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7-(6-methoxypyrimidin-4-yl)-2-methyl-2,7-diazaspiro[4.5]decane
N-[(2-fluorophenyl)methyl]-N-(2-hydroxyethyl)-3,4,7-trimethyl-1H-indole-2-carboxamide
1-[2-(dimethylamino)ethyl]-5-oxo-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}pyrrolidine-3-carboxamide
1-{2-[(3R,4R)-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidin-1-yl]-2-oxoethyl}-1,2-dihydropyridin-2-one
4-[(4-fluorophenyl)methyl]-1-(1-methyl-1H-imidazole-5-carbonyl)-3-(propan-2-yl)-1,4-diazepan-5-one
4-(3-ethoxypropanoyl)-1-[(3-methoxyphenyl)methyl]piperazin-2-one
1-methyl-3-(propan-2-yl)-N-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}-1H-pyrazole-5-carboxamide
4-(cyclopropylmethyl)-3-(propan-2-yl)-1-(4-propylpyrimidine-5-carbonyl)-1,4-diazepan-5-one
N-[2-(azepan-1-yl)ethyl]-N-ethyl-5-(oxolan-2-yl)thiophene-2-carboxamide
(1R,2S)-1-(4-pentyl-1H-1,2,3-triazol-1-yl)-2,3-dihydro-1H-inden-2-ol
4-{[5-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]methyl}piperazine-1-sulfonamide
N-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-3-(trimethyl-1H-pyrazol-4-yl)propanamide
(3S,4R)-3-methoxy-1-{[4-methoxy-3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}piperidin-4-amine
4-(4-methylphenyl)-5-(pyridin-4-yl)-2-(pyrrolidin-1-yl)pyrimidine
(3R)-3-[1-benzyl-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-5-yl]-1,2,3,4-tetrahydroisoquinoline
3-[({1-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]piperidin-3-yl}oxy)methyl]pyridine
dimethyl[(4-methyl-5-{1-[(4-phenyl-1,3-thiazol-2-yl)methyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]amine
N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
4-ethyl-1-methyl-3-{1-[(3-methyl-1-benzofuran-2-yl)methyl]piperidin-3-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
2-{2-methyl-2,7-diazaspiro[4.5]decane-7-carbonyl}thiophene-3-sulfonamide
N-[3-(4-{[3-(2H-1,3-benzodioxol-5-yl)propanamido]methyl}-5-methyl-1,3-oxazol-2-yl)phenyl]-3-methylbutanamide
(3R,4R)-1-(cyclohexylmethyl)-4-(4-hydroxypiperidin-1-yl)piperidin-3-ol
1-methyl-4-{[1-(2-methylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1H-pyrazole
(3aS,7aR)-5-methyl-2-(4,5,6,7-tetrahydro-1-benzothiophene-2-carbonyl)-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
(3S,4R)-1-(4-carboxybenzoyl)-4-(3-methoxyphenyl)pyrrolidine-3-carboxylic acid
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1-[3-(1H-pyrazol-5-yl)phenyl]piperidin-4-amine
N-[cyclohexyl(thiophen-2-yl)methyl]-2-(methylamino)acetamide
1-(1-benzyl-4-phenylpiperidine-4-carbonyl)piperazine
2-[(1S,4S)-5-(2-methoxy-5-phenylphenyl)-6-oxo-2,5-diazabicyclo[2.2.1]heptan-2-yl]-N-methylacetamide
N-[3-(5-amino-1,3,4-thiadiazol-2-yl)propyl]-2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamide
1-[(2-methoxypyrimidin-5-yl)methyl]-4-[(3-phenyl-1,2-oxazol-5-yl)methyl]piperidin-4-ol
N-[5-(1-methyl-1H-pyrazol-4-yl)pyridin-2-yl]cyclopropanecarboxamide
N3-cyclooctyl-N5-cyclopropyl-4-oxo-1-(oxolan-2-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
(5-{[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}furan-2-yl)methanol
2-(2H-1,3-benzodioxol-5-yl)-1-[6-(hydroxymethyl)-1,4-oxazepan-4-yl]ethan-1-one
N-[4-(2-methyl-5-oxopyrrolidin-1-yl)phenyl]-4-(pyridin-4-yl)piperazine-1-carboxamide
2-(3-methylbut-2-en-1-yl)-8-[2-(pyridin-2-yl)acetyl]-2,8-diazaspiro[4.5]decan-3-one
N-{2-[7-(cyclohexylmethyl)-2,7-diazaspiro[4.5]decan-2-yl]-2-oxoethyl}acetamide
2-(diethylamino)-1-{3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl}ethan-1-one
N-[(2,5-dichlorophenyl)methyl]-1-ethyl-6-methyl-2-oxo-1,2-dihydropyridine-3-carboxamide
9-(5-ethyl-2-methylpyrimidin-4-yl)-1,4-dimethyl-1,4,9-triazaspiro[5.5]undecane
N-(1-{1-[4-(ethylamino)pyrimidin-2-yl]piperidin-4-yl}-1H-pyrazol-5-yl)cyclopropanecarboxamide
3-{[3-(5-fluoro-2-methoxybenzoyl)piperidin-1-yl]methyl}-1-methyl-1H-indole
1,3-dimethyl-4-[2-(1-methyl-1H-indol-3-yl)acetyl]piperazin-2-one
1-(3,5-difluoropyridine-2-carbonyl)-4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine
2-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3-oxopiperazin-2-yl}-N-[(1-methyl-2,3-dihydro-1H-indol-5-yl)methyl]acetamide
6-(2-aminoethyl)-2-methyl-N-[2-(pyridin-2-yl)ethyl]pyrimidin-4-amine
(1R,3S)-7-[(dimethyl-1,3-thiazol-2-yl)methyl]-3-(2-hydroxyethoxy)-7-azaspiro[3.5]nonan-1-ol
2-(4-ethoxyphenyl)-4-{[2-(2-methoxyphenyl)pyrrolidin-1-yl]methyl}-5-methyl-1,3-oxazole