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({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)(methyl)[(2,4,6-trimethoxyphenyl)methyl]amine
4-{2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]-2-oxoethyl}-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one
(4aS,7aR)-1-(1H-indol-5-ylmethyl)-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[2-(2-methyl-1,3-thiazol-4-yl)ethyl]-3-[3-(trifluoromethyl)benzoyl]piperidine
(3R,4R)-1-(4-aminopyrimidin-2-yl)-4-(4-hydroxypiperidin-1-yl)piperidin-3-ol
N-cyclobutyl-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
N-(butan-2-yl)-6-methyl-5-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridine-2-carboxamide
4-{[1-(3-fluoro-2-methoxybenzoyl)pyrrolidin-3-yl]methyl}benzoic acid
3-(3-methyl-1,2,4-thiadiazol-5-yl)-1-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}urea
3-{[1-(oxane-4-carbonyl)pyrrolidin-3-yl]methyl}benzamide
({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)(methyl)(2-phenylethyl)amine
N-methyl-5-[1-(piperidin-1-yl)ethyl]-N-[(trimethyl-1H-pyrazol-4-yl)methyl]furan-2-carboxamide
2-(dimethylamino)-N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-(3-methylphenyl)acetamide
N-[3-(5-sulfamoylthiophen-2-yl)phenyl]acetamide
(3S,4R)-1-(oxan-4-yl)-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
(3R,4R)-1-{[5-(1,5-dimethyl-1H-pyrrol-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-4-(hydroxymethyl)piperidin-3-ol
N-{2-[(4-chlorophenyl)sulfanyl]ethyl}-N-(2-hydroxyethyl)-2-(2-oxopyrrolidin-1-yl)acetamide
1-{[3-(difluoromethoxy)phenyl]methyl}-3-(dimethyl-1H-1,2,4-triazol-3-yl)urea
1-(furan-2-carbonyl)-4-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-1,4-diazepane
8-[(3-ethyl-1,2-oxazol-5-yl)methyl]-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1,5-dimethyl-3-{[4-(3-methylthiophen-2-yl)-1H-1,2,3-triazol-1-yl]methyl}-1H-indazole
4-{3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}pyrimidin-2-amine
N-(2-acetamidophenyl)-2-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]acetamide
8-[2-(3-methyl-6-oxo-1,6-dihydropyridazin-1-yl)acetyl]-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-{1-[(4-methoxyphenyl)methyl]piperidin-4-yl}-4-(pyrrolidine-1-carbonyl)piperidine
3-{2-[(4S)-4-hydroxy-4-(methoxymethyl)-3,3-dimethylpiperidin-1-yl]-2-oxoethyl}-5,5-dimethylimidazolidine-2,4-dione
3-[3-methoxy-5-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-1-methyl-1-[2-(oxan-2-yl)ethyl]urea
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-[(1-propyl-1H-imidazol-2-yl)methyl]piperidin-3-ol
2-({[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}(thiophen-3-ylmethyl)amino)butan-1-ol
1-(2-{[(2,3,5-trimethyl-1H-indol-7-yl)methyl]amino}pyrimidin-4-yl)piperidin-3-ol
2-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-4-[4-(5-methylthiophene-2-carbonyl)piperazin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
N-(2,3-dihydro-1H-inden-2-yl)-N-methyl-4-oxo-4H-chromene-2-carboxamide
N-{1-[7-(cyclohexylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}-3-phenylpropanamide
(4aS,8aR)-1-[2-(1H-imidazol-4-yl)ethyl]-6-(pyridine-4-carbonyl)-decahydro-1,6-naphthyridin-2-one
4-[(3-{[4-(pyridin-4-yl)piperazin-1-yl]methyl}phenyl)methyl]morpholine
1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-N,5-dimethyl-N-(2-methylpropyl)-1H-pyrazole-4-carboxamide
1-{[5-(oxan-2-yl)furan-2-yl]methyl}-N-[3-(1H-pyrazol-5-yl)phenyl]piperidine-4-carboxamide
4-(naphthalen-2-yloxy)-1-(1,3-thiazol-2-yl)piperidine-4-carboxylic acid
1-[(2R,3R,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-ethoxypropan-1-one
3-(2-ethyl-1H-imidazol-1-yl)-1-{3-[2-(pyridin-4-yl)pyridin-4-yl]pyrrolidin-1-yl}propan-1-one
5-{[2,5-dimethoxy-4-(methylsulfanyl)phenyl]methyl}-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
(3S,4R)-4-phenyl-1-{[2-(thiophen-2-yl)pyrimidin-5-yl]methyl}pyrrolidine-3-carboxylic acid
N5-cyclooctyl-N3-(2-methoxyethyl)-4-oxo-N3-(propan-2-yl)-1-(pyridin-2-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
1-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)-1H-1,2,4-triazole
2,6-dimethyl-4-({[1-(pyrazin-2-yl)propan-2-yl]amino}methyl)phenyl acetate
(3S,9aR)-3-[(benzyloxy)methyl]-8-(3-methylbenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
methyl (2S)-2-{[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]amino}propanoate
N-[(2R,3R)-1'-(2,3-dihydro-1-benzofuran-5-ylmethyl)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(thiophen-2-yl)acetamide
N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzamide
methyl 2-[(4-chloro-2-propanamidophenyl)formamido]-2-methylpropanoate