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3-fluoro-N-methyl-N-[(4-phenyl-1,3-thiazol-2-yl)methyl]imidazo[1,2-a]pyridine-2-carboxamide
N-[(3S)-2-oxoazepan-3-yl]-2-[(prop-2-en-1-yl)amino]benzamide
1-{1-[3-(2H-1,3-benzodioxol-5-yl)-2-methylpropyl]piperidin-4-yl}-N-cyclopropyl-1H-1,2,3-triazole-4-carboxamide
4-(hydroxymethyl)-1-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}azepan-4-ol
N-{[5-(2-methoxyethyl)-1,2,4-oxadiazol-3-yl]methyl}imidazo[2,1-b][1,3]thiazole-6-carboxamide
(3-chlorophenyl)(1-cyclohexyl-1H-1,2,4-triazol-5-yl)methanol
1-(2-methoxyphenyl)-N-methyl-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H-pyrazole-4-carboxamide
9-(4,6-dimethoxypyrimidin-2-yl)-1-oxa-9-azaspiro[5.5]undecan-5-ol
4-[(3R,4R)-4-(azepan-1-yl)-3-hydroxypiperidine-1-carbonyl]-1,2-dihydroquinolin-2-one
7-{[4-(propan-2-yl)phenyl]methyl}-2-(pyridine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
7-[2-(1,1,2,2-tetrafluoroethoxy)benzoyl]-2,7-diazaspiro[4.4]nonane-1,3-dione
N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-3-hydroxy-4-methylbenzamide
1-{2-[2-methyl-4-(2-methylphenyl)-5-oxopiperazin-1-yl]-2-oxoethyl}azepan-2-one
(5S,9aS,9bS)-2-cyclopentyl-5-[4-(pyrimidin-2-yloxy)phenyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-[3-(dimethylamino)benzoyl]-3-methylpiperidine-3-carbonitrile
2-(dimethylamino)-1-{2-[2-(pyridin-2-yl)ethyl]piperidin-1-yl}ethan-1-one
1-[(3-chloro-5-fluoro-4-methoxyphenyl)methyl]-3-ethylpiperidine-3-carboxylic acid
(2S,4S)-4-amino-1-[(4-methyl-3,4-dihydro-2H-1,4-benzoxazin-7-yl)sulfonyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
8-chloro-6-{2-[4-(3-hydroxyprop-1-yn-1-yl)phenyl]-1H-imidazol-1-yl}-3,4-dihydro-2H-1,4-benzoxazin-3-one
1-(2-methylbutyl)-4-[4-(2-methylpropyl)-1H-1,2,3-triazol-1-yl]piperidine
N-(1-carbamoylcyclohexyl)-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
1-{[(3R,4R)-1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}piperidin-4-ol
N,N-dimethyl-1-(3-phenoxybenzoyl)azepan-4-amine
3-ethyl-N-[(5-methylthiophen-2-yl)methyl]-N-(pyridin-4-ylmethyl)-1H-pyrazole-5-carboxamide
(4aS,7aR)-1-(3,5-dimethylbenzoyl)-4-(3-methylbutanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]ethyl}-5-(2-methylphenyl)-1,2,4-triazin-3-amine
2-(3-fluoro-4-methoxyphenyl)-2-[4-(1H-pyrazol-1-ylmethyl)piperidin-1-yl]acetic acid
{3-[(4-fluorophenyl)methyl]-1-[(5-methylthiophen-2-yl)methyl]piperidin-3-yl}methanol
2-(2,4-difluorophenoxy)-N-[1-(pyrazin-2-yl)propan-2-yl]acetamide
N,N-dimethyl-5-({methyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amino}methyl)pyridin-2-amine
2-[(4-methoxyphenyl)methyl]-4-{[3-(1H-pyrazol-1-yl)phenyl]methyl}morpholine
2-cyano-N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)benzamide
1-methyl-5-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}piperidin-2-one
N-(2-methoxy-5-methylphenyl)-2-({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}amino)acetamide
(5S,9aS,9bS)-5-(3-hydroxy-4-methoxyphenyl)-2-[(2-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-(3-oxo-3-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propyl)pyrrolidin-2-one
N-[1-(3-fluoro-4-methoxyphenyl)ethyl]-4-methyl-3-(2-oxoimidazolidin-1-yl)benzamide
N4-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]-5-ethylpyrimidine-2,4-diamine
1-[6-methyl-3-({methyl[(3-methyl-1,2-oxazol-5-yl)methyl]amino}methyl)quinolin-2-yl]piperidin-3-ol
(3R,4R)-3-methyl-4-(oxan-4-yl)-1-(5-propylpyrimidin-4-yl)piperidin-4-ol
2-{1-[2-(1H-pyrazol-1-yl)benzoyl]azetidin-3-yl}pyridine
4-(ethanesulfonyl)-2-(4H-1,2,4-triazol-4-yl)phenol
3-[1-methyl-5-(1-phenyl-1H-pyrazol-4-yl)-1H,4H-pyrazolo[3,4-d]imidazol-3-yl]pyridine
(3aR,6aR)-2-(6-methylpyridine-2-carbonyl)-5-(oxan-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
9-{[3-(2-aminoethyl)phenyl]methyl}-2-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-(diethylamino)-3-{5-[(4,4-dimethylpiperidin-1-yl)methyl]-2-methoxyphenoxy}propan-2-ol
2-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyrazine
N-{[3-(benzyloxy)phenyl]methyl}-1,9-dioxaspiro[5.5]undecan-4-amine
4-(3-fluorophenyl)-N-{[4-(2-methylpropoxy)phenyl]methyl}-N-(pyridin-4-ylmethyl)benzamide
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)pyrrolidine-1-carboxamide