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2-[2-(thiophene-2-carbonyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl]pyridine
N-(3-methoxypropyl)-1-methyl-5-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-{8-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-5-methyl-N-[2-(pyridin-4-yl)ethyl]-1H-pyrazole-4-carboxamide
2-(5-chloro-2-ethoxyphenyl)-2-(morpholin-4-yl)acetic acid
ethyl 4-{3-[(4-fluorophenyl)methyl]-1,2-oxazole-5-amido}piperidine-1-carboxylate
(3S)-1-[1-methyl-5-(3-propyl-1,2,4-oxadiazol-5-yl)-1H-1,3-benzodiazol-2-yl]pyrrolidin-3-ol
1-(1,2-diphenylethyl)-5-(2-{[(3-methoxyphenyl)methyl]amino}ethyl)pyrrolidin-2-one
1-(2-{3-benzyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl}-2-oxoethyl)-1,2-dihydropyrimidin-2-one
1-(1-{2-[4-(2-fluorophenyl)piperazin-1-yl]-6-(2-methoxyphenyl)pyridine-3-carbonyl}piperidin-4-yl)piperidin-4-ol
N-cyclopropyl-4-[(dipropylamino)methyl]-N-(oxan-4-yl)benzamide
N-ethyl-5-{[8-(6-methylpyridin-2-yl)-1,8-diazaspiro[4.5]decan-1-yl]methyl}pyrimidin-2-amine
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]acetamide
3-{2-[4-(2-hydroxyethyl)piperazin-1-yl]-2-oxoethyl}-3-(2-methylphenyl)-1-(pyridin-4-ylmethyl)pyrrolidine-2,5-dione
N-({1-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-3-yl}methyl)acetamide
3-{3-cyclopentyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}-4-(methoxymethyl)-5-methyl-1,2-oxazole
1-{2-[2-(4-chlorophenyl)morpholin-4-yl]-2-oxoethyl}-1,2-dihydropyrimidin-2-one
2-[1-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)-1,4-diazepan-6-yl]acetic acid
N-(cyclohexylmethyl)-3-[5-(5-methylthiophen-2-yl)-1,3,4-oxadiazol-2-yl]propanamide
N-[2-(4-fluorophenyl)ethyl]-N-{[7-methoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}furan-3-carboxamide
3-methyl-5-({4-[2-(1-methyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]phenyl}methyl)-4H-1,2,4-triazole
N-({7-[(2E)-3-(3,4-difluorophenyl)prop-2-enoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)thiophene-3-sulfonamide
(1R,5S,8R)-N,N-dimethyl-3-{[2-(piperidin-1-yl)pyrimidin-5-yl]methyl}-3-azabicyclo[3.2.1]octan-8-amine
7-acetamido-N-(furan-2-ylmethyl)-N-methyl-1-[2-(pyridin-2-yl)ethyl]-1H-1,3-benzodiazole-5-carboxamide
benzyl (7R,9aR)-7-[(1S)-1-hydroxyethyl]-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
5-methyl-2-[4-({methyl[(6-methylpyridin-2-yl)methyl]amino}methyl)phenyl]-6-(trifluoromethyl)-3,4-dihydropyrimidin-4-one
N-methyl-N-[2-(2-methyl-1H-indol-1-yl)ethyl]-4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzamide
(2S)-2-{[1-(5-ethyl-2-methylpyrimidin-4-yl)piperidin-4-yl]amino}-3-phenylpropan-1-ol
7-chloro-4-[1-methyl-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-{[8-(furan-3-carbonyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}-2-(naphthalen-1-yl)acetamide
N-[(3R,4R)-3-hydroxypiperidin-4-yl]-2-phenylimidazo[1,2-a]pyridine-6-carboxamide
2-(dimethylamino)-N-(3-methyl-1-{7-[3-(thiophen-2-yl)propanoyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}butyl)acetamide
N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carboxamide
1-methanesulfonyl-3-(4-methoxy-3,5-dimethylbenzoyl)piperidine
4-chloro-5-{[(1R,5S,8S)-8-methoxy-3-azabicyclo[3.2.1]octan-3-yl]methyl}-N,N-dimethyl-1,3-thiazol-2-amine
4-(3-phenoxypropanoyl)-1-phenylpiperazin-2-one
(5S,9aS,9bS)-5-(3-hydroxyphenyl)-2-[(5-methylfuran-2-yl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-[(2-hydroxyphenyl)methyl]-N-[4-(pyridin-3-yloxy)phenyl]piperidine-2-carboxamide
N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-(3-hydroxy-3-methylbutyl)benzamide
(3S,4R)-1-{2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]acetyl}-4-phenylpyrrolidine-3-carboxylic acid
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-N,2-dimethyl-1H-1,3-benzodiazole-6-carboxamide
(benzylsulfamoyl)[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]amine
N-({7-[4-(4-methoxyphenyl)-4-oxobutanoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(piperidin-1-yl)acetamide
{[2-(3-methoxyphenyl)-7-(methylsulfanyl)quinolin-3-yl]methyl}(methyl)(1,2-oxazol-3-ylmethyl)amine
3-(4,5-dimethyl-1H-pyrazol-3-yl)-1-[(3R,4S)-3-(dimethylamino)-4-(propan-2-yl)pyrrolidin-1-yl]propan-1-one
2-(3-chlorophenoxy)-N-ethyl-N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}propanamide
N-[3-(2,3-dihydro-1H-isoindol-2-yl)propyl]-1-methyl-6-oxo-1,6-dihydropyridazine-3-carboxamide
methyl 1-({4-[4-(2-methylpropyl)benzoyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperidine-4-carboxylate
N-(2-{7-[(2,5-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2,4-dimethylbenzamide
1-(7-chloroquinolin-4-yl)-3-(piperidin-1-ylmethyl)pyrrolidin-3-ol
(3aR,7aS)-2-{2-cyclopropyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}-2,3,3a,4,7,7a-hexahydro-1H-isoindole