoro-N-{1-[1-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
2-benzyl-8-[2-(pyridin-2-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
1-cyclohexyl-4-[(1-methyl-1H-pyrazol-5-yl)methyl]-1,4-diazepane
2-(furan-2-yl)-1-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}azepane
N4,N4,5-trimethyl-N2-[1-(morpholin-4-ylmethyl)cyclopentyl]pyrimidine-2,4-diamine
8-(2,3-dimethyl-1H-indole-5-carbonyl)-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
4-[1-(2,5-difluorobenzoyl)piperidin-3-yl]-5-(4-fluorophenyl)-2-methylpyrimidine
2-({2-[(4-methoxyphenyl)methyl]morpholin-4-yl}methyl)-1-methyl-1H-1,3-benzodiazole
3-(3-fluorophenyl)-3-{2-oxo-2-[2-(1,3-thiazol-2-yl)piperidin-1-yl]ethyl}-1-(pyridin-3-ylmethyl)pyrrolidine-2,5-dione
N-[(1-methylpiperidin-4-yl)methyl]-4-(2-oxopiperidin-1-yl)-N-(2-phenylethyl)butanamide
11-{[(2,6-difluorophenyl)methyl]amino}-4-[2-(morpholin-4-yl)ethyl]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl)(thiophen-3-ylmethyl)amine
5-(2-{[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]amino}ethyl)-1-(cyclohexylmethyl)pyrrolidin-2-one
3-hydroxy-1-methyl-3-{[4-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]methyl}piperidin-2-one
2-{1-[(2-ethoxyphenyl)methyl]-4-{[2-(2-methylphenyl)pyrimidin-5-yl]methyl}piperazin-2-yl}ethan-1-ol