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ethyl 4-{[3-(oxolan-3-yl)propyl]amino}piperidine-1-carboxylate
4-[3-(2-chlorophenoxy)azetidine-1-carbonyl]-1-oxaspiro[4.5]decan-2-one
[(3R,4R)-1-(5-amino-4-chloro-1H-pyrazole-3-carbonyl)-4-(azepan-1-ylmethyl)pyrrolidin-3-yl]methanol
ethyl 1-[4-(1H-1,2,4-triazol-1-yl)phenyl]-1H-imidazole-2-carboxylate
1-[(2-phenyl-1H-imidazol-4-yl)methyl]-4-[(2E)-3-phenylprop-2-en-1-yl]piperazine
N-[(2,4-dimethoxyphenyl)methyl]-3-(1-propanoylpiperidin-3-yl)propanamide
(1S,5R)-6-{[2-(furan-2-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-1,3,3-trimethyl-6-azabicyclo[3.2.1]octane
N-(1-carbamoylcyclopentyl)-4-(3-hydroxy-3-methylbutyl)benzamide
2-cyclopentyl-8-[5-(propan-2-yl)pyrimidin-4-yl]-2,8-diazaspiro[5.5]undecan-3-one
1-{4-[(2-propoxypropyl)amino]piperidin-1-yl}ethan-1-one
{[3-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amine
methyl 3-(2-chloro-6-fluorobenzamido)-6-{[methyl(1,2-oxazol-3-ylmethyl)amino]methyl}thieno[2,3-b]pyridine-2-carboxylate
(1s,4s)-4-{4-[3-methyl-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]-1H-1,2,3-triazol-1-yl}cyclohexan-1-amine
2-methoxy-1-[3-(4-methoxyphenoxymethyl)piperidin-1-yl]ethan-1-one
(3S,4S)-1-[1-(furan-2-ylmethyl)piperidine-4-carbonyl]-4-(morpholin-4-yl)pyrrolidin-3-ol
6-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
N-[(3-fluorophenyl)methyl]-2-[(3S)-3-hydroxypyrrolidin-1-yl]-1-methyl-1H-1,3-benzodiazole-5-carboxamide
4-[3-(1H-pyrazol-1-yl)phenyl]-1H-pyrazolo[3,4-d]pyrimidin-6-amine
11-{[(3-chlorophenyl)methyl]amino}-4-(pyridin-2-ylmethyl)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
4-[2-amino-3-cyano-6-(furan-2-ylmethyl)-5,6,7,8-tetrahydro-1,6-naphthyridin-4-yl]benzoic acid
1-[1-(4,6-dimethylpyrimidin-2-yl)piperidin-4-yl]-4-phenylpiperidine-4-carbonitrile
ethyl 1-[2-(2-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]piperidine-4-carboxylate
2-(3-chloro-6-oxo-1,6-dihydropyridazin-1-yl)-N-methyl-N-[1-(2-phenylethyl)piperidin-3-yl]acetamide
1-(1-ethyl-1H-pyrazole-5-carbonyl)-3-(3-methoxypropyl)piperidine
1-[(3,4-dimethylphenyl)methyl]-4-(3-hydroxy-2-methylbenzoyl)piperazin-2-one
6-tert-butyl-2-(3-{1,4-diazabicyclo[3.2.2]nonan-4-ylmethyl}phenyl)-3,4-dihydropyrimidin-4-one
1-(1-methyl-4-phenylpiperidine-4-carbonyl)-4-(3-methylpyridin-2-yl)piperazine
2-{4-[3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidine-1-carbonyl]phenoxy}acetamide
5-[(2-methyl-1,3-thiazol-4-yl)methyl]-1-[4-(trifluoromethyl)phenyl]-1H-1,2,4-triazole
N-[(5-cyclopropyl-1,2-oxazol-3-yl)methyl]-N-methyl-5-propyl-1,3,4-oxadiazol-2-amine
1-[(4-methylphenyl)methyl]-4-{2-oxo-1-oxaspiro[4.4]nonane-4-carbonyl}piperazin-2-one
({5-[1-(3,5-difluorobenzoyl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
N-(3-{[(2-fluorophenyl)methyl]sulfanyl}propyl)-2-oxo-1-oxaspiro[4.4]nonane-4-carboxamide
5-methyl-1-(4-methylphenyl)-4-(2-methylpyrimidine-5-carbonyl)piperazin-2-one
N-[4-(3-acetylphenyl)phenyl]-4-(2-methoxyethyl)piperazine-1-carboxamide
1-[5-(4-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]-4-methylpiperazine
4-[(2-methylphenyl)sulfanyl]-1-(oxane-4-carbonyl)piperidine
3-{[(3S,4S)-3-hydroxy-4-(3-methoxyphenyl)piperidin-1-yl]methyl}-1-methyl-1,2-dihydroquinolin-2-one
2-(pyridin-4-yl)-4-(pyrrolidine-1-carbonyl)pyridine
N-{[4-(2-methylpropoxy)phenyl]methyl}-N-(pyridin-4-ylmethyl)thiophene-2-carboxamide
2-fluoro-6-[2-(4-fluorophenoxy)ethyl]benzamide
4-[1-(furan-2-ylmethyl)piperidine-3-carbonyl]-1,4-oxazepane
9-[(3-chloro-2,4-difluorophenyl)methyl]-2-methyl-2,9-diazaspiro[5.5]undecan-3-one
N-[4-(3-methoxyphenyl)phenyl]-1-(3-methyl-1H-pyrazole-4-carbonyl)piperidine-3-carboxamide
7-cyclopentanecarbonyl-N,N-dimethyl-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
5-[1-butyl-3-(1H-indol-3-yl)-1H-1,2,4-triazol-5-yl]-1-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
8-(2-ethylpyrimidine-5-carbonyl)-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-4-(thiophen-2-ylmethyl)-1,4-diazepane
2-({4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]piperidin-1-yl}methyl)pyridine
3-ethyl-2-{4-[2-(methylsulfanyl)ethyl]piperazine-1-carbonyl}-1H-indole