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2-{1-[(3,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[2-(oxan-4-yl)ethyl]acetamide
4-[2-(furan-3-yl)pyridine-4-carbonyl]morpholine
N-[(2,5-difluorophenyl)methyl]-2-[(3,4-dimethoxyphenyl)methyl]-1,3-benzoxazole-6-carboxamide
1-{5-[1-(2-fluoro-4-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-1H-pyrazol-3-yl}ethan-1-one
methyl 2-(3-{2-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-2-yl}propanamido)acetate
9-oxo-8-(2-phenylethyl)-N-propyl-2,8-diazaspiro[5.5]undecane-2-carboxamide
1-(1-{4-methyl-6H,7H,8H-cyclopenta[g]quinazolin-2-yl}piperidine-4-carbonyl)-3-phenylpiperidine
N-{5-chloro-2-[(3S)-3-acetamidopyrrolidine-1-carbonyl]phenyl}propanamide
N-(dicyclopropylmethyl)-5-(2-methoxyacetamido)-N,1-dimethyl-2-(pyridin-4-yl)-1H-1,3-benzodiazole-7-carboxamide
4-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepin-2-yl]-3,6-dimethyl-[1,2]oxazolo[5,4-d]pyrimidine
2-(2H-1,3-benzodioxol-5-yl)-N-methyl-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
1-[4-({3-phenyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}methyl)thiophen-2-yl]ethan-1-one
6-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-N-methylpyridazin-3-amine
4-methyl-N-(3-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}butyl)benzene-1-sulfonamide
(3S,4R)-N,N-dimethyl-1-[(3-methylthiophen-2-yl)methyl]-4-(propan-2-yl)pyrrolidin-3-amine
ethyl({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]amine
N-{[1-(dimethylamino)cyclopentyl]methyl}-6-(propan-2-yl)pyrimidin-4-amine
2-[4-(pyridin-3-ylmethyl)piperazin-1-yl]pyridine-4-carboxamide
N-cyclopropyl-3-{1-[(2-hydroxyphenyl)methyl]piperidin-3-yl}propanamide
1-(cyclopropylmethyl)-4-(1-methyl-1H-imidazole-5-carbonyl)-2-(propan-2-yl)-1,4-diazepane
N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-2,6-dihydroxybenzamide
4-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonane-3-carbonyl]-2,7,8-trimethylquinoline
3-{[ethyl(2-methylprop-2-en-1-yl)amino]methyl}-7-methyl-1-(pyridin-2-ylmethyl)-1,2-dihydroquinolin-2-one
2-(3,5-dimethyl-1H-pyrazol-1-yl)-1-[4-(3-methoxybenzoyl)piperazin-1-yl]propan-1-one
(4aR,8aS)-1-(3-hydroxypropyl)-6-[(3-methoxyphenyl)methyl]-decahydro-1,6-naphthyridin-2-one
2,N3,N3-trimethyl-N7-(5,6,7,8-tetrahydronaphthalen-1-yl)-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3,7-dicarboxamide
1-[(3-fluorophenyl)methyl]-4-({2-methylthieno[2,3-d]pyrimidin-4-yl}amino)pyrrolidin-2-one
1-(4-chloro-2-methylbenzoyl)-4-(hydroxymethyl)azepan-4-ol
4-chloro-1-methyl-3-{[2-(3-methyl-1,2-oxazol-5-yl)pyrrolidin-1-yl]methyl}-1H-indazole
N-[2-({[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}amino)ethyl]-4-methylpyridin-2-amine
N-[2-(3-{[(furan-3-ylmethyl)(methyl)amino]methyl}phenoxy)propyl]naphthalene-1-carboxamide
methyl 3-(2-fluorobenzamido)-5-{[2-(3-methylphenyl)acetamido]methyl}benzoate
5-ethanesulfonamido-1-methyl-2-phenyl-N-[2-(pyridin-4-yl)ethyl]-1H-1,3-benzodiazole-7-carboxamide
5-(2-cyclohexylacetyl)-1-(2-phenylethyl)-N-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-(2-acetamidophenyl)-5-oxopyrrolidine-3-carboxylic acid
2-(3-methoxyphenyl)-N-[2-(2-oxopyrrolidin-1-yl)ethyl]-1,3-benzoxazole-6-carboxamide
6-[4-(2-methoxyphenoxy)piperidin-1-yl]-9H-purin-2-amine
2-[1-(2,3-dihydro-1H-inden-2-yl)-5-(1-methyl-1H-1,3-benzodiazol-5-yl)-1H-1,2,4-triazol-3-yl]acetamide
1-(2-{1-[(3-methylthiophen-2-yl)sulfonyl]piperidin-2-yl}ethyl)pyrrolidin-2-one
N-[(8-methyl-2-{octahydropyrrolo[1,2-a]piperazin-2-yl}quinolin-3-yl)methyl]cyclopropanamine
N-[(3R,4R)-3-hydroxy-1-(4,4,4-trifluorobutanoyl)piperidin-4-yl]pyrazine-2-carboxamide
1-methyl-N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-1H-indole-6-carboxamide
6-(6-{[2-(dimethylamino)ethyl]amino}-1H-pyrrolo[2,3-b]pyridin-4-yl)-1,2,3,4-tetrahydroquinazoline-2,4-dione
N-(pyridin-4-yl)spiro[2.4]heptane-1-carboxamide
4-hydroxy-N-methyl-2-(2-methyl-1,3-thiazol-4-yl)-N-[1-(1,2-oxazol-3-yl)ethyl]pyrimidine-5-carboxamide
1-cyclopentyl-3-(4-methoxyphenyl)-3-{2-oxo-2-[4-(pyridin-3-yloxy)piperidin-1-yl]ethyl}pyrrolidine-2,5-dione
N-(1,4-dioxan-2-ylmethyl)-N-methyl-2-[2-oxo-3-(trifluoromethyl)-1,2-dihydropyridin-1-yl]acetamide
1-[3-(pyridin-2-yl)propanoyl]-N-[4-(1,3-thiazol-4-yl)phenyl]piperidine-3-carboxamide
methyl 1-[(3R,5S)-1-[(3-fluorophenyl)methyl]-5-{[3-(methylsulfanyl)phenyl]carbamoyl}pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
5-[3-(4-methylphenyl)propanoyl]-1-(2-methylpropyl)-N-(pyridin-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide