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9-methoxy-3-[2-(3-methoxyphenyl)acetyl]-7-oxo-N-(thiophen-3-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-(3-ethoxypropyl)-3-[(3S,4R)-1-(pyridin-3-ylmethyl)-4-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-3-yl]propanamide
{[2-(2-methylpropoxy)-7-(methylsulfanyl)quinolin-3-yl]methyl}(pyridin-4-ylmethyl)amine
3-(3-fluorophenyl)-1-[2-(piperidin-1-yl)ethyl]-6-(1,2,5-thiadiazole-3-carbonyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
5-[6-amino-5-cyano-4-(3-ethyl-1H-pyrazol-5-yl)pyridin-2-yl]-2,4-dimethyl-1H-pyrrole-3-carboxylic acid
(3S,4S)-1-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-4-cyclopropylpyrrolidine-3-carboxylic acid
N,1,6-trimethyl-N-{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-(4-{[3-(morpholin-4-yl)piperidin-1-yl]methyl}phenyl)imidazolidin-2-one
8-[(2,3-difluorophenyl)methyl]-1-(3-methylbutyl)-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-4-(naphthalen-1-yl)-4H-1,2,4-triazole
methyl 8-(2-cyclopentyl-2-phenylacetyl)-1-(2-methoxyethoxy)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
5-{2-[(1-methoxypropan-2-yl)amino]ethyl}-1,3,4-thiadiazol-2-amine
1-ethyl-7-methyl-N-(2-methylpropyl)-4-oxo-N-(3-phenylprop-2-yn-1-yl)-1,4-dihydro-1,8-naphthyridine-3-carboxamide
2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}-1-[2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]ethan-1-one
methyl 3-(2-fluorobenzoyl)-7-oxo-9-[2-(thiophen-3-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]-1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperidine
4-[3-(2-fluorophenyl)pyrrolidine-1-carbonyl]-1,2-dihydroquinolin-2-one
1-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]-4-(2-phenoxyethyl)piperazine
2-(piperidine-1-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
4-methyl-N-({5-methyl-2-[3-(3-methylbutanamido)phenyl]-1,3-oxazol-4-yl}methyl)pentanamide
4-[4-(1H-imidazol-1-ylmethyl)phenyl]pyridine
3-hydroxy-1-{[4-(propan-2-yl)phenyl]methyl}-3-({[2-(1,3-thiazol-4-yl)ethyl]amino}methyl)piperidin-2-one
N-{[2-(dimethylamino)pyridin-3-yl]methyl}-2-(3-fluoro-4-hydroxyphenyl)acetamide
[(3R,4R)-1-[(2,3-dimethoxyphenyl)methyl]-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
8-fluoro-N-{[1-(furan-2-ylmethyl)piperidin-3-yl]methyl}-4-oxo-1,4-dihydroquinoline-2-carboxamide
1-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-5-(2-methylprop-1-en-1-yl)-4-phenyl-1H-imidazole
5-[1-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}acetyl)piperidin-4-yl]-3-(oxolan-2-ylmethyl)-5-propylimidazolidine-2,4-dione
methyl 3-(3-chlorothiophene-2-carbonyl)-7-oxo-9-(pyridin-2-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
(3aR,6aS)-5-(6-chloro-8-methylquinolin-4-yl)-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-tert-butyl-4-[4-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]pyrrolidin-2-one
N3-cyclooctyl-N5-(3-methylbutyl)-4-oxo-1-(pyridin-2-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
N-methyl-3-{1-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]piperidin-3-yl}-N-(1-methylpiperidin-4-yl)propanamide
2-(3,4-dimethoxyphenyl)-N-{[5-fluoro-7-(pyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-4-(pyrazin-2-yl)-1,4-diazepan-6-ol
5-(5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-sulfonyl}thiophen-3-yl)-1,2-oxazole
1-(2-methoxyethyl)-N-methyl-N-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}-6-oxopiperidine-3-carboxamide
3-[1-(4-methyl-1,2,5-oxadiazole-3-carbonyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)propanamide
3-(1H-1,2,3-benzotriazol-1-yl)-1-[4-(3-methylpyridin-4-yl)-1,4-diazepan-1-yl]propan-1-one
7-(2-methoxypyridine-3-carbonyl)-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
2-[6-oxo-4-(pyrrolidin-1-yl)-1,6-dihydropyridazin-1-yl]-N-[2-(pyridin-3-yloxy)ethyl]acetamide
4-[2-fluoro-6-(propan-2-yloxy)phenyl]-3-methylpyridine
8-cyclopropanecarbonyl-2-(3-fluorobenzoyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-methyl-2-(2-{methyl[(5-methyl-1H-pyrazol-3-yl)methyl]amino}-4-(morpholin-4-yl)pyrimidin-5-yl)propanoic acid
5-cyclopropyl-N-methyl-1-[5-methyl-4-(thiophen-2-yl)pyrimidin-2-yl]-N-[2-(pyridin-2-yl)ethyl]-1H-pyrazole-4-carboxamide
2-ethyl-5-[(2S)-2-(methoxymethyl)pyrrolidine-1-carbonyl]pyrimidine
4-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-N,N-dimethylaniline
N-(1-{1-[(2-hydroxy-5-methoxyphenyl)methyl]piperidin-4-yl}-2-(3-methoxyphenyl)ethyl)-N-methylfuran-2-carboxamide
4-[6-(5-fluoro-2-methoxyphenyl)pyridine-3-carbonyl]morpholine
ethyl 1-{[4-(2-hydroxyethoxy)phenyl]methyl}-4-[(3-methoxyphenyl)methyl]piperidine-4-carboxylate
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-[3-(pyrrolidin-1-yl)propyl]pyrimidin-2-amine