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2-(dimethyl-1,2-oxazole-4-carbonyl)-7-(pyrrolidine-1-sulfonyl)-1,2,3,4-tetrahydroisoquinoline
1-(5-propyl-1,2-oxazole-3-carbonyl)-4-(1,3-thiazol-2-yl)piperazine
N-[(3S,5S)-5-(diethylcarbamoyl)-1-(furan-2-ylmethyl)pyrrolidin-3-yl]-3-methyl-1,2-oxazole-5-carboxamide
3-benzyl-8-[1-(2-fluorophenyl)propan-2-yl]-1-(3-methoxypropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-amino-4-methyl-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}-1,3-benzothiazole-6-carboxamide
methyl 7-oxo-9-(3-phenylpropoxy)-3-(pyrazine-2-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
{[3-(2,4-dimethoxyphenyl)-1H-pyrazol-4-yl]methyl}[(1-ethyl-1H-imidazol-2-yl)methyl]methylamine
1-cyclohexanecarbonyl-N-methyl-N-(1H-pyrazol-5-ylmethyl)pyrrolidine-2-carboxamide
3-{1-[4-phenyl-5-(1-propyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]ethyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
4-[5-(1,2-oxazole-3-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl]morpholine
2-[2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetyl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
N-[2-(2-fluorophenyl)-1-[1-(quinolin-4-ylmethyl)piperidin-4-yl]ethyl]-N-methylthiophene-3-carboxamide
2-[4-(2,3-dihydro-1-benzofuran-5-ylmethyl)-6-hydroxy-1,4-diazepan-1-yl]acetic acid
3-{[2-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]methyl}-4H-chromen-4-one
3-{2-[(2-fluoro-4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-methyl-N-{[2-(trifluoromethyl)phenyl]methyl}propanamide
N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-3-(pyridin-4-yl)-1H-pyrazole-5-carboxamide
4-{4-[(3R)-3-hydroxypyrrolidine-1-carbonyl]benzenesulfonyl}-1-methylpiperazin-2-one
1-(1-{2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetyl}piperidin-3-yl)-3-phenylpropan-1-one
N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)-1-oxo-1,2-dihydroisoquinoline-4-carboxamide
(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-6-(2-methoxypyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-{[(1R,9aR)-1-hydroxy-octahydro-1H-quinolizin-1-yl]methyl}-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-cyclopropyl-1-[(3-methoxyphenyl)methyl]-5-(quinoxaline-5-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-(oxolan-2-ylmethyl)cyclohex-1-ene-1-carboxamide
[4-(6-methoxypyrimidin-4-yl)phenyl]methanol
[(3S,5R)-1-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-4-yl]-5-[(dimethylamino)methyl]piperidin-3-yl]methanol
2,3,4-trimethoxy-N-{[8-(3-methylbutanoyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}benzamide
1-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}-4-[(3-methylpyridin-2-yl)methyl]piperazine
methyl 3-({[1-(2-methoxyethyl)piperidin-4-yl]methyl}(oxolan-2-ylmethyl)carbamoyl)propanoate
3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)-1-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}propan-1-one
N-cyclopropyl-3-{methyl[2-(oxan-4-yl)ethyl]sulfamoyl}benzamide
2-methyl-1-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
1-[2-(3-chlorophenyl)ethyl]-2-(methoxymethyl)-6-methyl-3-[4-(2-methylphenyl)piperazine-1-carbonyl]-1,4-dihydropyridin-4-one
7-(2-cyclohexylethyl)-2-(thiophene-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
6-ethyl-2-methyl-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}quinoline-4-carboxamide
N-(1-{7-[(2-fluoro-5-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)pyridine-2-carboxamide
N,N-diethyl-3-{[1-(1-methyl-1H-pyrazol-5-yl)propyl]sulfamoyl}benzamide
3,4,7-trimethyl-2-(4-phenyl-1,4-diazepane-1-carbonyl)-1H-indole
8-{6-cyclopropyl-3-methyl-[1,2]oxazolo[5,4-b]pyridine-4-carbonyl}-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
N-[(4-fluoro-3-methylphenyl)methyl]-N-(3-methoxypropyl)-1-methylpiperidin-4-amine
2-(2-phenylethyl)-9-(pyrimidin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
5-methoxy-1-methyl-N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]-1H-indole-2-carboxamide
9-{3-[(2-methylprop-2-en-1-yl)oxy]benzoyl}-3-oxa-9-azaspiro[5.5]undecane
2-[(5-methylpyrazin-2-yl)methyl]-8-[2-(pyridin-3-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
1-(2-methylpropyl)-3-(pyrrolidine-1-carbonyl)-N-[2-(thiophen-2-yl)ethyl]-4,5,6,7-tetrahydro-1H-indazol-5-amine
4-(5-ethyl-1,3-oxazole-4-carbonyl)-1-(4-methoxyphenyl)-2,2-dimethylpiperazine
3-methyl-N-[1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]-5,6-dihydro-1,4-dioxine-2-carboxamide
N-[2-(5-chloro-1H-1,3-benzodiazol-2-yl)ethyl]-3-(1H-1,2,4-triazol-1-yl)propanamide
4-{2-[1-(furan-3-ylmethyl)-3-oxopiperazin-2-yl]acetyl}-1-[(4-methylphenyl)methyl]piperazin-2-one
(1S,9R)-11-[5-(2-chloro-4-fluorophenoxymethyl)-1,2-oxazole-3-carbonyl]-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
1,3-dimethyl-N-[(3-methylpyridin-2-yl)methyl]-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine