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1-{3-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-4-(morpholin-4-yl)phenyl}ethan-1-one
N-[(4-chlorophenyl)(pyridin-4-yl)methyl]-2-(propan-2-yl)-1,3-benzoxazole-5-carboxamide
3-(dimethyl-1H-1,2,4-triazol-3-yl)-1-[2-(6-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]urea
3-[(2,4-difluorophenyl)methyl]-1-(6-ethylpyrimidin-4-yl)piperidine-3-carboxylic acid
1-[9-hydroxy-7-(4-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(2-methoxyethoxy)ethan-1-one
4-(1H-pyrazol-3-yl)-N-{2-[3-(trifluoromethyl)phenyl]ethyl}benzamide
2-(naphthalen-1-ylmethyl)-4-[3-(1H-pyrazol-1-yl)propyl]morpholine
1-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-4-(3-phenylpropyl)-1,4-diazepane
3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-1-(4-phenyl-1,2,3,6-tetrahydropyridin-1-yl)propan-1-one
N-[(3S,4R)-1-{4-[(5-methyl-1H-1,2,3,4-tetrazol-1-yl)methyl]benzoyl}-4-propylpyrrolidin-3-yl]acetamide
methyl 5-[(4-hydroxybutan-2-yl)amino]-1-methyl-3-(3-phenylpropanamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-{3-[1-(cyclohexylmethyl)-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-5-yl]propyl}pyrrolidin-2-one
2-(ethoxymethyl)-N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-{[4-(but-3-yn-1-yloxy)phenyl]methyl}-N-(oxolan-2-ylmethyl)-4-(1H-pyrazol-1-yl)benzamide
({4-ethyl-5-[1-(6-methylpyridazin-3-yl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
N-({7-[2-(4-methoxyphenyl)acetyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2H-1,3-benzodioxole-5-carboxamide
4-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]-N-[(3-phenyl-1H-pyrazol-4-yl)methyl]butanamide
ethyl 2-[9-(2-methoxybenzoyl)-3,9-diazaspiro[5.5]undecan-3-yl]acetate
(4aS,7aR)-1-{[5-(2-methylpropyl)thiophen-2-yl]methyl}-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-[1-(2,3-dihydro-1-benzofuran-2-carbonyl)piperidin-4-yl]-5-[(4-fluorophenyl)methyl]-3-(2-methoxyethyl)imidazolidine-2,4-dione
2-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]benzamide
4-({4-methyl-5-[1-(6-methylpyrimidin-4-yl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)morpholine
2-(4-{5-methyl-4-[(3-phenylpropyl)amino]thieno[2,3-d]pyrimidine-6-carbonyl}piperazin-1-yl)ethan-1-ol
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-1-(7-methoxy-4-methylquinazolin-2-yl)piperidine-3-carboxamide
4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]-1-(5-methoxyfuran-2-carbonyl)piperidine
4-[5-(cyclopent-1-en-1-ylmethyl)-3-(oxolan-3-yl)-1H-1,2,4-triazol-1-yl]benzonitrile
2-(4-{[5-methyl-2-(1H-pyrazol-1-yl)phenyl]methyl}-1-(2-phenylethyl)piperazin-2-yl)ethan-1-ol
N-(2-fluoroethyl)-3-{[(1S)-2-hydroxy-1-phenylethyl]sulfamoyl}benzamide
2-[5-cyclopropyl-4-(4-phenylpiperazine-1-carbonyl)-1H-pyrazol-1-yl]-4-(3-methoxyphenyl)pyrimidine
2-(2-ethoxypyridin-3-yl)-2-[methyl({[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl})amino]acetic acid
{1-[2-(methylamino)pyrimidine-5-carbonyl]-3-(3-methylbut-2-en-1-yl)piperidin-3-yl}methanol
N-benzyl-N-ethyl-3-(1,2,3,6-tetrahydropyridin-1-yl)propanamide
[(4-methoxy-2,3,6-trimethylphenyl)methyl]bis(1,3-oxazol-4-ylmethyl)amine
5-{1-[(3,5-dimethylphenyl)methyl]piperidin-4-yl}-5-[(4-fluorophenyl)methyl]-3-(2-methoxyethyl)imidazolidine-2,4-dione
N-[(4-{[(2-fluorophenyl)methyl]amino}-8-methylquinazolin-2-yl)methyl]-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetamide
2-{4-[(2,3-difluoro-6-methoxyphenyl)methyl]morpholin-3-yl}-1-(2,5-dihydro-1H-pyrrol-1-yl)ethan-1-one
1,6-dimethyl-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-cyclohexyl-1-{4-[2-(oxolan-2-yl)-5-(trifluoromethyl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}ethan-1-one
N-{[4-(cyclohex-3-en-1-ylmethoxy)phenyl]methyl}-N-cyclopropyl-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
1-ethyl-8-[(3-fluorophenyl)methyl]-3-[(3-methoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-{4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
(2S,4S)-N-ethyl-4-(6-methyl-4-oxo-4H-pyran-2-amido)-1-(oxan-4-yl)pyrrolidine-2-carboxamide
4-[(1R,2R)-2-phenylcyclopropanecarbonyl]-1-(2-phenylethyl)-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
1-{[2-fluoro-5-(trifluoromethyl)phenyl]methyl}-5-(2-{[(4-methoxyphenyl)methyl]amino}ethyl)pyrrolidin-2-one
1-(5-methoxy-1H-indole-2-carbonyl)-N,N-dimethylazepan-4-amine
3-(1-methyl-1H-pyrazol-4-yl)-1-[3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]propan-1-one
2-methoxy-3-methyl-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}benzamide
5-[(dimethylsulfamoyl)amino]-1-methyl-2-(2-methylpropyl)-N-[3-(methylsulfanyl)propyl]-1H-1,3-benzodiazole-7-carboxamide
4-{1-[4-(azepan-1-yl)-4-oxobutanoyl]piperidin-3-yl}benzoic acid
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)-3-(1H-1,2,3,4-tetrazol-1-yl)propanamide