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2-(3-hydroxyphenyl)-N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
2-(2-fluorophenyl)-N-({5-methyl-2-[4-(2-phenylacetamido)phenyl]-1,3-oxazol-4-yl}methyl)acetamide
3-(1-methyl-1H-imidazol-2-yl)-6-{pyrazolo[1,5-a]pyridin-7-yl}pyridazine
2-[(4aR,7aS)-4-[(3-chloro-4-fluorophenyl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]acetic acid
1-methyl-N-{[1-(morpholin-4-yl)cycloheptyl]methyl}-3-propyl-1H-pyrazole-5-carboxamide
2-(2-hydroxyethyl)-3-oxo-N-(3,4,5-trifluorophenyl)piperazine-1-carboxamide
2-benzyl-9-cyclohexanecarbonyl-2,9-diazaspiro[5.5]undecan-3-one
3-[(3S,7S,8aS)-3-[(2S)-butan-2-yl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[4-(propan-2-yl)phenyl]urea
2-[7-methyl-2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-1-[4-(morpholin-4-yl)piperidin-1-yl]ethan-1-one
N-[2-(2-chlorophenyl)ethyl]-2-(furan-2-amido)-7-oxo-4,5,6,7-tetrahydro-1,3-benzothiazole-5-carboxamide
5-[(3,4-dimethoxyphenyl)methyl]-5-(3-{4-[(2-methoxyphenyl)methyl]piperazin-1-yl}-3-oxopropyl)pyrrolidin-2-one
4-{[2-(2-chlorophenyl)-2-(dimethylamino)ethyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carboxylic acid
N-({3-[(3-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazol-5-yl}methyl)-4,5,6,7-tetrahydro-2H-indazole-3-carboxamide
1-(3-chlorothiophene-2-carbonyl)-4-{[2-(trifluoromethyl)phenyl]methyl}-1,4-diazepan-5-one
5,6-dimethyl-1-[5-(pyrrolidine-1-carbonyl)furan-2-yl]-1H-1,3-benzodiazole
1-{[2-(3-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-(3-methoxyphenoxymethyl)piperidine
2-[(3-acetylphenyl)methyl]-7-(2,2-dimethylpropyl)-2,7-diazaspiro[4.5]decan-6-one
3-[4-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-1-(oxan-4-yl)piperidine
1-[(2-chlorophenyl)methyl]-N-[3-(dimethylamino)propyl]-N-methylpiperidin-3-amine
3-[(3R,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[(1R)-1-phenylethyl]urea
N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carboxamide
2-{1-[(5-propylfuran-2-yl)methyl]piperidin-2-yl}acetic acid
N-(3-hydroxy-3-phenylpropyl)-N-methyl-4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}butanamide
2-{2-methyl-1H-imidazo[4,5-b]pyridin-6-yl}benzamide
4-(2-amino-5-butyl-6-methylpyrimidin-4-yl)-1-[(4-methylphenyl)methyl]piperazin-2-one
6-(cyclopropylmethoxy)-4-[2-(pyridin-2-ylsulfanyl)acetyl]-1-(pyridin-3-ylmethyl)-1,4-diazepan-2-one
N-cyclobutyl-7-(cyclopropylmethyl)-6-(2-fluoro-4-methoxyphenyl)-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
2-(3-{[(2-hydroxy-2-phenylethyl)(methyl)amino]methyl}phenyl)-6-(propan-2-yl)-3,4-dihydropyrimidin-4-one
ethyl 4-{3-[(2H-1,3-benzodioxol-5-yl)amino]piperidin-1-yl}piperidine-1-carboxylate
1-[2-methoxy-2-(thiophen-2-yl)ethyl]-4-(1,3-thiazol-2-yl)-1H-1,2,3-triazole
3-(furan-2-yl)-N-({5-methyl-2-[4-(2-phenylacetamido)phenyl]-1,3-oxazol-4-yl}methyl)benzamide
1-[(2-tert-butyl-5-carbamoylfuran-3-yl)methyl]-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
5-chloro-2-(1-cycloheptyl-1H-1,2,3-triazole-4-carbonyl)-1,2,3,4-tetrahydroisoquinoline
N-({7-chloro-2-[3-(hydroxymethyl)piperidin-1-yl]quinolin-3-yl}methyl)-2-cyclopentyl-N-(2-methoxyethyl)acetamide
2-(6-methoxynaphthalen-2-yl)-4-[(3-methylpyridin-2-yl)methyl]morpholine
3-(3-methoxyphenyl)-N-methyl-N-(quinolin-3-ylmethyl)-1H-pyrazole-4-carboxamide
1-(azocan-1-yl)-3-(2-methoxy-5-{[methyl(pyridin-2-ylmethyl)amino]methyl}phenoxy)propan-2-ol
2,2-dimethylpropyl N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}carbamate
(4aS,7aR)-1-[(3-fluorophenyl)methyl]-4-(3-methylbutanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-(3,5-dimethylphenyl)-6-(2,7,8-trimethylquinoline-4-carbonyl)-6-azaspiro[2.5]octane-1-carboxamide
{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}(2-methoxyethyl)[(3-phenyl-1H-pyrazol-4-yl)methyl]amine
9-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
5-(methoxymethyl)-N-{4-[5-methyl-4-({[4-(methylsulfanyl)phenyl]formamido}methyl)-1,3-oxazol-2-yl]phenyl}furan-2-carboxamide
5-(1,5-dimethyl-1H-pyrazol-4-yl)-N-[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]-1,2-oxazole-3-carboxamide
2,6-diamino-4-[5-(1H-pyrazol-3-yl)thiophen-2-yl]-5,6,7,8-tetrahydroquinoline-3-carbonitrile
(2S,4R)-4-(dimethylamino)-1-[(2E)-2-methylbut-2-en-1-yl]pyrrolidine-2-carboxylic acid
ethyl({[5-(oxolan-2-yl)thiophen-2-yl]methyl})[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]amine
N-methyl-3-(2-methylpyrrolidine-1-carbonyl)-N-(thiophen-3-ylmethyl)benzene-1-sulfonamide
N-[(2R,3R)-1'-[(3-chlorophenyl)methyl]-2-(2-methoxyethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
2-(3-fluoro-4-phenylphenyl)-2-(morpholin-4-yl)acetic acid