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5-[(1R,3S)-1,3-dihydroxy-7-azaspiro[3.5]nonane-7-carbonyl]-2-(propan-2-yl)-3,4-dihydropyrimidin-4-one
3-methoxy-N-{2-[4-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)morpholin-2-yl]ethyl}propanamide
ethyl 4-[(4-chlorophenyl)methyl]-1-[3-(pyridin-4-yl)propanoyl]piperidine-4-carboxylate
N,1-dimethyl-N-[(3-methylthiophen-2-yl)methyl]-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-[2-(2,5-difluorophenyl)acetyl]-9-methoxy-10-(thiomorpholine-4-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
5-fluoro-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-methoxybenzamide
5-(furan-2-ylmethyl)-2-(3,4,5-trimethoxyphenyl)-2,3,4,5-tetrahydro-1,5-benzothiazepine
1-(5-methoxyfuran-2-carbonyl)-4-(3-methylphenoxy)piperidine-4-carboxylic acid
2-{1-[(1-cyclopropanecarbonylpiperidin-4-yl)methyl]-1H-1,2,3-triazol-4-yl}pyridine
5-{1-[(5-chloro-2-hydroxyphenyl)methyl]-4-hydroxypiperidin-4-yl}-N-cyclopentyl-1-benzofuran-2-carboxamide
2-{[5-(1-ethyl-1H-pyrazol-3-yl)-4-(3-methylphenyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
3-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidine-1-carbonyl]-5-chloropyridine
3-(2-chlorophenyl)-1-(cyclopropylmethyl)-6-(thiolan-3-yl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
2,6-dihydroxy-N-{3-[(5-methylpyridin-2-yl)amino]propyl}benzamide
2-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-5-(morpholin-4-yl)-2,3-dihydropyridazin-3-one
(1S,5R)-6-(3,4-diethoxybenzoyl)-3-methyl-3,6-diazabicyclo[3.2.2]nonane
N-[(3,4-dimethoxyphenyl)methyl]-3-(2-methoxyphenyl)-N-(pyridin-2-ylmethyl)propanamide
1-(4-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-(trimethyl-1H-pyrazol-1-yl)ethan-1-one
5-ethyl-5-{1-[4-methyl-3-(2-oxoimidazolidin-1-yl)benzoyl]piperidin-4-yl}-3-(2-methylprop-2-en-1-yl)imidazolidine-2,4-dione
2-{4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-1,3-benzothiazole
2-(naphthalen-1-yl)benzamide
methyl (2S,4S,5R)-4-[(2-hydroxyethyl)(methyl)carbamoyl]-1,2-dimethyl-5-phenylpyrrolidine-2-carboxylate
N-ethyl-3-(4-hydroxyphenyl)-N-(pyridin-4-ylmethyl)benzamide
1-methyl-3-{1-[(2-methylphenyl)methyl]piperidin-3-yl}-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}-3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carboxamide
5-(3-acetylphenoxymethyl)-N-[2-hydroxy-2-(prop-2-en-1-yl)pent-4-en-1-yl]-1,2-oxazole-3-carboxamide
4-methyl-6-(4-{[4-(methylsulfanyl)phenyl]methyl}piperazin-1-yl)pyrimidin-2-amine
1-(3-{[(heptan-4-yl)amino]methyl}piperidin-1-yl)-2-methylpropan-1-one
1-(4,7-dimethylquinazolin-2-yl)-N-(3-methylbutyl)piperidine-4-carboxamide
2-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]phenoxy}pyrimidine
(1,4-dioxan-2-ylmethyl)({[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl})methylamine
N-cyclopropyl-3-{1-[2-(methylsulfanyl)acetyl]piperidin-3-yl}propanamide
N,N-dimethyl-2-oxo-1,2-dihydrospiro[indole-3,3'-piperidine]-1'-sulfonamide
4-{1-[1,3-dioxo-2-(thiophen-2-ylmethyl)-2,3-dihydro-1H-isoindol-4-yl]piperidine-4-carbonyl}piperazine-1-carbaldehyde
6-{[4-(1H-1,3-benzodiazol-2-yl)cyclohexyl]methyl}-2-methyl-2H,6H,7H-pyrazolo[4,3-d]pyrimidin-7-one
N-(2H-1,3-benzodioxol-5-ylmethyl)-4-(4-{[2-methyl-2-(morpholin-4-yl)propyl]amino}piperidin-1-yl)benzamide
methyl({[3-(prop-2-en-1-yl)-4-(prop-2-en-1-yloxy)phenyl]methyl})[1-(pyridin-2-yl)ethyl]amine
{4-[1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazole-4-carbonyl]-1,4-oxazepan-6-yl}methanol
3-methyl-8-[2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)acetyl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
[(2,2-dimethyl-1-phenylcyclopropyl)methyl](methyl){4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}amine
1-(3-{[3-(dimethylamino)propyl](methyl)amino}piperidin-1-yl)-4-methylpentane-1,2-dione
2-[4-(cyclopropylmethyl)-1-(propan-2-yl)piperazin-2-yl]ethan-1-ol
3-(naphthalen-1-ylmethyl)-N-(1,2-oxazol-3-ylmethyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
3-[(3R,4S)-1-(5-cyclopropyl-3-methyl-1H-pyrazole-4-carbonyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
3-(but-2-yn-1-yl)-5-[1-(2,3-dihydro-1-benzofuran-5-ylmethyl)piperidin-4-yl]-5-(3-phenylpropyl)imidazolidine-2,4-dione
{1-[1-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methanamine
3-methyl-N-{2-[2-(pyridin-2-yl)-1H-imidazol-1-yl]ethyl}pyridin-4-amine
3-(2-acetylphenyl)-5-[(propan-2-yl)sulfamoyl]benzoic acid
1-(azepan-1-yl)-3-(2-methoxy-4-{[methyl(2-methylprop-2-en-1-yl)amino]methyl}phenoxy)propan-2-ol
N-[4-(4-{[1-(1-phenyl-1H-pyrazol-4-yl)ethyl]amino}piperidin-1-yl)phenyl]pyrazine-2-carboxamide