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3-(2-chlorophenyl)-1-methyl-3-[2-oxo-2-(3-propanoylpiperidin-1-yl)ethyl]pyrrolidine-2,5-dione
3-fluoro-6-methyl-N-[(3R)-piperidin-3-yl]imidazo[1,2-a]pyridine-2-carboxamide
4-{1-[4-(1H-pyrazol-4-yl)butanoyl]pyrrolidin-3-yl}benzoic acid
5-hydroxy-N-[1-(pyridin-4-yl)propyl]pyridine-2-carboxamide
2-[4-(5-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-methyl-4H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]benzonitrile
2-[5-(2-methylpyrimidin-5-yl)-4-phenyl-1H-imidazol-1-yl]acetic acid
1-(3-phenyl-1,2,4-thiadiazol-5-yl)-4-{1H-pyrrolo[2,3-b]pyridin-6-yl}piperazine
(2S,4S)-4-amino-1-{2-[(5-methyl-1H-1,3-benzodiazol-2-yl)sulfanyl]acetyl}-N-(propan-2-yl)pyrrolidine-2-carboxamide
4-{4-[(1H-indol-2-ylmethyl)amino]piperidin-1-yl}-N-[(3S)-2-oxoazepan-3-yl]benzamide
5-{1-[3-(2H-1,3-benzodioxol-5-yl)propanoyl]piperidin-4-yl}-3-(2,3-dihydro-1H-inden-2-yl)-5-methylimidazolidine-2,4-dione
3-butyl-4-[4-hydroxy-2-(pyridin-3-yl)pyrimidine-5-carbonyl]-1-methylpiperazin-2-one
1-{3-fluoro-5-methylimidazo[1,2-a]pyridine-2-carbonyl}-4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine
2-(4-methoxy-3,5-dimethylphenyl)pyridine-4-carbonitrile
7-(cyclobutylmethyl)-2-(5-propyl-1,3,4-thiadiazol-2-yl)-2,7-diazaspiro[4.5]decan-6-one
5-[(3-fluorophenyl)methyl]-5-{1-[2-(3-methyl-1H-pyrazol-1-yl)acetyl]piperidin-4-yl}-3-(2-methylpropyl)imidazolidine-2,4-dione
2-(1-oxo-1,2-dihydroisoquinoline-4-carbonyl)-7-propyl-2,7-diazaspiro[4.5]decan-6-one
methyl 3-{[(2S)-4-methyl-2-phenylpiperazine-1-carbonyl]amino}benzoate
1-[3-(2H-1,3-benzodioxol-5-yl)propanoyl]-4-(pyrimidin-2-yl)piperazine-2-carboxylic acid
N-(5-methanesulfonamido-2-methylphenyl)-3-(4H-1,2,4-triazol-3-yl)piperidine-1-carboxamide
6-[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-N,N-dimethylpyridine-2-carboxamide
2-[(2-phenylazetidin-1-yl)sulfonyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
4-[4-(3-methoxybenzoyl)piperazin-1-yl]-4-oxobutane-1-sulfonamide
[(2,5-dimethoxyphenyl)methyl](methyl){[5-(methylsulfanyl)-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl]methyl}amine
N-[(3S)-1-({4-[4-(furan-3-yl)-6-oxo-1,6-dihydropyrimidin-2-yl]phenyl}methyl)pyrrolidin-3-yl]acetamide
N-cyclopropyl-1-[(3-methoxyphenyl)methyl]-5-(4-methyl-2-oxopentanoyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[(3S,4R)-1-(2-methyl-1H-1,3-benzodiazole-5-carbonyl)-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
3-[2-methoxy-5-(pyrrolidin-1-ylmethyl)phenoxy]-6-phenylpyridazine
3,4-difluoro-N-{2-[4-(4-fluorophenyl)-5-{[(2-methylphenyl)methyl]sulfanyl}-4H-1,2,4-triazol-3-yl]ethyl}benzene-1-sulfonamide
(3R,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-7-({[3-(methylsulfanyl)phenyl]methyl}amino)-octahydropyrrolo[1,2-a]piperazine-1,4-dione
4-({1-[(2E)-4-methylpent-2-en-1-yl]piperidin-4-yl}oxy)-N-(pyridin-2-ylmethyl)benzamide
methyl 5-oxo-5-(3-{[4-(1,3-thiazol-4-yl)phenyl]carbamoyl}piperidin-1-yl)pentanoate
3-(2-methylphenyl)-3-phenyl-N-(1-propylpiperidin-4-yl)propanamide
3-{[(1R,3S,5S)-3-hydroxy-8-azabicyclo[3.2.1]octan-8-yl]methyl}-6,8-dimethyl-1,2-dihydroquinolin-2-one
2-(3-chlorophenyl)-1-[2-(1H-imidazol-4-yl)ethyl]-1H-imidazole
N-(2H-1,3-benzodioxol-5-yl)-3-[4-(trifluoromethyl)benzoyl]piperidine-1-carboxamide
3-({[1-(1H-imidazol-2-ylmethyl)piperidin-4-yl]oxy}methyl)pyridine
3-[1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)piperidin-4-yl]-N-(2-methoxyethyl)propanamide
2-(1-butyl-1H-pyrazol-4-yl)-7-fluoro-4-(morpholine-4-carbonyl)quinoline
2-[2,5-dioxo-3-phenyl-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]-N-methyl-N-[(4-methylphenyl)methyl]acetamide
methyl 1-benzyl-3-cyclopropaneamido-5-[(oxan-4-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
3-(4-chlorophenyl)-N-methyl-3-phenyl-N-(1,3-thiazol-2-ylmethyl)propanamide
1-{3-[(3R,4R)-3-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-(hydroxymethyl)pyrrolidine-1-carbonyl]phenyl}ethan-1-one
3-methoxy-4-({3-[5-(2-methylphenyl)-2-(pyridin-4-yl)pyrimidin-4-yl]piperidin-1-yl}methyl)phenol
1-{5-cyclobutanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-ethoxyethan-1-one
5-fluoro-1-methyl-2-({4-[(3-methylphenyl)methyl]piperazin-1-yl}methyl)-1H-indole
1-(4-fluorophenyl)-4-[1-(2-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]butane-1,4-dione
3,5-dimethyl-N-(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-yl)-1,2-oxazole-4-carboxamide
[2-(2-chloro-6-methylphenoxy)ethyl]({3-[(dimethylamino)methyl]phenyl}methyl)amine
(3S,9aR)-8-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3-propyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
[(2-fluorophenyl)methyl][1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]amine